DE60006026D1 - Verfahren zur Herstellung von 8-cyclopentyl-6-ethyl-3 (substituierten)-5,8-dihydro-4H-1,2,3A,7,8-penta aza-as-Indacenen und dafür geeigneter Zwischenprodukte - Google Patents

Verfahren zur Herstellung von 8-cyclopentyl-6-ethyl-3 (substituierten)-5,8-dihydro-4H-1,2,3A,7,8-penta aza-as-Indacenen und dafür geeigneter Zwischenprodukte

Info

Publication number: DE60006026D1
Authority: DE; Germany
Prior art keywords: indacenes; cyclopentyl; dihydro; ethyl; substituted
Prior art date: 1999-04-30
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Application number

DE60006026T

Other languages

English (en)

Other versions

DE60006026T2 (de

Inventor

Frank John Urban

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Products Inc

Original Assignee

Pfizer Products Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-04-30

Filing date

2000-04-07

Publication date

2003-11-27

2000-04-07 Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc

2003-11-27 Application granted granted Critical

2003-11-27 Publication of DE60006026D1 publication Critical patent/DE60006026D1/de

2004-06-17 Publication of DE60006026T2 publication Critical patent/DE60006026T2/de

2020-04-08 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Pulmonology (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Hydrogenated Pyridines (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

DE60006026T 1999-04-30 2000-04-07 Verfahren zur Herstellung von 8-cyclopentyl-6-ethyl-3 (substituierten)-5,8-dihydro-4H-1,2,3A,7,8-penta aza-as-Indacenen und dafür geeigneter Zwischenprodukte Expired - Fee Related DE60006026T2 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US13194999P	1999-04-30	1999-04-30
US131949P		1999-04-30

Publications (2)

Publication Number	Publication Date
DE60006026D1 true DE60006026D1 (de)	2003-11-27
DE60006026T2 DE60006026T2 (de)	2004-06-17

Family

ID=22451736

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DE60006026T Expired - Fee Related DE60006026T2 (de)	1999-04-30	2000-04-07	Verfahren zur Herstellung von 8-cyclopentyl-6-ethyl-3 (substituierten)-5,8-dihydro-4H-1,2,3A,7,8-penta aza-as-Indacenen und dafür geeigneter Zwischenprodukte
DE60015819T Expired - Fee Related DE60015819T2 (de)	1999-04-30	2000-04-07	Pyrazolopyridinon als Zwischenprodukt

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
DE60015819T Expired - Fee Related DE60015819T2 (de)	1999-04-30	2000-04-07	Pyrazolopyridinon als Zwischenprodukt

Country Status (24)

Country	Link
US (1)	US6326495B2 (de)
EP (1)	EP1048667B1 (de)
JP (1)	JP3510560B2 (de)
KR (1)	KR100346619B1 (de)
CN (2)	CN1160353C (de)
AR (1)	AR029450A1 (de)
AT (2)	ATE282039T1 (de)
AU (1)	AU761391B2 (de)
BR (1)	BR0002070A (de)
CA (1)	CA2307080C (de)
DE (2)	DE60006026T2 (de)
DK (2)	DK1048667T3 (de)
ES (2)	ES2232805T3 (de)
HU (1)	HUP0001700A3 (de)
ID (1)	ID25705A (de)
IL (1)	IL135809A0 (de)
IN (1)	IN192746B (de)
MX (1)	MXPA00004214A (de)
PL (1)	PL339985A1 (de)
PT (2)	PT1380585E (de)
RU (1)	RU2189985C2 (de)
TR (1)	TR200001161A2 (de)
TW (1)	TWI256392B (de)
ZA (1)	ZA200002057B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MY148239A (en)	2009-08-13	2013-03-29	China Petroleum & Chemical	A catalyst component for olefin polymerization and a catalyst comprising the same
BR112013005689A2 (pt)	2010-09-08	2016-05-03	Sumitomo Chemical Co	método para produção de compostos de piridazinona e intermediário dos mesmos

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SU1094303A1 (ru) *	1982-12-24	1987-12-30	Институт физико-органической химии и углехимии АН УССР	3-Трифторметил-7-метилимидазо- @ 4,5-с @ -1,2,4-триазоло @ 4,3-а @ пиридин,обладающий спазмолитическим действием
US4940715A (en) *	1988-05-17	1990-07-10	Kissei Pharmaceutical Co., Ltd.	5H-pyrazolo[4,3-A] quinolizin-5-one compounds exhibiting therapeutic activities
NZ266525A (en)	1993-07-06	1997-10-24	Pfizer	4,5,6,7-tetrahydro-1h-pyrazolo[3,4-c]pyridine derivatives and medicaments
KR970707124A (ko)	1994-10-20	1997-12-01	스피겔 알렌 제이	비사이클릭 테트라하이드로 피라졸로피리딘 및 약제로서 이의 용도(bicyclic tetrahydro pyrazolopyridines and their use as medicaments)
JP3107827B2 (ja)	1995-06-06	2000-11-13	ファイザー・インコーポレーテッド	トリサイクリック５，６−ジヒドロ−９Ｈ−ピラゾロ［３，４−ｃ］−１，２，４−トリアゾロ［４，３−ａ］ピリジン類

2000
- 2000-03-01 US US09/516,549 patent/US6326495B2/en not_active Expired - Fee Related
- 2000-04-07 DE DE60006026T patent/DE60006026T2/de not_active Expired - Fee Related
- 2000-04-07 AT AT03024166T patent/ATE282039T1/de not_active IP Right Cessation
- 2000-04-07 ES ES03024166T patent/ES2232805T3/es not_active Expired - Lifetime
- 2000-04-07 DE DE60015819T patent/DE60015819T2/de not_active Expired - Fee Related
- 2000-04-07 AT AT00302947T patent/ATE252582T1/de not_active IP Right Cessation
- 2000-04-07 PT PT03024166T patent/PT1380585E/pt unknown
- 2000-04-07 DK DK00302947T patent/DK1048667T3/da active
- 2000-04-07 PT PT00302947T patent/PT1048667E/pt unknown
- 2000-04-07 DK DK03024166T patent/DK1380585T3/da active
- 2000-04-07 EP EP00302947A patent/EP1048667B1/de not_active Expired - Lifetime
- 2000-04-07 ES ES00302947T patent/ES2207464T3/es not_active Expired - Lifetime
- 2000-04-24 IN IN447DE2000 patent/IN192746B/en unknown
- 2000-04-24 IL IL13580900A patent/IL135809A0/xx unknown
- 2000-04-25 TW TW089107724A patent/TWI256392B/zh not_active IP Right Cessation
- 2000-04-26 JP JP2000125351A patent/JP3510560B2/ja not_active Expired - Fee Related
- 2000-04-26 ZA ZA200002057A patent/ZA200002057B/xx unknown
- 2000-04-27 TR TR2000/01161A patent/TR200001161A2/xx unknown
- 2000-04-27 AR ARP000102007A patent/AR029450A1/es unknown
- 2000-04-28 AU AU30180/00A patent/AU761391B2/en not_active Ceased
- 2000-04-28 CN CNB001081403A patent/CN1160353C/zh not_active Expired - Fee Related
- 2000-04-28 MX MXPA00004214A patent/MXPA00004214A/es active IP Right Grant
- 2000-04-28 HU HU0001700A patent/HUP0001700A3/hu unknown
- 2000-04-28 RU RU2000111018/04A patent/RU2189985C2/ru not_active IP Right Cessation
- 2000-04-28 ID IDP20000356D patent/ID25705A/id unknown
- 2000-04-28 CA CA002307080A patent/CA2307080C/en not_active Expired - Fee Related
- 2000-04-28 CN CNB031476457A patent/CN1249064C/zh not_active Expired - Fee Related
- 2000-04-29 KR KR1020000023025A patent/KR100346619B1/ko not_active Expired - Fee Related
- 2000-04-30 PL PL00339985A patent/PL339985A1/xx not_active Application Discontinuation
- 2000-05-02 BR BR0002070-2A patent/BR0002070A/pt not_active IP Right Cessation

Also Published As

Publication number	Publication date
KR20010029673A (ko)	2001-04-06
DE60015819T2 (de)	2005-12-08
EP1048667A1 (de)	2000-11-02
HK1031881A1 (en)	2001-06-29
ATE252582T1 (de)	2003-11-15
HUP0001700A3 (en)	2001-05-28
CN1249064C (zh)	2006-04-05
ID25705A (id)	2000-11-02
ATE282039T1 (de)	2004-11-15
TWI256392B (en)	2006-06-11
TR200001161A2 (tr)	2000-12-21
RU2189985C2 (ru)	2002-09-27
CN1478779A (zh)	2004-03-03
DE60006026T2 (de)	2004-06-17
AU3018000A (en)	2000-11-02
MXPA00004214A (es)	2002-03-08
DE60015819D1 (de)	2004-12-16
EP1048667B1 (de)	2003-10-22
AU761391B2 (en)	2003-06-05
PT1048667E (pt)	2004-03-31
IN192746B (de)	2004-05-15
HK1062678A1 (zh)	2004-11-19
JP3510560B2 (ja)	2004-03-29
PL339985A1 (en)	2000-11-06
CA2307080C (en)	2003-12-23
BR0002070A (pt)	2000-10-31
HUP0001700A2 (en)	2001-03-28
ZA200002057B (en)	2001-10-26
DK1048667T3 (da)	2004-03-01
PT1380585E (pt)	2005-03-31
ES2232805T3 (es)	2005-06-01
CN1274724A (zh)	2000-11-29
US20010039347A1 (en)	2001-11-08
AR029450A1 (es)	2003-07-02
ES2207464T3 (es)	2004-06-01
DK1380585T3 (da)	2005-03-07
JP2000344771A (ja)	2000-12-12
KR100346619B1 (ko)	2002-07-26
US6326495B2 (en)	2001-12-04
HU0001700D0 (en)	2000-07-28
CN1160353C (zh)	2004-08-04
IL135809A0 (en)	2001-05-20
CA2307080A1 (en)	2000-10-30

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Legal Events

Date	Code	Title	Description
2004-11-18	8364	No opposition during term of opposition
2008-02-14	8339	Ceased/non-payment of the annual fee