PL372724A1 - (S)-4-amino-5-chloro-2-metoksy-N-[1-[1-(2-tetrahydrofurylokarbonylo)-4-piperydynylometylo]-4-piperydynylo] benzamid, sposób jego wytwarzania, zawierająca go kompozycja farmaceutyczna oraz jego związek pośredni - Google Patents
(S)-4-amino-5-chloro-2-metoksy-N-[1-[1-(2-tetrahydrofurylokarbonylo)-4-piperydynylometylo]-4-piperydynylo] benzamid, sposób jego wytwarzania, zawierająca go kompozycja farmaceutyczna oraz jego związek pośredniInfo
- Publication number
- PL372724A1 PL372724A1 PL03372724A PL37272403A PL372724A1 PL 372724 A1 PL372724 A1 PL 372724A1 PL 03372724 A PL03372724 A PL 03372724A PL 37272403 A PL37272403 A PL 37272403A PL 372724 A1 PL372724 A1 PL 372724A1
- Authority
- PL
- Poland
- Prior art keywords
- tetrahydrofurylcarbonyl
- piperidinylmethyl
- benzamide
- piperidinyl
- chloro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2002141262 | 2002-05-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
PL372724A1 true PL372724A1 (pl) | 2005-07-25 |
Family
ID=29267809
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL03372724A PL372724A1 (pl) | 2002-05-16 | 2003-05-15 | (S)-4-amino-5-chloro-2-metoksy-N-[1-[1-(2-tetrahydrofurylokarbonylo)-4-piperydynylometylo]-4-piperydynylo] benzamid, sposób jego wytwarzania, zawierająca go kompozycja farmaceutyczna oraz jego związek pośredni |
Country Status (27)
Country | Link |
---|---|
US (1) | US6696468B2 (pl) |
EP (1) | EP1362857B1 (pl) |
JP (1) | JP3643107B2 (pl) |
KR (1) | KR20040107520A (pl) |
CN (1) | CN1653063A (pl) |
AR (1) | AR040021A1 (pl) |
AT (1) | ATE273304T1 (pl) |
AU (1) | AU2003230245A1 (pl) |
BR (1) | BR0309933A (pl) |
CA (1) | CA2483368A1 (pl) |
CZ (1) | CZ20041084A3 (pl) |
DE (1) | DE60300021T2 (pl) |
DK (1) | DK1362857T3 (pl) |
ES (1) | ES2227500T3 (pl) |
HK (1) | HK1060118A1 (pl) |
HU (1) | HUP0501016A2 (pl) |
IL (1) | IL165012A0 (pl) |
MX (1) | MXPA04011332A (pl) |
NO (1) | NO20045469L (pl) |
PL (1) | PL372724A1 (pl) |
PT (1) | PT1362857E (pl) |
RU (1) | RU2004136853A (pl) |
SK (1) | SK50192004A3 (pl) |
TR (1) | TR200403020T2 (pl) |
TW (1) | TW200400186A (pl) |
WO (1) | WO2003097638A1 (pl) |
ZA (1) | ZA200409053B (pl) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE9904377D0 (sv) * | 1999-12-01 | 1999-12-01 | Astra Pharma Prod | Pharmaceutical combinations |
SE0200843D0 (sv) | 2002-03-19 | 2002-03-19 | Astrazeneca Ab | Chemical compounds |
SE0200844D0 (sv) | 2002-03-19 | 2002-03-19 | Astrazeneca Ab | Chemical compounds |
SE0300957D0 (sv) | 2003-04-01 | 2003-04-01 | Astrazeneca Ab | Chemical compounds |
TW200533348A (en) * | 2004-02-18 | 2005-10-16 | Theravance Inc | Indazole-carboxamide compounds as 5-ht4 receptor agonists |
TWI351282B (en) | 2004-04-07 | 2011-11-01 | Theravance Inc | Quinolinone-carboxamide compounds as 5-ht4 recepto |
US8309575B2 (en) | 2004-04-07 | 2012-11-13 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
US7728006B2 (en) * | 2004-04-07 | 2010-06-01 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
DE602005014566D1 (de) * | 2004-11-05 | 2009-07-02 | Theravance Inc | Chinolinon-carboxamid-verbindungen |
JP5086091B2 (ja) * | 2004-11-05 | 2012-11-28 | セラヴァンス, インコーポレーテッド | 5−ht4受容体アゴニスト化合物 |
AU2005319190A1 (en) * | 2004-12-22 | 2006-06-29 | Theravance, Inc. | Indazole-carboxamide compounds |
EA013567B1 (ru) * | 2005-03-02 | 2010-06-30 | Тереванс, Инк. | Хинолиноновые соединения в качестве агонистов рецептора 5-ht |
US7256294B2 (en) * | 2005-05-25 | 2007-08-14 | Theravance, Inc. | Crystalline form of a benzimidazole-carboxamide medicinal compound |
MY147756A (en) | 2005-05-25 | 2013-01-15 | Theravance Inc | Benzimidazole-carboxamide compounds as 5-ht4 receptor agonists |
TW200722419A (en) * | 2005-05-27 | 2007-06-16 | Astrazeneca Ab | Chemical compounds |
WO2006126948A1 (en) * | 2005-05-27 | 2006-11-30 | Astrazeneca Ab | Piperidines for the treatment of chemokine mediated diseases |
US8314127B2 (en) | 2005-07-21 | 2012-11-20 | Astrazeneca Ab | Piperidine derivatives |
GB0525068D0 (en) | 2005-12-08 | 2006-01-18 | Novartis Ag | Organic compounds |
TWI423967B (zh) * | 2008-02-21 | 2014-01-21 | Dainippon Sumitomo Pharma Co | 醯胺衍生物及含有其之醫藥組合物 |
US8349852B2 (en) | 2009-01-13 | 2013-01-08 | Novartis Ag | Quinazolinone derivatives useful as vanilloid antagonists |
AR080056A1 (es) | 2010-02-01 | 2012-03-07 | Novartis Ag | Derivados de ciclohexil-amida como antagonistas de los receptores de crf |
CN102762572A (zh) | 2010-02-01 | 2012-10-31 | 诺瓦提斯公司 | 作为CRF-1受体拮抗剂的吡唑并[5,1b]*唑衍生物 |
JP5748777B2 (ja) | 2010-02-02 | 2015-07-15 | ノバルティス アーゲー | Crf受容体アンタゴニストとしてのシクロヘキシルアミド誘導体 |
UY34094A (es) | 2011-05-27 | 2013-01-03 | Novartis Ag | Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina |
CA2867043A1 (en) | 2012-05-03 | 2013-11-07 | Novartis Ag | L-malate salt of 2,7-diaza-spiro[4.5]dec-7-yle derivatives and crystalline forms thereof as ghrelin receptor agonists |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH111472A (ja) | 1996-04-30 | 1999-01-06 | Dainippon Pharmaceut Co Ltd | ベンズアミド誘導体及びそれを含有する医薬組成物 |
WO1999055674A1 (fr) | 1998-04-28 | 1999-11-04 | Dainippon Pharmaceutical Co., Ltd. | Derives de 1-[(1-substituee-4-piperidinyle)methyle]-4-piperidine, procede de production de ceux-ci, compositions medicinales contenant ces composes et intermediaires de ces composes |
JP2000080081A (ja) | 1998-06-24 | 2000-03-21 | Dainippon Pharmaceut Co Ltd | 1―〔(1―置換―4―ピペリジニル)メチル〕―4―ピペリジン誘導体及びそれを含有する医薬組成物 |
JP2001122784A (ja) | 1999-10-27 | 2001-05-08 | Dainippon Pharmaceut Co Ltd | 1−[(1−置換−4−ピペリジニル)メチル]−4−ピペリジン誘導体からなる医薬 |
-
2002
- 2002-12-18 US US10/321,615 patent/US6696468B2/en not_active Expired - Fee Related
-
2003
- 2003-01-03 PT PT03250050T patent/PT1362857E/pt unknown
- 2003-01-03 AT AT03250050T patent/ATE273304T1/de not_active IP Right Cessation
- 2003-01-03 EP EP03250050A patent/EP1362857B1/en not_active Expired - Lifetime
- 2003-01-03 DE DE60300021T patent/DE60300021T2/de not_active Expired - Fee Related
- 2003-01-03 ES ES03250050T patent/ES2227500T3/es not_active Expired - Lifetime
- 2003-01-03 DK DK03250050T patent/DK1362857T3/da active
- 2003-05-08 TW TW092112525A patent/TW200400186A/zh unknown
- 2003-05-15 KR KR10-2004-7018158A patent/KR20040107520A/ko not_active Application Discontinuation
- 2003-05-15 IL IL16501203A patent/IL165012A0/xx unknown
- 2003-05-15 SK SK5019-2004A patent/SK50192004A3/sk unknown
- 2003-05-15 CN CNA03811089XA patent/CN1653063A/zh active Pending
- 2003-05-15 HU HU0501016A patent/HUP0501016A2/hu unknown
- 2003-05-15 JP JP2003137413A patent/JP3643107B2/ja not_active Expired - Fee Related
- 2003-05-15 AU AU2003230245A patent/AU2003230245A1/en not_active Abandoned
- 2003-05-15 TR TR2004/03020T patent/TR200403020T2/xx unknown
- 2003-05-15 RU RU2004136853/04A patent/RU2004136853A/ru not_active Application Discontinuation
- 2003-05-15 CA CA002483368A patent/CA2483368A1/en not_active Abandoned
- 2003-05-15 BR BR0309933-4A patent/BR0309933A/pt not_active Application Discontinuation
- 2003-05-15 PL PL03372724A patent/PL372724A1/pl not_active Application Discontinuation
- 2003-05-15 MX MXPA04011332A patent/MXPA04011332A/es unknown
- 2003-05-15 AR ARP030101702A patent/AR040021A1/es unknown
- 2003-05-15 WO PCT/JP2003/006051 patent/WO2003097638A1/en not_active Application Discontinuation
- 2003-05-15 CZ CZ20041084A patent/CZ20041084A3/cs unknown
-
2004
- 2004-04-22 HK HK04102812A patent/HK1060118A1/xx not_active IP Right Cessation
- 2004-11-09 ZA ZA200409035A patent/ZA200409053B/en unknown
- 2004-12-15 NO NO20045469A patent/NO20045469L/no unknown
Also Published As
Publication number | Publication date |
---|---|
JP2004043453A (ja) | 2004-02-12 |
TR200403020T2 (tr) | 2005-05-23 |
HK1060118A1 (en) | 2004-07-30 |
ATE273304T1 (de) | 2004-08-15 |
KR20040107520A (ko) | 2004-12-20 |
NO20045469L (no) | 2005-02-16 |
MXPA04011332A (es) | 2005-02-14 |
US20030216433A1 (en) | 2003-11-20 |
EP1362857B1 (en) | 2004-08-11 |
EP1362857A1 (en) | 2003-11-19 |
PT1362857E (pt) | 2004-11-30 |
DK1362857T3 (da) | 2004-12-20 |
HUP0501016A2 (en) | 2006-02-28 |
BR0309933A (pt) | 2005-02-09 |
CA2483368A1 (en) | 2003-11-27 |
JP3643107B2 (ja) | 2005-04-27 |
DE60300021D1 (de) | 2004-09-16 |
CZ20041084A3 (cs) | 2005-02-16 |
US6696468B2 (en) | 2004-02-24 |
WO2003097638A1 (en) | 2003-11-27 |
DE60300021T2 (de) | 2005-09-08 |
RU2004136853A (ru) | 2005-06-27 |
AR040021A1 (es) | 2005-03-09 |
ES2227500T3 (es) | 2005-04-01 |
TW200400186A (en) | 2004-01-01 |
ZA200409053B (en) | 2005-07-12 |
CN1653063A (zh) | 2005-08-10 |
SK50192004A3 (sk) | 2005-04-01 |
AU2003230245A1 (en) | 2003-12-02 |
IL165012A0 (en) | 2005-12-18 |
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Legal Events
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REFS | Decisions on refusal to grant patents (taken after the publication of the particulars of the applications) |