PL355531A1 - Sposób wytwarzania citalopramu - Google Patents

Sposób wytwarzania citalopramu

Info

Publication number: PL355531A1
Authority: PL; Poland
Prior art keywords: preparation; citalopram; phtalid; cyano; new
Prior art date: 1999-12-30

Application number

PL99355531A

Other languages

English (en)

Other versions

PL198803B1 (pl

Inventor

Hans Petersen

Michael Harold Rock

Original Assignee

H.Lundbeck A/S

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-12-30

Filing date

1999-12-30

Publication date

2004-05-04

1999-12-30 Application filed by H.Lundbeck A/S filed Critical H.Lundbeck A/S

2004-05-04 Publication of PL355531A1 publication Critical patent/PL355531A1/pl

2008-07-31 Publication of PL198803B1 publication Critical patent/PL198803B1/pl

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J23/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
- B01J23/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals
- B01J23/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals of the platinum group metals
- B01J23/44—Palladium
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J23/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
- B01J23/70—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of the iron group metals or copper
- B01J23/74—Iron group metals
- B01J23/755—Nickel

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Materials Engineering (AREA)
Chemical Kinetics & Catalysis (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Steroid Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Furan Compounds (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Cephalosporin Compounds (AREA)

PL355531A 1999-12-30 1999-12-30 Sposób wytwarzania 5-cyjano-3H-izobenzofuran-1-onu PL198803B1 (pl)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/DK1999/000740 WO2001049672A1 (en)	1999-12-30	1999-12-30	Method for the preparation of citalopram

Publications (2)

Publication Number	Publication Date
PL355531A1 true PL355531A1 (pl)	2004-05-04
PL198803B1 PL198803B1 (pl)	2008-07-31

Family

ID=8157174

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL355531A PL198803B1 (pl)	1999-12-30	1999-12-30	Sposób wytwarzania 5-cyjano-3H-izobenzofuran-1-onu

Country Status (28)

Country	Link
US (2)	US20020198391A1 (pl)
EP (1)	EP1246813B1 (pl)
JP (1)	JP2003519218A (pl)
KR (1)	KR100653141B1 (pl)
CN (1)	CN1211377C (pl)
AT (1)	ATE253568T1 (pl)
AU (1)	AU1858400A (pl)
BR (1)	BR9917604A (pl)
CA (1)	CA2395733C (pl)
CZ (1)	CZ20022627A3 (pl)
DE (1)	DE69912652T2 (pl)
DK (1)	DK1246813T3 (pl)
EA (1)	EA004055B1 (pl)
ES (1)	ES2207312T3 (pl)
HK (1)	HK1052512B (pl)
HR (1)	HRP20020633A2 (pl)
HU (1)	HUP0203840A3 (pl)
IL (2)	IL150367A0 (pl)
IS (1)	IS2167B (pl)
MX (1)	MXPA02006504A (pl)
NO (1)	NO328359B1 (pl)
PL (1)	PL198803B1 (pl)
PT (1)	PT1246813E (pl)
SI (1)	SI1246813T1 (pl)
SK (1)	SK11052002A3 (pl)
TR (1)	TR200201688T2 (pl)
UA (1)	UA73336C2 (pl)
WO (1)	WO2001049672A1 (pl)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE69907037T3 (de)	1999-04-14	2010-02-18	H. Lundbeck A/S	Verfahren zur herstellung von citalopram
IL150335A0 (en)	1999-12-28	2002-12-01	Lundbeck & Co As H	Method for the preparation of citalopram
DK1254129T3 (da)	2000-01-14	2004-03-29	Lundbeck & Co As H	Fremgangsmåde til fremstilling af 5-cyanophthalid
IES20010157A2 (en)	2000-03-03	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
IES20010206A2 (en)	2000-03-13	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
IL151566A0 (en)	2000-03-13	2003-04-10	Lundbeck & Co As H	Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
HUP0300274A2 (hu)	2000-03-13	2003-06-28	H. Lundbeck A/S	Eljárás citalopram előállítására
SK14512002A3 (sk)	2000-03-14	2003-03-04	H. Lundbeck A/S	Spôsob výroby citalopramu, medziprodukt a citalopram výrobený týmto spôsobom
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
US6339182B1 (en) *	2000-06-20	2002-01-15	Chevron U.S.A. Inc.	Separation of olefins from paraffins using ionic liquid solutions
US20050154052A1 (en) *	2003-03-24	2005-07-14	Hetero Drugs Limited	Novel crystalline forms of (s)-citalopram oxalate
CN100457747C (zh) *	2006-11-21	2009-02-04	浙江大学	抗抑郁药西酞普兰关键中间体5-氰基苯酞的制备工艺
CN103127815B (zh) *	2013-02-19	2015-10-28	浙江大学	一种利用卤硫作用提高二氧化硫捕集性能的方法

Family Cites Families (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143702A (pl)	1965-03-18
GB1526331A (en) *	1976-01-14	1978-09-27	Kefalas As	Phthalanes
US4665181A (en) *	1984-05-17	1987-05-12	Pennwalt Corporation	Anti-inflammatory phthalazinones
GB8419963D0 (en)	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
US5296507A (en)	1990-09-06	1994-03-22	H.Lundbeck A/S	Treatment of cerbrovascular disorders
JPH0881456A (ja) *	1994-09-14	1996-03-26	Sumitomo Chem Co Ltd	１，１，３，３−テトラクロロ−１，３−ジヒドロイソベンゾフラン誘導体の製造法
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
NZ501737A (en) *	1997-07-08	2001-10-26	H	Method for the preparation of citalopram using Grignard reagent 4-halogen-fluorophenyl and 3-halogen-N,N-dimethyl-propylamine
UA62985C2 (en) *	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
DE1042310T1 (de) *	1997-11-11	2001-04-19	Lundbeck & Co As H	Verfahren zur herstellung von citaloprame
PL199423B1 (pl)	1998-10-20	2008-09-30	Lundbeck & Co As H	Sposób wytwarzania citalopramu
PT1140886E (pt)	1998-12-23	2003-08-29	Lundbeck & Co As H	Metodo para a preparacao de 5- cianoftalida
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
DE69907037T3 (de)	1999-04-14	2010-02-18	H. Lundbeck A/S	Verfahren zur herstellung von citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
CH692421A5 (de)	1999-10-25	2002-06-14	Lundbeck & Co As H	Verfahren zur Herstellung von Citalopram.
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
IL150335A0 (en)	1999-12-28	2002-12-01	Lundbeck & Co As H	Method for the preparation of citalopram
DK1254129T3 (da)	2000-01-14	2004-03-29	Lundbeck & Co As H	Fremgangsmåde til fremstilling af 5-cyanophthalid
FR2805812A1 (fr)	2000-02-24	2001-09-07	Lundbeck & Co As H	Procede de preparation du citalopram
IES20010143A2 (en)	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
FI20011622L (fi)	2000-08-18	2002-02-19	Lundbeck & Co As H	Menetelmä sitalopraamin valmistamiseksi
TR200201166T1 (tr)	2000-12-22	2002-10-21	H.Lundbecks A/S	Saf sitalopram hazırlanması için yöntem
EP1181272B1 (en)	2000-12-28	2002-08-28	H. Lundbeck A/S	Process for the preparation of pure citalopram

1999
- 1999-12-30 CZ CZ20022627A patent/CZ20022627A3/cs unknown
- 1999-12-30 EA EA200200728A patent/EA004055B1/ru not_active IP Right Cessation
- 1999-12-30 IL IL15036799A patent/IL150367A0/xx unknown
- 1999-12-30 UA UA2002065265A patent/UA73336C2/uk unknown
- 1999-12-30 SK SK1105-2002A patent/SK11052002A3/sk unknown
- 1999-12-30 SI SI9930473T patent/SI1246813T1/xx unknown
- 1999-12-30 DE DE69912652T patent/DE69912652T2/de not_active Expired - Lifetime
- 1999-12-30 DK DK99962133T patent/DK1246813T3/da active
- 1999-12-30 TR TR2002/01688T patent/TR200201688T2/xx unknown
- 1999-12-30 KR KR1020027008572A patent/KR100653141B1/ko not_active IP Right Cessation
- 1999-12-30 PL PL355531A patent/PL198803B1/pl not_active IP Right Cessation
- 1999-12-30 AU AU18584/00A patent/AU1858400A/en not_active Abandoned
- 1999-12-30 HU HU0203840A patent/HUP0203840A3/hu unknown
- 1999-12-30 CA CA002395733A patent/CA2395733C/en not_active Expired - Fee Related
- 1999-12-30 JP JP2001550212A patent/JP2003519218A/ja active Pending
- 1999-12-30 AT AT99962133T patent/ATE253568T1/de not_active IP Right Cessation
- 1999-12-30 BR BR9917604-1A patent/BR9917604A/pt not_active Application Discontinuation
- 1999-12-30 EP EP99962133A patent/EP1246813B1/en not_active Expired - Lifetime
- 1999-12-30 ES ES99962133T patent/ES2207312T3/es not_active Expired - Lifetime
- 1999-12-30 WO PCT/DK1999/000740 patent/WO2001049672A1/en active IP Right Grant
- 1999-12-30 CN CNB998170674A patent/CN1211377C/zh not_active Expired - Fee Related
- 1999-12-30 PT PT99962133T patent/PT1246813E/pt unknown
- 1999-12-30 MX MXPA02006504A patent/MXPA02006504A/es active IP Right Grant
2002
- 2002-06-19 IS IS6433A patent/IS2167B/is unknown
- 2002-06-23 IL IL150367A patent/IL150367A/en not_active IP Right Cessation
- 2002-06-27 US US10/186,337 patent/US20020198391A1/en not_active Abandoned
- 2002-06-28 NO NO20023150A patent/NO328359B1/no not_active IP Right Cessation
- 2002-07-26 HR HRP20020633 patent/HRP20020633A2/hr not_active Application Discontinuation
2003
- 2003-07-08 HK HK03104874.0A patent/HK1052512B/zh not_active IP Right Cessation
2005
- 2005-11-23 US US11/285,922 patent/US7271273B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
PT1246813E (pt)	2004-02-27
DE69912652T2 (de)	2004-06-09
EA004055B1 (ru)	2003-12-25
NO20023150D0 (no)	2002-06-28
KR100653141B1 (ko)	2006-12-01
ATE253568T1 (de)	2003-11-15
NO328359B1 (no)	2010-02-01
IS6433A (is)	2002-06-19
MXPA02006504A (es)	2002-12-09
IL150367A (en)	2010-06-16
IS2167B (is)	2006-11-15
US7271273B2 (en)	2007-09-18
EP1246813B1 (en)	2003-11-05
US20020198391A1 (en)	2002-12-26
EP1246813A1 (en)	2002-10-09
UA73336C2 (en)	2005-07-15
WO2001049672A1 (en)	2001-07-12
JP2003519218A (ja)	2003-06-17
SI1246813T1 (en)	2004-08-31
NO20023150L (no)	2002-06-28
AU1858400A (en)	2001-07-16
BR9917604A (pt)	2002-12-31
HUP0203840A3 (en)	2005-02-28
ES2207312T3 (es)	2004-05-16
DK1246813T3 (da)	2004-03-01
DE69912652D1 (de)	2003-12-11
HUP0203840A2 (en)	2003-05-28
KR20020073495A (ko)	2002-09-26
HK1052512A1 (en)	2003-09-19
US20060079700A1 (en)	2006-04-13
IL150367A0 (en)	2002-12-01
CN1391566A (zh)	2003-01-15
HK1052512B (zh)	2006-03-03
PL198803B1 (pl)	2008-07-31
HRP20020633A2 (en)	2004-12-31
CA2395733A1 (en)	2001-07-12
EA200200728A1 (ru)	2002-12-26
SK11052002A3 (sk)	2003-01-09
CA2395733C (en)	2007-03-20
CZ20022627A3 (cs)	2002-10-16
TR200201688T2 (tr)	2002-11-21
CN1211377C (zh)	2005-07-20

Publication	Publication Date	Title
MXPA03005222A (es)	2004-03-26	Derivado de metanosulfonamido-benzofurano, su procedimiento de preparacion y su utilizacion como intermediario de sisntesis.
HK1048122A1 (en)	2003-03-21	Method for the preparation of citalopram.
ZA200108855B (en)	2002-08-28	Method for the preparation of citalopram.
IL150367A0 (en)	2002-12-01	Method for the preparation of citalopram
HK1049002A1 (en)	2003-04-25	Method for the preparation of citalopram.
MXPA03010909A (es)	2004-02-17	Derivados de epotilona.
WO2001079461A3 (en)	2002-01-31	Polypeptides having haloperoxidase activity
ZA200106683B (en)	2002-08-05	Method for the preparation of citalopram.
HK1054378A1 (en)	2003-11-28	Method for the preparation of citalopram.
ZA200110179B (en)	2002-12-11	Process for the preparation of pure citalopram.
ZA200309471B (en)	2004-12-06	Method for the preparation of escitalopram.
AU2002258971A1 (en)	2002-11-05	Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-benzodioxan
PL346463A1 (en)	2001-09-24	Method of obtaining derivatives of resorcinol, method of obtaining novel derivatives of 2-oxazabicyclo[2.2.2.]-octan-5-one, method of obtaining novel derivatives of 1,3-cyclohezandione, method of obtaining novel derivatives of 2-cyclohexanone, novel derivatives of 2-oxazabicyclo[2.2.2.]-octan-5-one, novel derivatives of 1,3-cyclohexanodione, and novel derivatives of 2-cyclohexenonea
BG105197A (en)	2001-10-31	Polymorph form of a medicament
MXPA03005418A (es)	2003-09-24	Conjunto unitario de anillo de tono.
BG107047A (en)	2003-04-30	Method for the preparation of citalopram
AU5823901A (en)	2001-11-20	Method for the preparation of citalopram
BG107046A (en)	2003-05-30	Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
MXPA02011762A (es)	2004-05-17	Proceso para la preparacion de compuestos metales de transicion y su empleo para la polimerizacion de olefinas.
AU2002303529A1 (en)	2002-11-11	Antidepressant azaheterocyclylmethyl derivatives of 1,4,5-trioxa-phenanthrene
BG106958A (en)	2003-03-31	Method for the preparation of citalopram
HK1049485A1 (en)	2003-05-16	DithiepinoÄ6,5-BÜpyridines, and related compositions, methods of producing and uses.
ZA9710343B (en)	1998-06-10	Utilization of an egg-based preparation as an antidepressant.
BG102318A (en)	1999-08-31	Epoxy-azetidinons, their preparation and application
ZA200106687B (en)	2002-02-14	Method for the preparation of citalopram.

Legal Events

Date	Code	Title	Description
2012-02-29	LAPS	Decisions on the lapse of the protection rights	Effective date: 20101230