NO330500B1 - Trisykliske trombinreseptorantagonister - Google Patents

Trisykliske trombinreseptorantagonister Download PDF

Info

Publication number: NO330500B1
Authority: NO; Norway
Prior art keywords: nhc; pharmaceutically acceptable; mmol; acceptable salt; compound
Prior art date: 2002-04-16

Application number

NO20044963A

Other languages

English (en)

Norwegian (no)

Other versions

NO20044963L (no

Inventor

William J Greenlee

Samuel Chackalamannil

Yuguang Wang

Yan Xia

Martin C Clasby

Mariappan Chelliah

Enrico P Veltri

Wenxue Wu

Original Assignee

Schering Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-04-16

Filing date

2004-11-15

Publication date

2011-05-02

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29250954&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO330500(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-11-15 Application filed by Schering Corp filed Critical Schering Corp

2004-11-15 Publication of NO20044963L publication Critical patent/NO20044963L/no

2011-05-02 Publication of NO330500B1 publication Critical patent/NO330500B1/no

Links

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Classifications

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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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Plural Heterocyclic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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NO20044963A 2002-04-16 2004-11-15 Trisykliske trombinreseptorantagonister NO330500B1 (no)

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US37307202P	2002-04-16	2002-04-16
PCT/US2003/011510 WO2003089428A1 (en)	2002-04-16	2003-04-14	Tricyclic thrombin receptor antagonists

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NO2015016C NO2015016I1 (no)	2002-04-16	2015-07-09	Vorapaxar, eller et farmasøytisk akseptabelt salt eller solvat derav

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NO2015016C NO2015016I1 (no)	2002-04-16	2015-07-09	Vorapaxar, eller et farmasøytisk akseptabelt salt eller solvat derav

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JP (2)	JP4558331B2 (zh)
KR (1)	KR101026929B1 (zh)
CN (1)	CN1659162B (zh)
AR (1)	AR039570A1 (zh)
AT (3)	ATE455774T1 (zh)
AU (1)	AU2003221932B2 (zh)
BR (1)	BRPI0309309B8 (zh)
CA (1)	CA2482858C (zh)
CY (3)	CY1107184T1 (zh)
DE (3)	DE60335679D1 (zh)
DK (2)	DK1495018T3 (zh)
EC (1)	ECSP045368A (zh)
ES (3)	ES2357876T3 (zh)
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HK (3)	HK1070887A1 (zh)
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TW (1)	TWI343919B (zh)
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WO2009097970A1 (de)	2008-02-05	2009-08-13	Sanofi-Aventis	Triazolopyridazine als par1-inhibitoren, ihre herstellung und verwendung als arzneimittel
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Also Published As

Publication number	Publication date
DE60331114D1 (de)	2010-03-11
HK1123302A1 (en)	2009-06-12
RU2004133375A (ru)	2005-07-10
ZA200408342B (en)	2006-05-31
EP2062890A1 (en)	2009-05-27
JP2005528406A (ja)	2005-09-22
KR20040099441A (ko)	2004-11-26
HK1070887A1 (en)	2005-06-30
ES2338171T3 (es)	2010-05-04
MY144040A (en)	2011-07-29
SI1495018T1 (sl)	2008-04-30
AU2003221932A1 (en)	2003-11-03
EP1982984A3 (en)	2008-10-29
CN1659162B (zh)	2011-08-31
DE60317493T3 (de)	2018-07-12
US20070270439A1 (en)	2007-11-22
CY2015029I1 (el)	2016-04-13
LU92759I2 (en)	2015-08-31
DE60317493T2 (de)	2008-09-18
ATE494284T1 (de)	2011-01-15
PT2065384E (pt)	2011-03-16
FR15C0047I1 (zh)	2015-08-28
CA2482858A1 (en)	2003-10-30
NO2015016I2 (no)	2015-07-09
US7713999B2 (en)	2010-05-11
BR0309309A (pt)	2005-02-15
NZ575139A (en)	2010-08-27
EP1495018B1 (en)	2007-11-14
US7304078B2 (en)	2007-12-04
CN1659162A (zh)	2005-08-24
AR039570A1 (es)	2005-02-23
PL373332A1 (en)	2005-08-22
EP1982984A2 (en)	2008-10-22
EP1860106B1 (en)	2010-01-20
NZ535880A (en)	2007-11-30
JP4558331B2 (ja)	2010-10-06
RU2329264C9 (ru)	2009-04-20
RU2008106401A (ru)	2009-08-27
KR101026929B1 (ko)	2011-04-04
EP2062890B1 (en)	2011-01-05
TWI343919B (en)	2011-06-21
EP1982984B1 (en)	2013-02-13
ES2357876T3 (es)	2011-05-03
ATE455774T1 (de)	2010-02-15
SI2065384T1 (sl)	2011-05-31
DE60317493D1 (en)	2011-01-13
SG164279A1 (en)	2010-09-29
WO2003089428A1 (en)	2003-10-30
PT1495018E (pt)	2008-02-19
RU2329264C2 (ru)	2008-07-20
AU2003221932B2 (en)	2007-11-22
ATE378330T1 (de)	2007-11-15
EP1495018A1 (en)	2005-01-12
ES2297150T3 (es)	2008-05-01
EP1860106A1 (en)	2007-11-28
PE20040412A1 (es)	2004-07-12
PL214718B1 (pl)	2013-09-30
ECSP045368A (es)	2005-01-03
FR15C0047I2 (fr)	2016-05-06
DK2065384T3 (da)	2011-05-02
MXPA04010308A (es)	2005-02-03
HK1129893A1 (en)	2009-12-11
BRPI0309309B1 (pt)	2018-09-04
EP1495018B3 (en)	2011-03-16
LTC1495018I2 (lt)	2017-04-10
NL300746I2 (zh)	2016-01-21
TW200404068A (en)	2004-03-16
CA2482858C (en)	2010-11-30
ES2297150T7 (es)	2012-03-16
JP2010132710A (ja)	2010-06-17
EP2065384A1 (en)	2009-06-03
DK1495018T3 (da)	2008-02-18
IL164585A0 (en)	2005-12-18
NO20044963L (no)	2004-11-15
US20070179187A1 (en)	2007-08-02
US20030216437A1 (en)	2003-11-20
NL300746I1 (zh)	2016-01-21
BRPI0309309B8 (pt)	2021-05-25
DE60335679D1 (de)	2011-02-17
CY1107184T1 (el)	2012-10-24
IL164585A (en)	2010-11-30
EP2065384B1 (en)	2011-01-05
CY1111363T1 (el)	2015-08-05
NO2015016I1 (no)	2015-07-20
CY2015029I2 (el)	2016-04-13

Publication	Publication Date	Title
NO330500B1 (no)	2011-05-02	Trisykliske trombinreseptorantagonister
AU2001266900B2 (en)	2007-04-05	Thrombin receptor antagonists
AU2002335031B2 (en)	2005-06-30	Himbacine analogues as thrombin receptor antagonists
EP1999111B1 (en)	2013-12-18	Monocyclic and bicyclic himbacine derivatives useful as thrombin receptor antagonists
JP5139307B2 (ja)	2013-02-06	ナトリウムチャネルモジュレーターとしてのプロリンアミド誘導体
AU2002335031A1 (en)	2003-07-03	Himbacine analogues as thrombin receptor antagonists
JP2010517926A (ja)	2010-05-27	グルタミン酸受容体を増強する、統合失調症の治療に有用な４−フェニル−３−（２−プロピルスルホニルアミノ）テトラヒドロフラン誘導体
EP2007755B1 (en)	2012-06-27	Fused ring thrombin receptor antagonists
AU2008200842B2 (en)	2011-09-15	Tricyclic thrombin receptor antagonists

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