NO166131C - Analogifremgangsmaate for fremstilling av s(-)-pyridobenzoksazinforbindelser. - Google Patents

Analogifremgangsmaate for fremstilling av s(-)-pyridobenzoksazinforbindelser.

Info

Publication number: NO166131C
Authority: NO; Norway
Prior art keywords: compounds; pyridobenzoksazine; preparation; preparing; optically active
Prior art date: 1985-06-20

Application number

NO862426A

Other languages

English (en)

Other versions

NO862426D0 (no

NO862426L (no

NO166131B (no

Inventor

Isao Hayakawa

Shohgo Atarashi

Shuichi Yokohama

Masazumi Imamura

Katsuichi Sakano

Nobuyuki Higashihashi

Masayuki Ohshima

Original Assignee

Daiichi Seiyaku Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-20

Filing date

1986-06-18

Publication date

1991-06-05

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27281433&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO166131(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1985-10-11 Priority claimed from JP60226499A external-priority patent/JPH0720946B2/ja

1986-06-18 Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co

1986-06-18 Publication of NO862426D0 publication Critical patent/NO862426D0/no

1986-12-22 Publication of NO862426L publication Critical patent/NO862426L/no

1988-08-25 Priority to NO883791A priority Critical patent/NO169896C/no

1991-02-25 Publication of NO166131B publication Critical patent/NO166131B/no

1991-06-05 Publication of NO166131C publication Critical patent/NO166131C/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NO862426A 1985-06-20 1986-06-18 Analogifremgangsmaate for fremstilling av s(-)-pyridobenzoksazinforbindelser. NO166131C (no)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
NO883791A NO169896C (no)	1985-06-20	1988-08-25	3-s-3-alkylbenzoksazinderivater

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP13471285		1985-06-20
JP60226499A JPH0720946B2 (ja)	1985-10-11	1985-10-11	光学活性３−メチルベンゾオキサジン誘導体およびその製法
JP1649686		1986-01-28

Publications (4)

Publication Number	Publication Date
NO862426D0 NO862426D0 (no)	1986-06-18
NO862426L NO862426L (no)	1986-12-22
NO166131B NO166131B (no)	1991-02-25
NO166131C true NO166131C (no)	1991-06-05

Family

ID=27281433

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO862426A NO166131C (no)	1985-06-20	1986-06-18	Analogifremgangsmaate for fremstilling av s(-)-pyridobenzoksazinforbindelser.

Country Status (16)

Country	Link
US (3)	US5053407A (no)
EP (1)	EP0206283B1 (no)
KR (2)	KR920010048B1 (no)
AT (1)	ATE85057T1 (no)
BG (1)	BG60527B2 (no)
CA (1)	CA1304080C (no)
DE (2)	DE3687599T2 (no)
DK (1)	DK170473B1 (no)
ES (1)	ES8801251A1 (no)
FI (1)	FI90241C (no)
GR (1)	GR861625B (no)
HK (1)	HK91793A (no)
IE (1)	IE59463B1 (no)
NL (1)	NL980016I2 (no)
NO (1)	NO166131C (no)
YU (3)	YU44918B (no)

Families Citing this family (58)

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FR2655545B1 (fr) *	1989-12-11	1994-06-10	Rhone Poulenc Sante	Nouvelle application therapeutique des derives des fluoroquinolones.
TW208013B (no) *	1990-03-01	1993-06-21	Daiichi Co Ltd
FI96313C (fi) *	1990-11-28	1996-06-10	Daiichi Seiyaku Co	Menetelmä terapeuttisesti käyttökelpoisten ja optisesti aktiivisten 10-(3-amino-4,4-dialkyyli-1-pyrrolidinyyli)-9-fluori-2,3-dihydro-3(S)-metyyli-7-okso-7H-pyrido/1,2,3-de//1,4/bentsoksatsiini-6-karboksyylihappojen valmistamiseksi
ES2055656B1 (es) *	1992-10-07	1995-11-16	Etilo Derivados	Procedimiento para la obtencion de benzoxazinas utiles para sintesis de ofloxacina, levofloxacina y derivados.
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ES2256331T3 (es)	2000-12-21	2006-07-16	PHARMACIA & UPJOHN COMPANY LLC	Derivados de quinolina antimicrobianos y uso de los mismos para tratar infecciones bacterianas.
WO2002070726A1 (en)	2001-03-07	2002-09-12	Daiichi Pharmaceutical Co., Ltd.	Process for preparation of optically active propoxyaniline derivatives
JP4031992B2 (ja)	2001-04-27	2008-01-09	リサーチインスティチュートオブインダストリアルサイエンスアンドテクノロジー	優れた熱間加工性を持つ高マンガン二相ステンレス鋼及びその製造方法
US7425628B2 (en)	2001-10-03	2008-09-16	Teva Pharmaceutical Industries Ltd.	Methods for the purification of levofloxacin
ES2272781T5 (es)	2001-10-03	2010-04-06	Teva Pharmaceutical Industries Ltd.	Preparacion de levofloxacino hemihidratado.
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EP1465606A4 (en) *	2001-12-24	2009-04-22	Teva Pharma	DOSAGE FORM WITH PASTILLE CORE ACTIVE PRINCIPLE COATED IN COMPRESSED ANNULAR BODY OF POWDER OR GRANULAR SUBSTANCE, AND METHOD AND TOOLS FOR PRODUCTION OF SAID DOSAGE FORM
US20040052843A1 (en) *	2001-12-24	2004-03-18	Lerner E. Itzhak	Controlled release dosage forms
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AU2003262704A1 (en) *	2002-08-14	2004-08-30	Teva Pharmaceutical Industries Ltd.	Synthesis of gatifloxacin
US20040152701A1 (en) *	2002-12-02	2004-08-05	Dr. Reddy's Laboratories Limited	Novel anhydrous crystalline form of Levofloxacin and process for preparation there of
FR2859471B1 (fr)	2003-09-09	2006-02-03	Solvay	Procede pour la fabrication d'un compose enantiopur
KR20080004460A (ko)	2005-02-07	2008-01-09	미츠비시 웰파마 가부시키가이샤	광학 활성인 테트라히드로나프탈렌 유도체
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US7973022B2 (en)	2006-02-17	2011-07-05	Idexx Laboratories, Inc.	Fluoroquinolone carboxylic acid salt compositions
US20070197548A1 (en)	2006-02-17	2007-08-23	Murthy Yerramilli V S	Fluoroquinolone compositions
WO2008019292A2 (en) *	2006-08-04	2008-02-14	Trustees Of Boston University	Compositions and methods for potentiating antibiotic activity
WO2008077643A1 (en) *	2006-12-22	2008-07-03	Farmaprojects, S.A.	Process for the preparation of an antibacterial quinolone compound
EP1939206A1 (en) *	2006-12-22	2008-07-02	Farmaprojects, S.A.	Process for the preparation of an antibacterial quinolone compound
US7964723B2 (en)	2008-08-02	2011-06-21	Apeloa-Kangyu	And practical process for exclusively producing (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido-[1,2,3,de][1,4]benzoxazine-6-carboxylic acid hemihydrate
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PT2346509T (pt)	2008-10-07	2020-08-05	Horizon Orphan Llc	Inalação de levofloxacina para redução da inflamação pulmonar
MX2011012134A (es)	2009-05-15	2012-02-08	Redx Pharma Ltd	Derivados de farmaco de oxido-reduccion.
PT2473170T (pt)	2009-09-04	2019-08-23	Horizon Orphan Llc	Utilização de levofloxacina em aerossol para tratamento de fibrose cística
CN101659669B (zh) *	2009-09-04	2011-07-20	诚达药业股份有限公司	左旋氧氟沙星的制备方法
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Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5746986A (en) *	1980-09-02	1982-03-17	Dai Ichi Seiyaku Co Ltd	Pyrido(1,2,3-de)(1,4)benzoxazine derivative
JPS5852290A (ja) *	1981-09-21	1983-03-28	Dai Ichi Seiyaku Co Ltd	ピリドベンゾオキサジンカルボン酸誘導体
DE3543513A1 (de) *	1985-12-10	1987-06-11	Bayer Ag	Enantiomerenreine 1,8-verbrueckte 4-chinolon-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende arzneimittel und ihre verwendung zur herstellung von arzneimitteln

1986
- 1986-06-18 NO NO862426A patent/NO166131C/no not_active IP Right Cessation
- 1986-06-18 DK DK285086A patent/DK170473B1/da active Protection Beyond IP Right Term
- 1986-06-19 FI FI862643A patent/FI90241C/fi not_active IP Right Cessation
- 1986-06-19 ES ES556292A patent/ES8801251A1/es not_active Expired
- 1986-06-19 CA CA000512000A patent/CA1304080C/en not_active Expired - Lifetime
- 1986-06-19 YU YU1073/86A patent/YU44918B/xx unknown
- 1986-06-19 IE IE163186A patent/IE59463B1/en not_active IP Right Cessation
- 1986-06-20 AT AT86108442T patent/ATE85057T1/de active
- 1986-06-20 DE DE8686108442T patent/DE3687599T2/de not_active Expired - Lifetime
- 1986-06-20 EP EP86108442A patent/EP0206283B1/en not_active Expired - Lifetime
- 1986-06-20 KR KR1019860004934A patent/KR920010048B1/ko not_active Expired
- 1986-06-20 GR GR861625A patent/GR861625B/el unknown
- 1986-06-20 DE DE19863687599 patent/DE19875012I2/de active Active
- 1986-06-20 US US06/876,623 patent/US5053407A/en not_active Expired - Lifetime
1988
- 1988-10-05 YU YU1867/88A patent/YU45512B/xx unknown
1989
- 1989-03-23 US US07/327,653 patent/US4985557A/en not_active Expired - Lifetime
- 1989-10-30 YU YU2098/89A patent/YU45524B/xx unknown
1990
- 1990-10-31 KR KR1019900017517A patent/KR940003757B1/ko not_active Expired - Lifetime
1991
- 1991-08-28 US US07/754,198 patent/US5142046A/en not_active Expired - Lifetime
1993
- 1993-09-02 HK HK917/93A patent/HK91793A/en not_active IP Right Cessation
1994
- 1994-02-22 BG BG098511A patent/BG60527B2/bg unknown
1998
- 1998-04-22 NL NL980016C patent/NL980016I2/nl unknown

Also Published As

Publication number	Publication date
DK285086D0 (da)	1986-06-18
YU44918B (en)	1991-04-30
KR870000340A (ko)	1987-02-17
IE59463B1 (en)	1994-02-23
CA1304080C (en)	1992-06-23
HK91793A (en)	1993-09-10
EP0206283A3 (en)	1988-08-10
DE3687599D1 (de)	1993-03-11
KR940003757B1 (ko)	1994-04-30
YU209889A (en)	1990-04-30
ES8801251A1 (es)	1988-01-01
NO862426D0 (no)	1986-06-18
NO862426L (no)	1986-12-22
US4985557A (en)	1991-01-15
NL980016I1 (nl)	1998-07-01
ATE85057T1 (de)	1993-02-15
KR920010048B1 (ko)	1992-11-13
NO166131B (no)	1991-02-25
EP0206283B1 (en)	1993-01-27
YU107386A (en)	1988-02-29
EP0206283A2 (en)	1986-12-30
US5142046A (en)	1992-08-25
DK285086A (da)	1986-12-21
IE861631L (en)	1986-12-20
ES556292A0 (es)	1988-01-01
BG60527B2 (bg)	1995-07-28
YU45524B (en)	1992-05-28
US5053407A (en)	1991-10-01
KR920009279A (ko)	1992-05-28
FI90241C (fi)	1994-01-10
DK170473B1 (da)	1995-09-11
YU186788A (en)	1989-04-30
YU45512B (en)	1992-05-28
GR861625B (en)	1986-10-21
DE3687599T2 (de)	1993-05-19
FI862643A7 (fi)	1986-12-21
FI862643A0 (fi)	1986-06-19
DE19875012I2 (de)	2006-06-29
NL980016I2 (nl)	1998-08-03
FI90241B (fi)	1993-09-30

Publication	Publication Date	Title
NO166131C (no)	1991-06-05	Analogifremgangsmaate for fremstilling av s(-)-pyridobenzoksazinforbindelser.
NO911600D0 (no)	1991-04-23	Fremgangsmaate for fremstilling av n-(3-fluor-2-fosfonyl-metoksypropyl)-derivater av heterocykliske purin- og pyrimidinbaser.
ES2017498B3 (es)	1991-02-16	Derivado de 2-fenilbenzoxepina.
NO168243C (no)	1992-01-29	Analogifremgangsmaate for fremstilling av terapeutisk aktive alkansulfonanilid-derivater.
DK508885A (da)	1986-05-14	Esterderivat af antibiotekum l 17046 og fremgangsmaade til fremstilling deraf
ES548330A0 (es)	1986-11-16	Un metodo de preparacion de un compuesto de tiadiazina
NO853551L (no)	1986-03-13	Fremgangsmaate ved fremstilling av prolinderivater og lignende forbindelser med antihypertensiv aktivitet.
NO174963C (no)	1994-08-10	Analogifremgangsmåte for fremstilling av terapeutisk aktive 8-fluorantracyklinglucosider
EP0486687A4 (en)	1992-06-17	Quinolonecarboxylic acid derivatives
AU553765B2 (en)	1986-07-24	Biologically active heterocyclic hydroximidates and thiolhydroximidates and carbamate ester derivatives thereof
AU2013888A (en)	1989-02-02	Uricosuric composition
ES2039270T3 (es)	1993-09-16	Derivados de gamma-l-glutamil-4-nitroanilida y procedimiento para determinar actividad de gamma-gtp utilizandolos.
GR3002699T3 (en)	1993-01-25	Process for stabilising procaterol
HUT38920A (en)	1986-07-28	Process for producing anticonvulsive tetrahydro-1,2,4-oxadiazine-5-thion derivatives
SU1573830A1 (ru)	1999-08-10	Фосфорилированные оксиэтиловые эфиры 2,4-дихлорфеноксиуксусной кислоты, обладающие гербицидной активностью
SU1455633A1 (ru)	1999-05-27	О,о-диизопропил-о-[1, 1-диметил-2-пропилтио-2-(о-о-диизопропилфосфорил)- имино]-этилфосфат, обладающий бактерицидной активностью
SU1351063A1 (ru)	2006-12-20	Производные 2-тиазолзамещенного 5-нитрофурана, проявляющие антистафилококковую активность

Legal Events

Date	Code	Title	Description
2006-08-21	MK1K	Patent expired