NL970021I2 - Piperidylesters of -amiden met een alkyleenbrug enfarmaceutische preparaten die deze esters en amiden bevatten. - Google Patents
Piperidylesters of -amiden met een alkyleenbrug enfarmaceutische preparaten die deze esters en amiden bevatten.Info
- Publication number
- NL970021I2 NL970021I2 NL970021C NL970021C NL970021I2 NL 970021 I2 NL970021 I2 NL 970021I2 NL 970021 C NL970021 C NL 970021C NL 970021 C NL970021 C NL 970021C NL 970021 I2 NL970021 I2 NL 970021I2
- Authority
- NL
- Netherlands
- Prior art keywords
- amides
- esters
- alkylene
- pharmaceutical preparations
- preparations containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
- C07D451/12—Oxygen atoms acylated by aromatic or heteroaromatic carboxylic acids, e.g. cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH397982 | 1982-06-29 | ||
CH426782 | 1982-07-13 | ||
CH695082 | 1982-11-30 | ||
CH695182 | 1982-11-30 | ||
CH749482 | 1982-12-22 | ||
CH749582 | 1982-12-22 | ||
CH125683 | 1983-03-09 |
Publications (2)
Publication Number | Publication Date |
---|---|
NL970021I1 NL970021I1 (nl) | 1997-08-01 |
NL970021I2 true NL970021I2 (nl) | 1998-01-05 |
Family
ID=27561049
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL8302253A NL191991C (nl) | 1982-06-29 | 1983-06-24 | Piperidylesters of -amiden met een alkyleenbrug en farmaceutische prepa- raten die deze esters en amiden bevatten. |
NL970021C NL970021I2 (nl) | 1982-06-29 | 1997-06-02 | Piperidylesters of -amiden met een alkyleenbrug enfarmaceutische preparaten die deze esters en amiden bevatten. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL8302253A NL191991C (nl) | 1982-06-29 | 1983-06-24 | Piperidylesters of -amiden met een alkyleenbrug en farmaceutische prepa- raten die deze esters en amiden bevatten. |
Country Status (20)
Country | Link |
---|---|
US (3) | US4803199A (nl) |
AT (1) | AT391136B (nl) |
AU (2) | AU570002B2 (nl) |
CH (2) | CH669792A5 (nl) |
CY (1) | CY1500A (nl) |
DE (6) | DE3348332C2 (nl) |
DK (1) | DK172475B1 (nl) |
FI (1) | FI74707C (nl) |
FR (1) | FR2531083B1 (nl) |
GB (4) | GB2125398B (nl) |
HK (1) | HK60690A (nl) |
HU (1) | HU191053B (nl) |
IL (1) | IL69081A (nl) |
IT (1) | IT1173724B (nl) |
NL (2) | NL191991C (nl) |
NZ (1) | NZ204714A (nl) |
PT (1) | PT76937B (nl) |
SE (1) | SE463210B (nl) |
SG (1) | SG53789G (nl) |
WO (1) | WO1984000166A1 (nl) |
Families Citing this family (142)
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FR2531083B1 (fr) * | 1982-06-29 | 1986-11-28 | Sandoz Sa | Nouveaux derives de la piperidine, leur preparation et leur utilisation comme medicaments |
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GB8315495D0 (en) * | 1983-06-06 | 1983-07-13 | Sumitomo Chemical Co | Fungicidal aniline derivatives |
CH664567A5 (de) * | 1983-08-26 | 1988-03-15 | Sandoz Ag | Aromatische carbonsaeure- und sulfonsaeureester oder -amide. |
JPS6084281A (ja) * | 1983-09-14 | 1985-05-13 | Yoshitomi Pharmaceut Ind Ltd | 3−インド−ルカルボキサミド類 |
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US5175173A (en) * | 1983-12-22 | 1992-12-29 | Sun Jung Hui | Carboxamides useful as antiemetic or antipsychotic agents |
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CH667657A5 (de) * | 1985-01-07 | 1988-10-31 | Sandoz Ag | Carbocyclische und heterocyclische carbonylmethylen- und methylpiperidine und -pyrrolidine. |
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DE3689974T2 (de) * | 1985-03-14 | 1994-11-03 | Beecham Group Plc | Arzneimittel zur Behandlung von Emesis. |
DE3687080T2 (de) * | 1985-04-27 | 1993-03-25 | Beecham Group Plc | Azabicyclononyl-indazol-carboxamid mit 5-ht-antagonistischer wirkung. |
US4937247A (en) * | 1985-04-27 | 1990-06-26 | Beecham Group P.L.C. | 1-acyl indazoles |
GB8525913D0 (en) * | 1985-10-21 | 1985-11-27 | Beecham Group Plc | Compounds |
GB8623142D0 (en) * | 1986-09-26 | 1986-10-29 | Beecham Group Plc | Compounds |
GB8511988D0 (en) * | 1985-05-11 | 1985-06-19 | Beecham Group Plc | Compounds |
GB8515845D0 (en) * | 1985-06-22 | 1985-07-24 | Beecham Group Plc | Treatment |
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GB8520616D0 (en) * | 1985-08-16 | 1985-09-25 | Beecham Group Plc | Compounds |
GB8525844D0 (en) * | 1985-10-19 | 1985-11-20 | Beecham Group Plc | Compounds |
ES2053451T3 (es) * | 1986-01-07 | 1994-08-01 | Beecham Group Plc | Un procedimiento para la preparacion de un compuesto que tiene propiedades farmacologicas utiles. |
EP0235878A3 (en) * | 1986-01-16 | 1989-06-14 | Beecham Group Plc | Novel compounds |
US4722834A (en) * | 1986-03-05 | 1988-02-02 | A. H. Robins Company, Incorporated | Method of using 2-alkoxy-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamide-N-oxides to control emesis caused by anticancer drugs |
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US4772459A (en) * | 1986-09-09 | 1988-09-20 | Erbamont, Inc. | Method for controlling emesis caused by chemotherapeutic agents and antiemetic agents useful therein |
ATE146077T1 (de) * | 1986-09-22 | 1996-12-15 | Janssen Pharmaceutica Nv | Serotonin-antagonisten zur behandlung von wunden |
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US4906755A (en) * | 1986-11-03 | 1990-03-06 | Merrell Dow Pharmaceuticals Inc. | Esters of hexahydro-8-hydroxy-2,6-methano-2H-quinolizin-3-(4H)-one and related compounds |
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GB8701022D0 (en) * | 1987-01-19 | 1987-02-18 | Beecham Group Plc | Treatment |
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-
1983
- 1983-06-22 FR FR8310433A patent/FR2531083B1/fr not_active Expired
- 1983-06-22 FI FI832293A patent/FI74707C/fi not_active IP Right Cessation
- 1983-06-23 DE DE3348332A patent/DE3348332C2/de not_active Expired - Lifetime
- 1983-06-23 DE DE3348333A patent/DE3348333C2/de not_active Expired - Lifetime
- 1983-06-23 DE DE1994175004 patent/DE19475004I2/de active Active
- 1983-06-23 DE DE3348334A patent/DE3348334C2/de not_active Expired - Lifetime
- 1983-06-23 DE DE19833322574 patent/DE3322574A1/de active Granted
- 1983-06-23 DE DE3348331A patent/DE3348331C2/de not_active Expired - Lifetime
- 1983-06-24 NL NL8302253A patent/NL191991C/nl not_active IP Right Cessation
- 1983-06-24 WO PCT/CH1983/000081 patent/WO1984000166A1/de unknown
- 1983-06-27 SE SE8303651A patent/SE463210B/sv not_active IP Right Cessation
- 1983-06-27 AU AU16286/83A patent/AU570002B2/en not_active Expired
- 1983-06-27 IT IT48580/83A patent/IT1173724B/it active Protection Beyond IP Right Term
- 1983-06-27 PT PT76937A patent/PT76937B/pt unknown
- 1983-06-27 IL IL69081A patent/IL69081A/xx not_active IP Right Cessation
- 1983-06-27 NZ NZ204714A patent/NZ204714A/xx unknown
- 1983-06-27 DK DK198302951A patent/DK172475B1/da not_active IP Right Cessation
- 1983-06-27 GB GB08317365A patent/GB2125398B/en not_active Expired
- 1983-06-27 CY CY1500A patent/CY1500A/xx unknown
- 1983-06-28 AT AT2358/83A patent/AT391136B/de not_active IP Right Cessation
- 1983-06-28 HU HU832335A patent/HU191053B/hu unknown
-
1984
- 1984-06-24 CH CH904/84A patent/CH669792A5/de not_active IP Right Cessation
-
1985
- 1985-08-12 GB GB08520188A patent/GB2166728B/en not_active Expired
- 1985-08-12 GB GB08520186A patent/GB2166726B/en not_active Expired
- 1985-08-12 GB GB08520187A patent/GB2166727B/en not_active Expired
-
1987
- 1987-11-25 US US07/125,048 patent/US4803199A/en not_active Expired - Lifetime
- 1987-12-10 AU AU82434/87A patent/AU603399B2/en not_active Expired
-
1988
- 1988-06-24 CH CH3305/88A patent/CH669954A5/de not_active IP Right Cessation
- 1988-11-15 US US07/272,030 patent/US4910207A/en not_active Expired - Lifetime
-
1989
- 1989-08-23 SG SG537/89A patent/SG53789G/en unknown
-
1990
- 1990-01-17 US US07/466,550 patent/US5017582A/en not_active Expired - Lifetime
- 1990-08-09 HK HK606/90A patent/HK60690A/xx not_active IP Right Cessation
-
1997
- 1997-06-02 NL NL970021C patent/NL970021I2/nl unknown
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