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MX377124B - Compuestos heterociclicos y usos de los mismos. - Google Patents

Compuestos heterociclicos y usos de los mismos.

Info

Publication number
MX377124B
MX377124B MX2018003432A MX2018003432A MX377124B MX 377124 B MX377124 B MX 377124B MX 2018003432 A MX2018003432 A MX 2018003432A MX 2018003432 A MX2018003432 A MX 2018003432A MX 377124 B MX377124 B MX 377124B
Authority
MX
Mexico
Prior art keywords
heterocyclic compounds
compound
pharmaceutical compositions
compositions containing
therapeutic uses
Prior art date
Application number
MX2018003432A
Other languages
English (en)
Other versions
MX2018003432A (es
Inventor
Ben Powell
Jiazhong Zhang
Prabha N Ibrahim
Songyuan Shi
Wayne Spevak
Yan Ma
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57113709&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX377124(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of MX2018003432A publication Critical patent/MX2018003432A/es
Publication of MX377124B publication Critical patent/MX377124B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Abstract

En el presente documento se proporcionan compuestos heterocíclicos de la Fórmula (I), composiciones farmacéuticas que contienen este compuesto y sus usos terapéuticos, métodos para su preparación, compuestos intermediarios, composiciones farmacéuticas que contienen este compuesto y sus usos terapéuticos.
MX2018003432A 2015-09-21 2016-09-19 Compuestos heterociclicos y usos de los mismos. MX377124B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562221508P 2015-09-21 2015-09-21
PCT/US2016/052538 WO2017053243A1 (en) 2015-09-21 2016-09-19 Heterocyclic compounds and uses thereof

Publications (2)

Publication Number Publication Date
MX2018003432A MX2018003432A (es) 2018-06-08
MX377124B true MX377124B (es) 2025-03-07

Family

ID=57113709

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