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MX2012013879A - Derivados de hidroxipiridona, composiciones farmceuticas de los mismos y su uso terapeutico para tratar enfermedades proliferativas. - Google Patents

Derivados de hidroxipiridona, composiciones farmceuticas de los mismos y su uso terapeutico para tratar enfermedades proliferativas.

Info

Publication number
MX2012013879A
MX2012013879A MX2012013879A MX2012013879A MX2012013879A MX 2012013879 A MX2012013879 A MX 2012013879A MX 2012013879 A MX2012013879 A MX 2012013879A MX 2012013879 A MX2012013879 A MX 2012013879A MX 2012013879 A MX2012013879 A MX 2012013879A
Authority
MX
Mexico
Prior art keywords
pharmaceutical compositions
therapeutic use
proliferative diseases
treating proliferative
hydroxypyridone derivatives
Prior art date
Application number
MX2012013879A
Other languages
English (en)
Inventor
Kyle W H Chan
Frank Mercurio
Original Assignee
Biotheryx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biotheryx Inc filed Critical Biotheryx Inc
Publication of MX2012013879A publication Critical patent/MX2012013879A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

En la presente se proveen derivados de hidroxipiridona, por ejemplo, un compuesto de la Fórmula (I) y composiciones farmacéuticas de los mismos. También se proveen en la presente métodos de su uso para tratar, prevenir, o disminuir uno o más síntomas de una enfermedad proliferativa.
MX2012013879A 2010-06-01 2011-06-01 Derivados de hidroxipiridona, composiciones farmceuticas de los mismos y su uso terapeutico para tratar enfermedades proliferativas. MX2012013879A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35043110P 2010-06-01 2010-06-01
PCT/US2011/038700 WO2011153197A1 (en) 2010-06-01 2011-06-01 Hydroxypyridone derivatives, pharmaceutical compositions thereof, and their therapeutic use for treating proliferative diseases

Publications (1)

Publication Number Publication Date
MX2012013879A true MX2012013879A (es) 2013-04-03

Family

ID=44533060

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012013879A MX2012013879A (es) 2010-06-01 2011-06-01 Derivados de hidroxipiridona, composiciones farmceuticas de los mismos y su uso terapeutico para tratar enfermedades proliferativas.

Country Status (8)

Country Link
US (2) US8334307B2 (es)
EP (1) EP2576513A1 (es)
JP (1) JP5844354B2 (es)
CN (3) CN103038216A (es)
AU (1) AU2011261499B2 (es)
CA (1) CA2801001A1 (es)
MX (1) MX2012013879A (es)
WO (1) WO2011153197A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20170277149A1 (en) * 2013-10-22 2017-09-28 Lite-On Technology Corporation Control device with automatic adjustment
US9527815B2 (en) 2014-06-18 2016-12-27 Biotheryx, Inc. Hydroxypyridone derivatives, pharmaceutical compositions thereof, and their therapeutic use for treating inflammatory, neurodegenerative, or immune-mediated diseases
GB201420348D0 (en) * 2014-11-17 2014-12-31 Univ Northumbria Newcastle Compounds for treating neurodegenerative diseases
KR20210145787A (ko) 2019-04-02 2021-12-02 알리고스 테라퓨틱스 인코포레이티드 Prmt5를 표적으로 하는 화합물
CN110354121B (zh) * 2019-07-08 2023-05-02 温州医科大学 环吡酮胺在制备治疗肿瘤药物中的应用和包含环吡酮胺的组合药物及用途
CN113603640A (zh) * 2021-08-06 2021-11-05 成都化润药业有限公司 一种羟吡酮乙胺盐的合成方法
CN113588852A (zh) * 2021-08-16 2021-11-02 浙江鼎泰药业股份有限公司 一种高活性透皮贴膏中挥发性成分含量的测定方法
KR20230104423A (ko) * 2021-12-31 2023-07-10 주식회사 케이씨아이 치환된 1-하이드록시-2-피리돈 화합물의 신규한 제조 방법

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Also Published As

Publication number Publication date
US20130072526A1 (en) 2013-03-21
WO2011153197A1 (en) 2011-12-08
CA2801001A1 (en) 2011-12-08
US9273005B2 (en) 2016-03-01
AU2011261499B2 (en) 2015-07-16
CN103038216A (zh) 2013-04-10
JP5844354B2 (ja) 2016-01-13
JP2013528619A (ja) 2013-07-11
US20120022115A1 (en) 2012-01-26
US8334307B2 (en) 2012-12-18
AU2011261499A1 (en) 2013-01-10
EP2576513A1 (en) 2013-04-10
CN104926722A (zh) 2015-09-23
CN104945318A (zh) 2015-09-30

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