[go: up one dir, main page]

KR870001174A - 2-시아노아미노-피리미딘 유도체의 제조방법 - Google Patents

2-시아노아미노-피리미딘 유도체의 제조방법 Download PDF

Info

Publication number
KR870001174A
KR870001174A KR1019860005863A KR860005863A KR870001174A KR 870001174 A KR870001174 A KR 870001174A KR 1019860005863 A KR1019860005863 A KR 1019860005863A KR 860005863 A KR860005863 A KR 860005863A KR 870001174 A KR870001174 A KR 870001174A
Authority
KR
South Korea
Prior art keywords
optionally substituted
cyanamide
pyrimidine derivative
halogen
represents hydrogen
Prior art date
Application number
KR1019860005863A
Other languages
English (en)
Inventor
클루트 요아힘
뮐러 크라우스-헬무트
피스터 테오도르
Original Assignee
에리히 데브리쯔, 권터 슈마허
바이엘 아크티엔 게젤샤프트
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 에리히 데브리쯔, 권터 슈마허, 바이엘 아크티엔 게젤샤프트 filed Critical 에리히 데브리쯔, 권터 슈마허
Publication of KR870001174A publication Critical patent/KR870001174A/ko

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

내용 없음.

Description

2-시아노아미노-피리미딘 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (5)

  1. 일반식(II)의 2-알킬설포닐-피리미딘 유도체를 필요한 경우 촉매존재하, 필요한 경우 산수용체 존재하 및 필요한 경우 희석제의 존재하에 0 내지 150℃에서 시안아미드 또는 시안아미드의 금속염과 반응시킴을 특징으로 하는 일반식(I)의 2-시아노아미노-피리미딘 유도체의 제조방법.
    상기식에서, R1은 수소, 할로겐, 임의로 치환된 알킬 또는 임의로 치환된 알콕시를 나타내며, R2는 수소, 알킬 또는 할로겐을 나타내고, R3는 수소, 할로겐, 임의로 치환된 알킬 또는 임의로 치환된 알콕시를 나타내고, R4는 임의로 치환된 알킬을 나타낸다.
  2. 제1항에 있어서, 반응을 온도 10내지 100℃에서 수행함을 특징으로 하는 방법.
  3. 제1항에 있어서, 비양자성 극성용매를 희석제로 사용함을 특징으로 하는 방법.
  4. 제3항에 있어서, 디메틸포름아미드, 디메틸-아세트아미드, 아세토니트릴 또는 프로피오니트릴을 비양자성 극성용매로 사용함을 특징으로 하는 방법.
  5. 제1항에 있어서, 일반식(II)의 2-알킬설포닐-피리미딘 유도체몰당 1내지 2몰, 바람직하게는 1.1내지 1.5몰의 시안아미드 또는 이에 상응하는 양의 시안아미드 금속염을 사용함을 특징으로 하는 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860005863A 1985-07-20 1986-07-19 2-시아노아미노-피리미딘 유도체의 제조방법 KR870001174A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3525977.9 1985-07-20
DE19853525977 DE3525977A1 (de) 1985-07-20 1985-07-20 Verfahren zur herstellung von 2-cyanamino-pyrimidin-derivaten

Publications (1)

Publication Number Publication Date
KR870001174A true KR870001174A (ko) 1987-03-11

Family

ID=6276289

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019860005863A KR870001174A (ko) 1985-07-20 1986-07-19 2-시아노아미노-피리미딘 유도체의 제조방법

Country Status (8)

Country Link
US (1) US4711959A (ko)
EP (1) EP0209779A2 (ko)
JP (1) JPS6236366A (ko)
KR (1) KR870001174A (ko)
DE (1) DE3525977A1 (ko)
DK (1) DK343386A (ko)
IL (1) IL79438A0 (ko)
ZA (1) ZA865376B (ko)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH04504576A (ja) * 1989-04-17 1992-08-13 ビイク　グルデン　ロンベルク―ヒェーミッシェ　ファブリーク　ゲゼルシャフト　ミット　ベシュレンクテル　ハフツング 新規アリールピリダジン、その製造、使用およびこれを含有する医薬品
EP1577312A1 (en) 2000-06-13 2005-09-21 Basf Aktiengesellschaft Triazolopyrimidine intermediate compounds for fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines
KR20030011894A (ko) * 2000-06-13 2003-02-11 바스프 악티엔게젤샤프트 5-페닐 치환된 2-(시아노아미노)피리미딘 살균제
PL362686A1 (en) 2000-07-21 2004-11-02 Syngenta Participations Ag Process for the preparation of 4,6-dimethoxy-2-(methylsulfonyl)-1,3-pyrimidine
WO2006029904A1 (en) * 2004-09-17 2006-03-23 Basf Aktiengesellschaft Use of 2-substituted pyrimidines for combating nematode diseases of plants

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE624360A (ko) * 1961-10-31
US4199583A (en) * 1970-07-13 1980-04-22 The Upjohn Company Antifungal method, formulations and compounds
DE2501769A1 (de) * 1975-01-17 1976-07-22 Bayer Ag Substituierte pyrimidinyl(thiono)(thiol)-phosphor (phosphon)-saeureester, verfahren zu ihrer herstellung sowie ihre verwendung als insektizide, akarizide und nematozide
DE3334455A1 (de) * 1983-03-04 1984-09-06 Bayer Ag, 5090 Leverkusen Guanidin - derivate

Also Published As

Publication number Publication date
EP0209779A2 (de) 1987-01-28
DE3525977A1 (de) 1987-01-29
DK343386A (da) 1987-01-21
IL79438A0 (en) 1986-10-31
JPS6236366A (ja) 1987-02-17
US4711959A (en) 1987-12-08
ZA865376B (en) 1987-03-25
DK343386D0 (da) 1986-07-18

Similar Documents

Publication Publication Date Title
KR870003989A (ko) 치환 및 이치환 피리딘-2,3-디카르복실레이트의 제조방법과 치환된 니코티네이트의 제조방법
KR870003998A (ko) 퀴나졸린 유도체류의 제조방법
KR840000508A (ko) 4-아닐리노피리미딘 유도체의 제조방법
KR840005098A (ko) 피리딜(옥시/티오) 페녹시 화합물의 제조방법
KR870002056A (ko) 치환된 프로파르길옥시아세토니트릴 유도체의 제조 방법
KR830007638A (ko) 2-구아니디노-4-헤테로아릴티아졸의 제조방법
KR870001174A (ko) 2-시아노아미노-피리미딘 유도체의 제조방법
KR860008144A (ko) 1,3- 디알킬 -2- 이미다졸리디논의 제조방법
KR840006487A (ko) 세팔로스포린의 제조방법
KR830006302A (ko) 신규 피리미딘 유도체의 제조방법
KR840000481A (ko) 페녹시벤조산으로 부터 유도된 제초성 화합물의 제조방법
KR830001948A (ko) 페니실린 설폭사이드의 제조방법
KR830009077A (ko) 푸란 유도체의 제조방법
KR830007580A (ko) 신규 피리미딘 유도체의 제조방법
KR860008987A (ko) 2- 카르복시피라진 4-옥시드의 제조방법
KR840008647A (ko) 대칭 1,4-디하이드로피리딘디카복실 에스테르의 제조방법
KR870003066A (ko) 프로피온 아미딘 유도체의 제조방법
KR860003204A (ko) 디페닐메틸이민 유도체의 제조방법
KR870002110A (ko) 구아니디노티아졸 유도체의 제조방법
KR890002011A (ko) 5-할로 게노-6-아미노-니코틴산 할라이드. 이의 제조방법 및 용도
KR830006180A (ko) 뱃트물감제조용 신규중간물 α-벤즈아미도-5'(또는 8')-할로게노-1, 1'-디안트 리미드류 등의 α-벤즈아미도 -α'-할로게노-1, 1'-디안트리미드류의 제조방법
KR860007245A (ko) 피페라지닐메틸-1,2,4-트리아졸일메틸-카빈올의 제조방법
KR890009823A (ko) 2-(4-브로모페닐)-2-메틸 프로필 클로라이드의 제조방법
KR840000480A (ko) 페녹시 벤조산류에서 유도된 제초제 화합물류의 제조방법
KR920018016A (ko) 세미카바자이드 및, 폴리아미드 섬유 재료 및 이로부터 수득된 염색물을 안정화시키기 위한 이의 용도

Legal Events

Date Code Title Description
PA0109 Patent application

Patent event code: PA01091R01D

Comment text: Patent Application

Patent event date: 19860719

PG1501 Laying open of application
PC1203 Withdrawal of no request for examination
WITN Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid