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KR830004259A - α-아릴-1H-이미다졸-1-에탄올의 제조방법 - Google Patents

α-아릴-1H-이미다졸-1-에탄올의 제조방법 Download PDF

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Publication number
KR830004259A
KR830004259A KR1019800004332A KR800004332A KR830004259A KR 830004259 A KR830004259 A KR 830004259A KR 1019800004332 A KR1019800004332 A KR 1019800004332A KR 800004332 A KR800004332 A KR 800004332A KR 830004259 A KR830004259 A KR 830004259A
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KR
South Korea
Prior art keywords
carbon atoms
alkyl
compound
formula
hydrogen
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KR1019800004332A
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English (en)
Inventor
케네트 스펜서 호머
Original Assignee
진 크레머, 한스-루돌프 하우스
산도즈 리미티드
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Application filed by 진 크레머, 한스-루돌프 하우스, 산도즈 리미티드 filed Critical 진 크레머, 한스-루돌프 하우스
Publication of KR830004259A publication Critical patent/KR830004259A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/60—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/04—Compounds containing oxirane rings containing only hydrogen and carbon atoms in addition to the ring oxygen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

α-아릴-1H-이미다졸-1-에탄올의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 다음 일반식 Ⅱ화합물과 다음 일반식 Ⅲ화합물을 불활성 유기용매중에서 반응시키거나, 다음 일반식 Ⅰb 화합물의 CH3그룹을 산화시켜 다음 일반식 Ⅰa 화합물을 수득하거나, 다음 일반식 Ⅳ의 알콜로 일반식 Ⅰa 화합물을 에스테르화하여 다음 일반식 Ⅰc 화합물을 수득하는 것을 특징으로하여 다음 일반식 Ⅰ화합물을 제조하는 방법.
    상기에서
    R0는 탄소수 2 내지 6의 알킬, 탄소수 3 내지 6의 시클로알킬, 시클로알킬이 탄소수 3 내지 6이고 알킬이 탄소수 1 내지 3인 시클로알킬알킬인데, 상기의 시클로알킬 및 시클로알킬알킬은 환상에 탄소수 1 내지 3의 알킬그룹 하나 또는 둘로 임의 치환되며,
    R은 수소, 원자번호 9 내지 35의 할로겐, 탄소수 1 내지 4의 알킬, 탄소수 1 내지 4의 알콕시, 탄소수 1 내지 4의 알킬티오 또는 니트로이며,
    R'는 수소, 원자번호 9 내지 35의 할로겐, 탄소수 1 내지 4의 알킬, 탄소수 1 내지 4의 알콕시, 탄소수 1 내지 4의 알킬티오 또는 니트로, A환 3-위치의 -CF3, -CN, -COOR", A환 4위치의 일반식의 임의 치환된 페닐그룹 또는 일반식의 임의 치환된 페녹시그룹이며 R"는 수소 또는 탄소수 1 내지 4의 알킬이거나 R 및 R'는 함께 페닐환 A의 탄소원자상에 치환된 탄소수 1 또는 2의 알킬렌디옥시를 나타내고,
    Y0및 Y는 각각 수소, 원자번호 9 내지 35의 할로겐, 탄소수 1 내지 4의 알킬 또는 탄소수 1 내지 4의 알콕시이며, 단 R0가 n-부틸이면
    a) 최소한 R 및 R'중 하나는수소가 아니며
    b) R 또는 R'는 할로가 아니어야 하며
    X는 알칼리금속이고
    AlK는 C1-C4알킬이며 일반식 Ⅳ의 AlK는 C1-C4알킬이거나 그의 반응성의 관능성 유도체이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019800004332A 1979-11-13 1980-11-12 α-아릴-1H-이미다졸-1-에탄올의 제조방법 KR830004259A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9380079A 1979-11-13 1979-11-13
US93800 1998-06-09

Publications (1)

Publication Number Publication Date
KR830004259A true KR830004259A (ko) 1983-07-09

Family

ID=22240802

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019800004332A KR830004259A (ko) 1979-11-13 1980-11-12 α-아릴-1H-이미다졸-1-에탄올의 제조방법

Country Status (4)

Country Link
JP (1) JPS5686167A (ko)
KR (1) KR830004259A (ko)
BE (1) BE886127A (ko)
ZA (1) ZA807053B (ko)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2946956A1 (de) * 1979-11-21 1981-06-19 Bayer Ag, 5090 Leverkusen Hydroxybutyl-imidazol-derivate, verfahren zu ihrer herstellung sowie ihre verwendung als fungizide
CN1008735B (zh) * 1984-11-02 1990-07-11 拜尔公司 以取代的氮杂茂基甲基-环丙基-甲醇衍生物为活性成分的组合物
JP2539261B2 (ja) * 1987-12-09 1996-10-02 エスエス製薬株式会社 イミダゾ―ル誘導体
JP2006347882A (ja) * 2003-09-02 2006-12-28 Ss Pharmaceut Co Ltd ベンジルアルコール誘導体又はその塩
AR100743A1 (es) * 2014-06-06 2016-10-26 Basf Se Compuestos de [1,2,4]triazol sustituido

Also Published As

Publication number Publication date
ZA807053B (en) 1982-06-30
BE886127A (fr) 1981-05-13
JPS5686167A (en) 1981-07-13

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