JPS5470265A - Substituted indolinone and its preparation - Google Patents
Substituted indolinone and its preparationInfo
- Publication number
- JPS5470265A JPS5470265A JP13495277A JP13495277A JPS5470265A JP S5470265 A JPS5470265 A JP S5470265A JP 13495277 A JP13495277 A JP 13495277A JP 13495277 A JP13495277 A JP 13495277A JP S5470265 A JPS5470265 A JP S5470265A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- indolinone
- amino
- dichlorophenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Indole Compounds (AREA)
Abstract
NEW MATERIAL:1-(4-amino-2,6-dichlorophenyl) indolinone of formula I.
USE: An intermediate for 2-(2,6-dichloroanilino) phenylacetic acid useful as a raw material for medicines having pharmacological action, e.g. anti-inflammatory, analgesic, and antipyretic actions.
PROCESS: The amino group of 2,6-dichloro-4-nitroaniline is diazotized to give a diazonium salt, which is substituted by halogen, e.g. I, Br, Cl, etc. to form 2,6- dichloro-4-nitrohalobenzene (A). The compound (A) is reacted with aniline to form the compound of formula II, which is reacted with oxalyl chloride to form the compound of formula III. The compound of formula III is converted to the compound of formula IV by the Friedel-Crafts reaction. The compound of the formula IV is reduced to give 1-(4-amino-2,6-dichlorophenyl) indolinone via the compound of formula V.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP13495277A JPS5470265A (en) | 1977-11-10 | 1977-11-10 | Substituted indolinone and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP13495277A JPS5470265A (en) | 1977-11-10 | 1977-11-10 | Substituted indolinone and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5470265A true JPS5470265A (en) | 1979-06-05 |
Family
ID=15140395
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP13495277A Pending JPS5470265A (en) | 1977-11-10 | 1977-11-10 | Substituted indolinone and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5470265A (en) |
-
1977
- 1977-11-10 JP JP13495277A patent/JPS5470265A/en active Pending
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