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IT1243404B - Derivati della partricina - Google Patents

Derivati della partricina

Info

Publication number
IT1243404B
IT1243404B IT02226890A IT2226890A IT1243404B IT 1243404 B IT1243404 B IT 1243404B IT 02226890 A IT02226890 A IT 02226890A IT 2226890 A IT2226890 A IT 2226890A IT 1243404 B IT1243404 B IT 1243404B
Authority
IT
Italy
Prior art keywords
derivatives
partricin
same
basic nitrogen
group
Prior art date
Application number
IT02226890A
Other languages
English (en)
Other versions
IT9022268A1 (it
IT9022268A0 (it
Inventor
Tiberio Bruzzese
Massimo Signorini
Franco Ottoni
Original Assignee
Prodotti Antibiotici Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Prodotti Antibiotici Spa filed Critical Prodotti Antibiotici Spa
Publication of IT9022268A0 publication Critical patent/IT9022268A0/it
Priority to IT02226890A priority Critical patent/IT1243404B/it
Priority to EP91119817A priority patent/EP0489308B1/en
Priority to AT91119817T priority patent/ATE170529T1/de
Priority to DE69130107T priority patent/DE69130107T2/de
Priority to ES91119817T priority patent/ES2119750T3/es
Priority to KR1019910021700A priority patent/KR100205933B1/ko
Priority to US07/801,253 priority patent/US5298495A/en
Priority to JP03347995A priority patent/JP3113880B2/ja
Publication of IT9022268A1 publication Critical patent/IT9022268A1/it
Application granted granted Critical
Publication of IT1243404B publication Critical patent/IT1243404B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Compounds Of Unknown Constitution (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT02226890A 1990-12-03 1990-12-03 Derivati della partricina IT1243404B (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IT02226890A IT1243404B (it) 1990-12-03 1990-12-03 Derivati della partricina
ES91119817T ES2119750T3 (es) 1990-12-03 1991-11-21 Derivados de partricina.
AT91119817T ATE170529T1 (de) 1990-12-03 1991-11-21 Partricinderivate
DE69130107T DE69130107T2 (de) 1990-12-03 1991-11-21 Partricinderivate
EP91119817A EP0489308B1 (en) 1990-12-03 1991-11-21 Partricin derivatives
KR1019910021700A KR100205933B1 (ko) 1990-12-03 1991-11-29 파트리신 유도체
US07/801,253 US5298495A (en) 1990-12-03 1991-12-03 Partricin derivatives
JP03347995A JP3113880B2 (ja) 1990-12-03 1991-12-03 パートリシン誘導体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02226890A IT1243404B (it) 1990-12-03 1990-12-03 Derivati della partricina

Publications (3)

Publication Number Publication Date
IT9022268A0 IT9022268A0 (it) 1990-12-03
IT9022268A1 IT9022268A1 (it) 1992-06-04
IT1243404B true IT1243404B (it) 1994-06-10

Family

ID=11193919

Family Applications (1)

Application Number Title Priority Date Filing Date
IT02226890A IT1243404B (it) 1990-12-03 1990-12-03 Derivati della partricina

Country Status (8)

Country Link
US (1) US5298495A (it)
EP (1) EP0489308B1 (it)
JP (1) JP3113880B2 (it)
KR (1) KR100205933B1 (it)
AT (1) ATE170529T1 (it)
DE (1) DE69130107T2 (it)
ES (1) ES2119750T3 (it)
IT (1) IT1243404B (it)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1283149B1 (it) * 1996-07-12 1998-04-07 Prodotti Antibiotici Spa Complessi di n'-dimetilaminoacetilpartricina a dimetilaminoetilamide, o suoi sali, e colesterol 3-solfato
EP0829486A2 (de) * 1996-08-19 1998-03-18 Hoechst Aktiengesellschaft Neue Polyenantibiotika, 3874 H1 bis H6, Verfahren zu ihrer Herstellung und Verwendung
IT1294740B1 (it) * 1997-09-16 1999-04-12 Prospa Bv Derivati della partricina per il trattamento profilattico e/o curativo delle contaminazioni fungine di colture cellulari e di tessuti
US6121244A (en) * 1997-09-19 2000-09-19 Prospa B.V. Antitumoral method by administration of partricin derivatives
IT1295042B1 (it) * 1997-09-19 1999-04-27 Prospa Bv Uso di derivati della partricina nelle terapie antitumorali
IT1301807B1 (it) * 1998-06-25 2000-07-07 Tiberio Bruzzese Formulazioni farmaceutiche iniettabili di derivati della partricina.
CA2394833A1 (en) 2000-01-14 2001-07-19 Binh T. Dang Derivatives of polyene macrolides and preparation and use thereof
US6664241B2 (en) * 2000-05-31 2003-12-16 Micrologix Biotech Inc. Water-soluble amide derivatives of polyene macrolides and preparation and uses thereof
ITMI20032280A1 (it) * 2003-11-24 2005-05-25 Tiberio Bruzzese Formulazioni farmaceutiche contenenti derivati della partricina e loro uso orale per il trattamento di infezioni fungine e protozoarie localizzate
MX365184B (es) * 2010-12-21 2019-05-21 Centro De Investig Y De Estudios Avanzados Del I P N Nuevos compuestos analogos de la anfotericina y composiciones farmaceuticas que los contienen.
US20240317791A1 (en) * 2021-07-12 2024-09-26 Bioseutica B.V. A process for the production of amcipatricin diascorbate and the use of the same for the treatment of invasive fungal infections resistant to traditional antifungal agents
KR102444918B1 (ko) 2022-07-21 2022-09-22 주식회사 삼우에코 에어나이프의 전후진 장치

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1406774A (en) * 1973-02-15 1975-09-17 Prodotti Antibiotici Spa Esters of patricin and of partricin derivatives
PL122086B1 (en) * 1979-04-09 1982-06-30 Politechnika Gdanska Process for preparing amides of antibiotics from the group of polyene macrolides and their derivativesvykh makrolidov i ikh proizvodnykh
FR2654339B1 (fr) * 1989-11-14 1994-10-28 Mayoly Spindler Laboratoires Nouveaux derives solubles et non toxiques des macrolides polyeniques basiques, leur preparation et leurs applications.
IT1237772B (it) * 1989-11-16 1993-06-17 Tiberio Bruzzese Derivati di macrolidi polienici.
EP0431874A1 (en) * 1989-12-08 1991-06-12 Beecham Group p.l.c. Novel compounds
EP0431870A1 (en) * 1989-12-08 1991-06-12 Beecham Group p.l.c. Amphotericin B derivatives

Also Published As

Publication number Publication date
DE69130107T2 (de) 1999-01-21
EP0489308A1 (en) 1992-06-10
JPH04300892A (ja) 1992-10-23
IT9022268A1 (it) 1992-06-04
KR920012105A (ko) 1992-07-25
KR100205933B1 (ko) 1999-07-01
JP3113880B2 (ja) 2000-12-04
IT9022268A0 (it) 1990-12-03
ATE170529T1 (de) 1998-09-15
US5298495A (en) 1994-03-29
DE69130107D1 (de) 1998-10-08
EP0489308B1 (en) 1998-09-02
ES2119750T3 (es) 1998-10-16

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19971125