HK1052012A1 - 16, 17-Carbocyclic condensed steroid compounds having selective estrogenic activity. - Google Patents

16, 17-Carbocyclic condensed steroid compounds having selective estrogenic activity.

Info

Publication number: HK1052012A1
Authority: HK; Hong Kong
Prior art keywords: alkenyl; alkyl; alkynyl; group; mdash
Prior art date: 2000-06-06

Application number

HK03104310A

Other languages

English (en)

Inventor

Hubert Jan Jozef Loozen

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-06

Filing date

2003-06-17

Publication date

2003-08-29

2003-06-17 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2003-08-29 Publication of HK1052012A1 publication Critical patent/HK1052012A1/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C07J53/002—Carbocyclic rings fused
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Physical Education & Sports Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Gynecology & Obstetrics (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

HK03104310A 2000-06-06 2003-06-17 16, 17-Carbocyclic condensed steroid compounds having selective estrogenic activity. HK1052012A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP00201986		2000-06-06
PCT/EP2001/004868 WO2002000682A1 (en)	2000-06-06	2001-05-01	16, 17-carbocyclic condensed steroid compounds having selective estrogenic activity

Publications (1)

Publication Number	Publication Date
HK1052012A1 true HK1052012A1 (en)	2003-08-29

Family

ID=8171601

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HK03104310A HK1052012A1 (en)	2000-06-06	2003-06-17	16, 17-Carbocyclic condensed steroid compounds having selective estrogenic activity.

Country Status (27)

Country	Link
US (3)	US7868193B2 (de)
EP (1)	EP1294739B1 (de)
JP (1)	JP5095902B2 (de)
KR (1)	KR100769865B1 (de)
CN (1)	CN1235908C (de)
AR (1)	AR028080A1 (de)
AT (1)	ATE293124T1 (de)
AU (2)	AU5838601A (de)
BR (1)	BR0111445A (de)
CA (1)	CA2410220C (de)
CZ (1)	CZ20024014A3 (de)
DE (1)	DE60110069T2 (de)
DK (1)	DK1294739T3 (de)
ES (1)	ES2240454T3 (de)
HK (1)	HK1052012A1 (de)
HU (1)	HUP0301190A3 (de)
IL (1)	IL152957A0 (de)
MX (1)	MXPA02012117A (de)
NO (1)	NO324247B1 (de)
PE (1)	PE20020214A1 (de)
PL (1)	PL203732B1 (de)
PT (1)	PT1294739E (de)
RU (1)	RU2255090C2 (de)
SK (1)	SK286852B6 (de)
TW (1)	TWI225068B (de)
WO (1)	WO2002000682A1 (de)
ZA (1)	ZA200209452B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW201109346A (en) *	2009-06-10	2011-03-16	Organon Nv	Substituted 16,17-annellated steroid compounds for use in women's healthcare
US8367648B2 (en)	2009-06-10	2013-02-05	Msd Oss B.V.	Substituted 16,17-annellated steroid compounds for use in womens healthcare

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3194821A (en) *	1963-12-30	1965-07-13	Abbott Lab	17alpha-substituted 17beta-hydroxyestrenes
CA2200423C (en)	1996-03-26	2006-12-19	Sietse Mosselman	Novel estrogen receptor
IL123195A (en) *	1997-02-21	2002-11-10	Akzo Nobel Nv	Steroid compounds with anti-pregnancy activity and against bone thinning, preparation and pharmaceutical preparations containing them

2001
- 2001-04-17 TW TW090109186A patent/TWI225068B/zh not_active IP Right Cessation
- 2001-05-01 HU HU0301190A patent/HUP0301190A3/hu unknown
- 2001-05-01 CA CA002410220A patent/CA2410220C/en not_active Expired - Fee Related
- 2001-05-01 RU RU2002135594/04A patent/RU2255090C2/ru not_active IP Right Cessation
- 2001-05-01 ES ES01931676T patent/ES2240454T3/es not_active Expired - Lifetime
- 2001-05-01 KR KR1020027016657A patent/KR100769865B1/ko not_active IP Right Cessation
- 2001-05-01 PL PL359238A patent/PL203732B1/pl not_active IP Right Cessation
- 2001-05-01 IL IL15295701A patent/IL152957A0/xx not_active IP Right Cessation
- 2001-05-01 AT AT01931676T patent/ATE293124T1/de active
- 2001-05-01 DE DE60110069T patent/DE60110069T2/de not_active Expired - Lifetime
- 2001-05-01 AU AU5838601A patent/AU5838601A/xx active Pending
- 2001-05-01 DK DK01931676T patent/DK1294739T3/da active
- 2001-05-01 CN CNB018107451A patent/CN1235908C/zh not_active Expired - Fee Related
- 2001-05-01 EP EP01931676A patent/EP1294739B1/de not_active Expired - Lifetime
- 2001-05-01 SK SK1707-2002A patent/SK286852B6/sk not_active IP Right Cessation
- 2001-05-01 WO PCT/EP2001/004868 patent/WO2002000682A1/en active IP Right Grant
- 2001-05-01 AU AU2001258386A patent/AU2001258386B2/en not_active Ceased
- 2001-05-01 MX MXPA02012117A patent/MXPA02012117A/es active IP Right Grant
- 2001-05-01 PT PT01931676T patent/PT1294739E/pt unknown
- 2001-05-01 JP JP2002505804A patent/JP5095902B2/ja not_active Expired - Fee Related
- 2001-05-01 CZ CZ20024014A patent/CZ20024014A3/cs unknown
- 2001-05-01 BR BR0111445-0A patent/BR0111445A/pt not_active IP Right Cessation
- 2001-05-01 US US10/297,706 patent/US7868193B2/en not_active Expired - Fee Related
- 2001-05-03 PE PE2001000401A patent/PE20020214A1/es not_active Application Discontinuation
- 2001-05-04 AR ARP010102107A patent/AR028080A1/es unknown
2002
- 2002-11-20 ZA ZA200209452A patent/ZA200209452B/en unknown
- 2002-12-02 NO NO20025793A patent/NO324247B1/no not_active IP Right Cessation
2003
- 2003-06-17 HK HK03104310A patent/HK1052012A1/xx not_active IP Right Cessation
2010
- 2010-06-15 US US12/816,058 patent/US20100249083A1/en not_active Abandoned
2011
- 2011-05-20 US US13/112,184 patent/US20110224183A1/en not_active Abandoned

Also Published As

Publication number	Publication date
DE60110069T2 (de)	2005-09-22
HUP0301190A2 (hu)	2003-08-28
CA2410220A1 (en)	2002-01-03
CN1433426A (zh)	2003-07-30
HUP0301190A3 (en)	2010-03-29
MXPA02012117A (es)	2003-06-06
WO2002000682A1 (en)	2002-01-03
SK17072002A3 (sk)	2003-06-03
US20100249083A1 (en)	2010-09-30
US7868193B2 (en)	2011-01-11
AR028080A1 (es)	2003-04-23
KR20030028752A (ko)	2003-04-10
DE60110069D1 (de)	2005-05-19
CN1235908C (zh)	2006-01-11
SK286852B6 (sk)	2009-06-05
AU5838601A (en)	2002-01-08
PL203732B1 (pl)	2009-11-30
JP2004501931A (ja)	2004-01-22
BR0111445A (pt)	2003-06-03
NO324247B1 (no)	2007-09-17
TWI225068B (en)	2004-12-11
IL152957A0 (en)	2003-06-24
ES2240454T3 (es)	2005-10-16
DK1294739T3 (da)	2005-08-01
CA2410220C (en)	2009-04-28
NO20025793L (no)	2002-12-02
AU2001258386B2 (en)	2005-08-18
EP1294739A1 (de)	2003-03-26
US20040102426A1 (en)	2004-05-27
PT1294739E (pt)	2005-06-30
ZA200209452B (en)	2004-02-20
NO20025793D0 (no)	2002-12-02
EP1294739B1 (de)	2005-04-13
PL359238A1 (en)	2004-08-23
ATE293124T1 (de)	2005-04-15
KR100769865B1 (ko)	2007-10-25
JP5095902B2 (ja)	2012-12-12
US20110224183A1 (en)	2011-09-15
CZ20024014A3 (cs)	2003-04-16
RU2255090C2 (ru)	2005-06-27
PE20020214A1 (es)	2002-03-13

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Legal Events

Date	Code	Title	Description
2011-12-16	PC	Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)	Effective date: 20110501