ATE293124T1 - 16,17-carbocyclisch kondensierte steroid- verbindungen mit selektiver östrogenischer wirksamkeit - Google Patents

16,17-carbocyclisch kondensierte steroid- verbindungen mit selektiver östrogenischer wirksamkeit

Info

Publication number: ATE293124T1
Authority: AT; Austria
Prior art keywords: estrogenic activity; steroid compounds; selective estrogenic; carbocyclic condensed; carbocyclic
Prior art date: 2000-06-06

Application number

AT01931676T

Other languages

English (en)

Inventor

Hubert Jan Jozef Loozen

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-06

Filing date

2001-05-01

Publication date

2005-04-15

2001-05-01 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2005-04-15 Application granted granted Critical

2005-04-15 Publication of ATE293124T1 publication Critical patent/ATE293124T1/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C07J53/002—Carbocyclic rings fused
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Physical Education & Sports Medicine (AREA)
Reproductive Health (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Gynecology & Obstetrics (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

AT01931676T 2000-06-06 2001-05-01 16,17-carbocyclisch kondensierte steroid- verbindungen mit selektiver östrogenischer wirksamkeit ATE293124T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP00201986		2000-06-06
PCT/EP2001/004868 WO2002000682A1 (en)	2000-06-06	2001-05-01	16, 17-carbocyclic condensed steroid compounds having selective estrogenic activity

Publications (1)

Publication Number	Publication Date
ATE293124T1 true ATE293124T1 (de)	2005-04-15

Family

ID=8171601

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01931676T ATE293124T1 (de)	2000-06-06	2001-05-01	16,17-carbocyclisch kondensierte steroid- verbindungen mit selektiver östrogenischer wirksamkeit

Country Status (27)

Country	Link
US (3)	US7868193B2 (de)
EP (1)	EP1294739B1 (de)
JP (1)	JP5095902B2 (de)
KR (1)	KR100769865B1 (de)
CN (1)	CN1235908C (de)
AR (1)	AR028080A1 (de)
AT (1)	ATE293124T1 (de)
AU (2)	AU2001258386B2 (de)
BR (1)	BR0111445A (de)
CA (1)	CA2410220C (de)
CZ (1)	CZ20024014A3 (de)
DE (1)	DE60110069T2 (de)
DK (1)	DK1294739T3 (de)
ES (1)	ES2240454T3 (de)
HK (1)	HK1052012A1 (de)
HU (1)	HUP0301190A3 (de)
IL (1)	IL152957A0 (de)
MX (1)	MXPA02012117A (de)
NO (1)	NO324247B1 (de)
PE (1)	PE20020214A1 (de)
PL (1)	PL203732B1 (de)
PT (1)	PT1294739E (de)
RU (1)	RU2255090C2 (de)
SK (1)	SK286852B6 (de)
TW (1)	TWI225068B (de)
WO (1)	WO2002000682A1 (de)
ZA (1)	ZA200209452B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW201109346A (en) *	2009-06-10	2011-03-16	Organon Nv	Substituted 16,17-annellated steroid compounds for use in women's healthcare
US8367648B2 (en)	2009-06-10	2013-02-05	Msd Oss B.V.	Substituted 16,17-annellated steroid compounds for use in womens healthcare

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3194821A (en)	1963-12-30	1965-07-13	Abbott Lab	17alpha-substituted 17beta-hydroxyestrenes
CA2200423C (en)	1996-03-26	2006-12-19	Sietse Mosselman	Novel estrogen receptor
TW403736B (en) *	1997-02-21	2000-09-01	Akzo Nobel Nv	Steroid compounds having contraceptive and anti-osteoporosis activity

2001
- 2001-04-17 TW TW090109186A patent/TWI225068B/zh not_active IP Right Cessation
- 2001-05-01 CZ CZ20024014A patent/CZ20024014A3/cs unknown
- 2001-05-01 AU AU2001258386A patent/AU2001258386B2/en not_active Ceased
- 2001-05-01 WO PCT/EP2001/004868 patent/WO2002000682A1/en active IP Right Grant
- 2001-05-01 JP JP2002505804A patent/JP5095902B2/ja not_active Expired - Fee Related
- 2001-05-01 AU AU5838601A patent/AU5838601A/xx active Pending
- 2001-05-01 HU HU0301190A patent/HUP0301190A3/hu unknown
- 2001-05-01 PL PL359238A patent/PL203732B1/pl not_active IP Right Cessation
- 2001-05-01 BR BR0111445-0A patent/BR0111445A/pt not_active IP Right Cessation
- 2001-05-01 IL IL15295701A patent/IL152957A0/xx not_active IP Right Cessation
- 2001-05-01 KR KR1020027016657A patent/KR100769865B1/ko not_active IP Right Cessation
- 2001-05-01 SK SK1707-2002A patent/SK286852B6/sk not_active IP Right Cessation
- 2001-05-01 MX MXPA02012117A patent/MXPA02012117A/es active IP Right Grant
- 2001-05-01 AT AT01931676T patent/ATE293124T1/de active
- 2001-05-01 EP EP01931676A patent/EP1294739B1/de not_active Expired - Lifetime
- 2001-05-01 RU RU2002135594/04A patent/RU2255090C2/ru not_active IP Right Cessation
- 2001-05-01 CN CNB018107451A patent/CN1235908C/zh not_active Expired - Fee Related
- 2001-05-01 CA CA002410220A patent/CA2410220C/en not_active Expired - Fee Related
- 2001-05-01 US US10/297,706 patent/US7868193B2/en not_active Expired - Fee Related
- 2001-05-01 DK DK01931676T patent/DK1294739T3/da active
- 2001-05-01 ES ES01931676T patent/ES2240454T3/es not_active Expired - Lifetime
- 2001-05-01 DE DE60110069T patent/DE60110069T2/de not_active Expired - Lifetime
- 2001-05-01 PT PT01931676T patent/PT1294739E/pt unknown
- 2001-05-03 PE PE2001000401A patent/PE20020214A1/es not_active Application Discontinuation
- 2001-05-04 AR ARP010102107A patent/AR028080A1/es unknown
2002
- 2002-11-20 ZA ZA200209452A patent/ZA200209452B/en unknown
- 2002-12-02 NO NO20025793A patent/NO324247B1/no not_active IP Right Cessation
2003
- 2003-06-17 HK HK03104310A patent/HK1052012A1/xx not_active IP Right Cessation
2010
- 2010-06-15 US US12/816,058 patent/US20100249083A1/en not_active Abandoned
2011
- 2011-05-20 US US13/112,184 patent/US20110224183A1/en not_active Abandoned

Also Published As

Publication number	Publication date
RU2255090C2 (ru)	2005-06-27
KR100769865B1 (ko)	2007-10-25
PL359238A1 (en)	2004-08-23
AR028080A1 (es)	2003-04-23
CA2410220C (en)	2009-04-28
AU2001258386B2 (en)	2005-08-18
SK286852B6 (sk)	2009-06-05
HK1052012A1 (en)	2003-08-29
ES2240454T3 (es)	2005-10-16
HUP0301190A3 (en)	2010-03-29
JP5095902B2 (ja)	2012-12-12
NO324247B1 (no)	2007-09-17
US20110224183A1 (en)	2011-09-15
SK17072002A3 (sk)	2003-06-03
BR0111445A (pt)	2003-06-03
CZ20024014A3 (cs)	2003-04-16
IL152957A0 (en)	2003-06-24
US7868193B2 (en)	2011-01-11
PL203732B1 (pl)	2009-11-30
NO20025793D0 (no)	2002-12-02
US20100249083A1 (en)	2010-09-30
CA2410220A1 (en)	2002-01-03
CN1433426A (zh)	2003-07-30
PT1294739E (pt)	2005-06-30
PE20020214A1 (es)	2002-03-13
TWI225068B (en)	2004-12-11
EP1294739B1 (de)	2005-04-13
MXPA02012117A (es)	2003-06-06
WO2002000682A1 (en)	2002-01-03
US20040102426A1 (en)	2004-05-27
DE60110069T2 (de)	2005-09-22
DE60110069D1 (de)	2005-05-19
JP2004501931A (ja)	2004-01-22
ZA200209452B (en)	2004-02-20
CN1235908C (zh)	2006-01-11
NO20025793L (no)	2002-12-02
HUP0301190A2 (hu)	2003-08-28
AU5838601A (en)	2002-01-08
EP1294739A1 (de)	2003-03-26
KR20030028752A (ko)	2003-04-10
DK1294739T3 (da)	2005-08-01

Publication	Publication Date	Title
LU93311I2 (fr)	2017-01-26	Mancozèbe, valifenalate
ATE353909T1 (de)	2007-03-15	3-stickstoff-6,7-dioxygenierte steroid verbindungen und verwendungen davon
DE60111734D1 (de)	2005-08-04	[1,4']-bipiperidin verbindungen
BR0011935B1 (pt)	2010-06-15	aparelho de cortar tubulação.
DE50107988D1 (de)	2005-12-15	Substituierte 1,2,3,4-tetrahydrochinolin-2-carbonsäurederivate
NO20013860D0 (no)	2001-08-08	16-hydroksyostratriener som selektive ostrogener
ID26909A (id)	2001-02-15	Turunan-turunan 1,3,4-oksadiazolon
ATE317396T1 (de)	2006-02-15	14,15-beta-methylen substituierte androgene
HK1069171A1 (en)	2005-05-13	Substituted 6H-dibenzioÄc,hÜchromenes as estrogenic agents.
DK2067772T3 (da)	2011-07-18	Dibenz[b,f]azapin-mellemprodukter
DK1280784T3 (da)	2007-10-29	Biologisk aktive 4H-benzo[1,4]oxazin-3-oner
ATE293124T1 (de)	2005-04-15	16,17-carbocyclisch kondensierte steroid- verbindungen mit selektiver östrogenischer wirksamkeit
ITBO990671A0 (it)	1999-12-10	Maniglione antipanico.
ITGE990045A0 (it)	1999-04-27	Appaia calze.
ES1043131Y (es)	2000-05-01	Tejido perfeccionado.
DK0973790T3 (da)	2003-09-22	Estra-5(10),7-diener med østrogen aktivitet
DE69932256D1 (de)	2006-08-17	Elektroluminiszierendes, organisches element
DE59909590D1 (de)	2004-07-01	Azidfreie, gaserzeugende zusammensetzung
IT247441Y1 (it)	2002-08-22	Maniglione antipanico .
ES1046730Y (es)	2001-06-16	Lavadora perfeccionada.
ES1045500Y (es)	2001-03-01	Celosia graduable.
ES1039658Y (es)	2000-11-01	Celosia antivandalica.
ES1039123Y (es)	1999-03-16	Inodoro canino.
ES1040397Y (es)	1999-08-16	Expendedor de canutillos sorbedores perfeccionado.
ES1040614Y (es)	1999-10-16	Corbata preanudada.

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