FR2930941B1 - Derives d'azetidines, leur preparation et leur application en therapeutique - Google Patents

Derives d'azetidines, leur preparation et leur application en therapeutique

Info

Publication number: FR2930941B1
Authority: FR; France
Prior art keywords: preparation; therapeutic use; azetidine derivatives; azetidine; derivatives
Prior art date: 2008-05-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Application number

FR0802492A

Other languages

English (en)

Other versions

FR2930941A1 (fr

Inventor

Jean Francois Sabuco

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sanofi Aventis France

Original Assignee

Sanofi Aventis France

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-05-06

Filing date

2008-05-06

Publication date

2010-06-18

2008-05-06 Priority to FR0802492A priority Critical patent/FR2930941B1/fr

2008-05-06 Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France

2008-12-16 Priority to PT88729520T priority patent/PT2234966E/pt

2008-12-16 Priority to CN200880126985.5A priority patent/CN101945852B/zh

2008-12-16 Priority to BRPI0822054-9A priority patent/BRPI0822054A2/pt

2008-12-16 Priority to CA2709863A priority patent/CA2709863A1/fr

2008-12-16 Priority to EA201070758A priority patent/EA019315B1/ru

2008-12-16 Priority to ARP080105459A priority patent/AR069700A1/es

2008-12-16 Priority to SI200831115T priority patent/SI2234966T1/sl

2008-12-16 Priority to PE2008002084A priority patent/PE20091270A1/es

2008-12-16 Priority to KR1020107015774A priority patent/KR20100098563A/ko

2008-12-16 Priority to ES08872952.0T priority patent/ES2439258T3/es

2008-12-16 Priority to DK08872952.0T priority patent/DK2234966T3/da

2008-12-16 Priority to JP2010538830A priority patent/JP5460614B2/ja

2008-12-16 Priority to PCT/FR2008/001748 priority patent/WO2009106708A2/fr

2008-12-16 Priority to AU2008351943A priority patent/AU2008351943B2/en

2008-12-16 Priority to PL08872952T priority patent/PL2234966T3/pl

2008-12-16 Priority to EP08872952.0A priority patent/EP2234966B1/fr

2008-12-17 Priority to PA20088808101A priority patent/PA8808101A1/es

2008-12-17 Priority to CL2008003780A priority patent/CL2008003780A1/es

2008-12-18 Priority to TW097149442A priority patent/TW200930360A/zh

2008-12-18 Priority to UY31548A priority patent/UY31548A1/es

2009-11-13 Publication of FR2930941A1 publication Critical patent/FR2930941A1/fr

2010-06-16 Priority to IL206420A priority patent/IL206420A/en

2010-06-18 Priority to CO10073795A priority patent/CO6290755A2/es

2010-06-18 Priority to US12/818,274 priority patent/US8445478B2/en

2010-06-18 Application granted granted Critical

2010-06-18 Publication of FR2930941B1 publication Critical patent/FR2930941B1/fr

2010-07-14 Priority to MA33018A priority patent/MA32019B1/fr

2011-06-15 Priority to HK11106128.9A priority patent/HK1152038A1/xx

2013-04-23 Priority to US13/868,602 priority patent/US20130237513A1/en

2013-12-10 Priority to HRP20131168AT priority patent/HRP20131168T1/hr

2013-12-11 Priority to CY20131101118T priority patent/CY1114991T1/el

Status Expired - Fee Related legal-status Critical Current

2028-05-06 Anticipated expiration legal-status Critical

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Rheumatology (AREA)
Ophthalmology & Optometry (AREA)
Immunology (AREA)
Heart & Thoracic Surgery (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Cardiology (AREA)
Hematology (AREA)
Obesity (AREA)
Pain & Pain Management (AREA)
Endocrinology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pulmonology (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

FR0802492A 2007-12-18 2008-05-06 Derives d'azetidines, leur preparation et leur application en therapeutique Expired - Fee Related FR2930941B1 (fr)

Priority Applications (29)

Application Number	Priority Date	Filing Date	Title
FR0802492A FR2930941B1 (fr)	2008-05-06	2008-05-06	Derives d'azetidines, leur preparation et leur application en therapeutique
CN200880126985.5A CN101945852B (zh)	2007-12-18	2008-12-16	氮杂环丁烷衍生物、其制备和其在治疗中的应用
BRPI0822054-9A BRPI0822054A2 (pt)	2007-12-18	2008-12-16	Derivados de azetidinas, o respectivo preparo e a respectiva aplicação em terapêutica
CA2709863A CA2709863A1 (fr)	2007-12-18	2008-12-16	Derives d'azetidines, leur preparation et leur application en therapeutique
EA201070758A EA019315B1 (ru)	2007-12-18	2008-12-16	Производные азетидинов, их получение и применение в терапии
ARP080105459A AR069700A1 (es)	2007-12-18	2008-12-16	Derivados de azetidina,composiciones farmaceuticas que los comprenden, metodo de preparacion, intermediarios de sintesis,y usos de los mismos en el tratamiento o prevencion de trastornos psiquiatricos , del sistema inmune y gastrointestinales, entre otros.
SI200831115T SI2234966T1 (sl)	2007-12-18	2008-12-16	Derivati azetidinov, njihova priprava in njihova terapevtska uporaba
PE2008002084A PE20091270A1 (es)	2007-12-18	2008-12-16	Derivados de azetidinas con actividad sobre receptores cb1 y su preparacion
KR1020107015774A KR20100098563A (ko)	2007-12-18	2008-12-16	아제티딘 유도체, 그의 제법 및 치료에서의 그의 적용
ES08872952.0T ES2439258T3 (es)	2007-12-18	2008-12-16	Derivados de azetidina, su preparación y su aplicación en terapia
DK08872952.0T DK2234966T3 (da)	2007-12-18	2008-12-16	Azetidinderivater, fremstilling og terapeutisk anvendelse heraf
JP2010538830A JP5460614B2 (ja)	2007-12-18	2008-12-16	アゼチジン誘導体、それらの調製、およびそれらの治療における適用
PCT/FR2008/001748 WO2009106708A2 (fr)	2007-12-18	2008-12-16	Derives d'azetidines, leur preparation et leur application en therapeutique
AU2008351943A AU2008351943B2 (en)	2007-12-18	2008-12-16	Azetidine derivatives, their preparation and their application in therapy
PT88729520T PT2234966E (pt)	2007-12-18	2008-12-16	Derivados de azetidinas, sua preparação e sua aplicação em terapia
EP08872952.0A EP2234966B1 (fr)	2007-12-18	2008-12-16	Derives d'azetidines, leur preparation et leur application en therapeutique
PL08872952T PL2234966T3 (pl)	2007-12-18	2008-12-16	Pochodne azetydyn, ich wytwarzanie i zastosowanie ich w lecznictwie
PA20088808101A PA8808101A1 (es)	2007-12-18	2008-12-17	Derivados de azetidinas, su preparacion y su aplicacion en terapeutica
CL2008003780A CL2008003780A1 (es)	2007-12-18	2008-12-17	Compuestos derivados de azetidinas; procedimiento de preparacion; compuestos intermediarios; composicion farmaceutica; y uso para el tratamiento o la prevencion de trastornos psiquiatricos, dependencia o deshabituacion a una sustancia, trastornos cognitivos, enfermedades neurodegenerativas, entre otras.
TW097149442A TW200930360A (en)	2007-12-18	2008-12-18	Azetidine derivatives, preparation thereof and therapeutic use thereof
UY31548A UY31548A1 (es)	2007-12-18	2008-12-18	Derivados de azetidinas, su preparacion y su aplicacion en terapéutica
IL206420A IL206420A (en)	2007-12-18	2010-06-16	Aztidine derivatives, their preparation, intermediates for their preparation, pharmaceutical preparations containing them and their use in the preparation of medicines
CO10073795A CO6290755A2 (es)	2007-12-18	2010-06-18	Derivados de azetidinas su preparacion y su aplicacion en terapeutica
US12/818,274 US8445478B2 (en)	2007-12-18	2010-06-18	Azetidine derivatives, their preparation and their application in therapy
MA33018A MA32019B1 (fr)	2007-12-18	2010-07-14	Derives d'azetidines, leur preparation et leur application en therapeutique
HK11106128.9A HK1152038A1 (en)	2007-12-18	2011-06-15	Azetidine derivatives, their preparation and their application in therapy
US13/868,602 US20130237513A1 (en)	2007-12-18	2013-04-23	Azetidine derivatives, their preparation and their application in therapy
HRP20131168AT HRP20131168T1 (hr)	2007-12-18	2013-12-10	Derivati azetidina, njihovo dobivanje i njihova terapijska primjena
CY20131101118T CY1114991T1 (el)	2007-12-18	2013-12-11	Παραγωγα αζετιδινων, ο τροπος παρασκευης τους και η εφαρμογη τους στη θεραπευτικη

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0802492A FR2930941B1 (fr)	2008-05-06	2008-05-06	Derives d'azetidines, leur preparation et leur application en therapeutique

Publications (2)

Publication Number	Publication Date
FR2930941A1 FR2930941A1 (fr)	2009-11-13
FR2930941B1 true FR2930941B1 (fr)	2010-06-18

Family

ID=40225389

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FR0802492A Expired - Fee Related FR2930941B1 (fr)	2007-12-18	2008-05-06	Derives d'azetidines, leur preparation et leur application en therapeutique

Country Status (1)

Country	Link
FR (1)	FR2930941B1 (fr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2805817B1 (fr) *	2000-03-03	2002-04-26	Aventis Pharma Sa	Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation

2008
- 2008-05-06 FR FR0802492A patent/FR2930941B1/fr not_active Expired - Fee Related

Also Published As

Publication number	Publication date
FR2930941A1 (fr)	2009-11-13

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FR2910473B1 (fr)	2009-02-13	Derives de n-(amino-heteroaryl)-1h-pyrrolopyridine-2- carboxamides, leur preparation et leur application en therapeutique.
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FR2903985B1 (fr)	2008-09-05	Derives de n-(amino-heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique
FR2904316B1 (fr)	2008-09-05	Derives de n-(amino-heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique.
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FR2915199B1 (fr)	2010-01-22	Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.
FR2928149B1 (fr)	2011-01-14	Composes derives d'azetidines, leur preparation et leur application en therapeutique
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MA29017B1 (fr)	2007-11-01	Derives de 2-amido-4-phenylthiazole, leur preparation et leur application en therapeutique
FR2917412B1 (fr)	2009-08-21	Derives de 7-alkynyl, 1,8-naphthyridones, leur preparation et leur application en therapeutique
FR2915197B1 (fr)	2009-06-12	Derives de triazolopyridine-carboxamides, leur preparation et leur application therapeutique.
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FR2934995B1 (fr)	2010-08-27	Composes d'azetidines polysubstitues, leur preparation et leur application en therapeutique
FR2882054B1 (fr)	2007-04-13	Derives de 1,5-diarylpyrrole, leur preparation et leur application en therapeutique
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FR2927625B1 (fr)	2010-03-12	Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique
FR2938537B1 (fr)	2012-10-26	Derives de carbamates d'alkyl-heterocycles, leur preparation et leur application en therapeutique.
FR2940284B1 (fr)	2011-02-18	Derives de 6-cycloamino-2,3-di-pyridinyl-imidazo°1,2-b!- pyridazine,leur preparation et leur application en therapeutique
FR2930249B1 (fr)	2010-05-14	Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique.
FR2888847B1 (fr)	2007-08-31	Derives de n-(heteriaryl)-1-heteorarylalkyl-1h-indole-2- carboxamides, leur preparation et application en therapeutique
FR2925901B1 (fr)	2011-03-04	DERIVES DE N-HETEROCYCLIQUE-IMIDAZO°1,2-a!PYRIDINE-2- CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2925903B1 (fr)	2011-01-21	DERIVES 6-HETEROCYCLIQUE-IMIDAZO°1,2-a!PYRIDINE-2- CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE

Legal Events

Date	Code	Title	Description
2015-05-08	PLFP	Fee payment	Year of fee payment: 8
2017-03-03	ST	Notification of lapse	Effective date: 20170131