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FR1498465A - Procédé pour fabriquer des nouvelles 4, 5, 6, 7-tétrahydro-thiazolo [5, 4-c] pyridines - Google Patents

Procédé pour fabriquer des nouvelles 4, 5, 6, 7-tétrahydro-thiazolo [5, 4-c] pyridines

Info

Publication number
FR1498465A
FR1498465A FR70539A FR70539A FR1498465A FR 1498465 A FR1498465 A FR 1498465A FR 70539 A FR70539 A FR 70539A FR 70539 A FR70539 A FR 70539A FR 1498465 A FR1498465 A FR 1498465A
Authority
FR
France
Prior art keywords
thiazolo
pyridines
tetrahydro
making new
making
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR70539A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Application granted granted Critical
Publication of FR1498465A publication Critical patent/FR1498465A/fr
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/02Preparation by ring-closure or hydrogenation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/86Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/44Acylated amino or imino radicals
    • C07D277/46Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • EFIXED CONSTRUCTIONS
    • E02HYDRAULIC ENGINEERING; FOUNDATIONS; SOIL SHIFTING
    • E02FDREDGING; SOIL-SHIFTING
    • E02F9/00Component parts of dredgers or soil-shifting machines, not restricted to one of the kinds covered by groups E02F3/00 - E02F7/00
    • E02F9/20Drives; Control devices

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Mining & Mineral Resources (AREA)
  • Civil Engineering (AREA)
  • General Engineering & Computer Science (AREA)
  • Structural Engineering (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR70539A 1965-07-23 1966-07-22 Procédé pour fabriquer des nouvelles 4, 5, 6, 7-tétrahydro-thiazolo [5, 4-c] pyridines Expired FR1498465A (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
DET0029055 1965-07-23
DET0032991 1967-01-16
DET0032993 1967-01-16
DET0032992 1967-01-16
DET0032990 1967-01-16
DET0032994 1967-01-16

Publications (1)

Publication Number Publication Date
FR1498465A true FR1498465A (fr) 1967-10-20

Family

ID=27512321

Family Applications (3)

Application Number Title Priority Date Filing Date
FR70538A Expired FR6013M (fr) 1965-07-23 1966-07-22
FR70539A Expired FR1498465A (fr) 1965-07-23 1966-07-22 Procédé pour fabriquer des nouvelles 4, 5, 6, 7-tétrahydro-thiazolo [5, 4-c] pyridines
FR136259A Expired FR94123E (fr) 1965-07-23 1968-01-16 Procédés pour fabriquer de nouvelles 4,5,6,7-tétrahydro-thiazolo[5,4-c]pyridines.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FR70538A Expired FR6013M (fr) 1965-07-23 1966-07-22

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR136259A Expired FR94123E (fr) 1965-07-23 1968-01-16 Procédés pour fabriquer de nouvelles 4,5,6,7-tétrahydro-thiazolo[5,4-c]pyridines.

Country Status (7)

Country Link
BE (1) BE684415A (fr)
BR (1) BR6681517D0 (fr)
DE (1) DE1620508A1 (fr)
ES (9) ES329299A1 (fr)
FR (3) FR6013M (fr)
GB (1) GB1140387A (fr)
NL (2) NL6610324A (fr)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2556725A1 (fr) * 1983-12-16 1985-06-21 Erba Farmitalia Derives de 4,5,6,7-tetrahydrothiazolo (5,4-c) pyridine, procedes pour les preparer et medicament les contenant
DE3609053A1 (de) * 1985-03-23 1986-09-25 Farmitalia Carlo Erba S.p.A., Mailand/Milano Verfahren zur herstellung von kondensierten 2-substituierten thiazolderivaten
US8541592B2 (en) 2005-11-22 2013-09-24 Amgen Inc. Inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4847264A (en) * 1982-07-21 1989-07-11 Rorer Pharmaceutical Corporation Bicyclic nitrogen heterocyclic ethers and thioethers, and their pharmaceutical uses
DE3680929D1 (de) 1985-02-06 1991-09-26 Boehringer Ingelheim Kg Verwendung des 2-amino-6-allyl-5,6,7,8-tetrahydro-4h-thiazolo(4,5-d)azepins zur herstellung eines zur behandlung der parkinsonschen erkrankung bzw. des parkinsonismus geeigneten arzneimittels.
US5060904A (en) * 1987-05-01 1991-10-29 David Hegarty Multi-positionable support stand with movable center of gravity and article holding means
DE69818094T2 (de) * 1997-12-11 2004-07-08 Biochem Pharma Inc., Laval Antivirale verbindungen
SE0001899D0 (sv) * 2000-05-22 2000-05-22 Pharmacia & Upjohn Ab New compounds
RS44304A (en) 2001-11-22 2007-06-04 Biovitrum Ab., Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
AR041952A1 (es) 2002-11-14 2005-06-01 Novartis Ag N-sulfonilaminotiazol
CL2004000553A1 (es) * 2003-03-20 2005-02-04 Actelion Pharmaceuticals Ltd Uso de compuestos derivados de guanidina como antagonistas del receptor de neuropeptido ff; compuestos derivados de guanidina; procedimientos de preparacion; y composicion farmaceutica que los comprende.
CA2773371A1 (fr) 2003-11-12 2005-05-26 Daiichi Sankyo Company, Limited Procede de production de derive de thiazole
EP2379565A1 (fr) * 2008-12-19 2011-10-26 Schering Corporation Dérivés de pipéridine et de pipérazine et leurs méthodes d'utilisation
EP2414340A1 (fr) * 2009-04-03 2012-02-08 Dainippon Sumitomo Pharma Co., Ltd. Composés utilisables pour le traitement de troubles à médiation par le récepteur métabotropique 5 au glutamate et leurs procédés d'utilisation
JP6890179B2 (ja) 2016-12-02 2021-06-18 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft 二環式アミド化合物及びその使用方法
UA125448C2 (uk) 2017-07-14 2022-03-09 Ф. Хоффманн-Ля Рош Аг Біциклічні кетонові сполуки і способи їх застосування
PE20211247A1 (es) * 2017-10-31 2021-07-13 Hoffmann La Roche Sulfonas y sulfoxidos biciclicos y metodos de usos de los mismos
CN109134510A (zh) * 2018-11-13 2019-01-04 井冈山大学 制备2-氨基-5-cbz-4,5,6,7-四氢噻唑并[5,4-c]吡啶的新方法

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2556725A1 (fr) * 1983-12-16 1985-06-21 Erba Farmitalia Derives de 4,5,6,7-tetrahydrothiazolo (5,4-c) pyridine, procedes pour les preparer et medicament les contenant
DE3445192A1 (de) * 1983-12-16 1985-06-27 Farmitalia Carlo Erba S.p.A., Mailand/Milano 4,5,6,7-tetrahydrothiazolo(5,4-c) pyridinderivate, verfahren zu deren hestellung und pharmazeutische mittel
DE3609053A1 (de) * 1985-03-23 1986-09-25 Farmitalia Carlo Erba S.p.A., Mailand/Milano Verfahren zur herstellung von kondensierten 2-substituierten thiazolderivaten
US8541592B2 (en) 2005-11-22 2013-09-24 Amgen Inc. Inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1

Also Published As

Publication number Publication date
ES349321A1 (es) 1969-04-01
ES349318A1 (es) 1969-04-01
BR6681517D0 (pt) 1973-12-27
NL6610324A (fr) 1967-01-24
ES329299A1 (es) 1968-02-16
ES349317A1 (es) 1969-04-01
NL6800589A (fr) 1968-07-17
DE1620508A1 (de) 1969-09-18
FR6013M (fr) 1968-05-06
GB1140387A (en) 1969-01-15
BE684415A (fr) 1967-01-20
ES349319A1 (es) 1969-04-01
ES349314A1 (es) 1969-04-01
FR94123E (fr) 1969-07-04
ES349316A1 (es) 1969-04-01
ES349322A1 (es) 1969-04-01
ES349320A1 (es) 1969-04-01

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