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FI945904A - Mikrorakeina olevat mahasuojatut stabiilit omepratsolikoostumukset ja menetelmä niiden valmistamiseksi - Google Patents

Mikrorakeina olevat mahasuojatut stabiilit omepratsolikoostumukset ja menetelmä niiden valmistamiseksi Download PDF

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Publication number
FI945904A
FI945904A FI945904A FI945904A FI945904A FI 945904 A FI945904 A FI 945904A FI 945904 A FI945904 A FI 945904A FI 945904 A FI945904 A FI 945904A FI 945904 A FI945904 A FI 945904A
Authority
FI
Finland
Prior art keywords
microgranules
stomach
preparation
stable omeprazole
compositions
Prior art date
Application number
FI945904A
Other languages
English (en)
Swedish (sv)
Other versions
FI945904A0 (fi
FI111220B (fi
Inventor
Patrice Debregeas
Gerard Leduc
Original Assignee
Ethypharm Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9430771&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI945904(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ethypharm Sa filed Critical Ethypharm Sa
Publication of FI945904A0 publication Critical patent/FI945904A0/fi
Publication of FI945904A publication Critical patent/FI945904A/fi
Application granted granted Critical
Publication of FI111220B publication Critical patent/FI111220B/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epoxy Resins (AREA)
  • Sampling And Sample Adjustment (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Investigating Or Analyzing Non-Biological Materials By The Use Of Chemical Means (AREA)
FI945904A 1992-06-16 1994-12-15 Menetelmä stabiilin omepratsolimikroraekoostumuksen valmistamiseksi FI111220B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9207249 1992-06-16
FR9207249A FR2692146B1 (fr) 1992-06-16 1992-06-16 Compositions stables de microgranules d'omeprazole gastro-protégés et leur procédé d'obtention.
PCT/FR1993/000582 WO1993025204A1 (fr) 1992-06-16 1993-06-16 Compositions stables de microgranules d'omeprazole gastro-proteges et leur procede d'obtention
FR9300582 1993-06-16

Publications (3)

Publication Number Publication Date
FI945904A0 FI945904A0 (fi) 1994-12-15
FI945904A true FI945904A (fi) 1994-12-15
FI111220B FI111220B (fi) 2003-06-30

Family

ID=9430771

Family Applications (1)

Application Number Title Priority Date Filing Date
FI945904A FI111220B (fi) 1992-06-16 1994-12-15 Menetelmä stabiilin omepratsolimikroraekoostumuksen valmistamiseksi

Country Status (25)

Country Link
US (1) US5385739A (fi)
EP (1) EP0646006B1 (fi)
JP (1) JP3568950B2 (fi)
KR (1) KR100193966B1 (fi)
CN (1) CN1051225C (fi)
AT (1) ATE149835T1 (fi)
AU (1) AU669719B2 (fi)
CA (1) CA2138149C (fi)
CZ (1) CZ287260B6 (fi)
DE (1) DE69308849T2 (fi)
DK (1) DK0646006T3 (fi)
ES (1) ES2052458B1 (fi)
FI (1) FI111220B (fi)
FR (1) FR2692146B1 (fi)
GE (1) GEP20002015B (fi)
GR (2) GR1001535B (fi)
MD (1) MD1472G2 (fi)
MX (1) MX9303612A (fi)
NZ (1) NZ253179A (fi)
PL (1) PL172706B1 (fi)
RU (1) RU2103995C1 (fi)
SK (1) SK280198B6 (fi)
TJ (1) TJ230B (fi)
WO (1) WO1993025204A1 (fi)
ZA (1) ZA934266B (fi)

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US5834002A (en) 1994-05-02 1998-11-10 Josman Laboratories, Inc. Chewing gum containing colloidal bismuth subcitrate
US6426085B1 (en) 1994-05-02 2002-07-30 Josman Laboratories Inc. Use of bismuth-containing compounds in topical oral dosage forms for the treatment of halitosis
US6902738B2 (en) * 1994-05-02 2005-06-07 Josman Laboratories, Inc. Topical oral dosage forms containing bismuth compounds
ES2087823B1 (es) * 1994-07-13 1997-02-16 Estudes Et Richerches Pharma E Formulacion de microgranulos gastroresistentes de omeprazol y su procedimiento de fabricacion.
JP3743519B2 (ja) * 1994-10-18 2006-02-08 コーニンクレッカ フィリップス エレクトロニクス エヌ ヴィ シリコン−酸化物薄層の製造方法
ES2094694B1 (es) * 1995-02-01 1997-12-16 Esteve Quimica Sa Nueva formulacion farmaceuticamente estable de un compuesto de bencimidazol y su proceso de obtencion.
US6379651B1 (en) 1995-02-07 2002-04-30 Josman Laboratories Oral-topical dosage forms for delivering antibacterials/antibiotics to oral cavity to eradicate H. pylori as a concomitant treatment for peptic ulcers and other gastro-intestinal diseases
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US6372784B1 (en) 1995-02-07 2002-04-16 Josman Laboratories, Inc. Bismuth-containing compounds in topical dosage forms for treatment of corneal and dermal wounds
US5547844A (en) * 1995-02-23 1996-08-20 The Regents Of The University Of California Helicobacter pylori bacterial derived factor
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Also Published As

Publication number Publication date
PL172706B1 (en) 1997-11-28
EP0646006B1 (fr) 1997-03-12
GR3023391T3 (en) 1997-08-29
KR940000106A (ko) 1994-01-03
ATE149835T1 (de) 1997-03-15
FI945904A0 (fi) 1994-12-15
SK280198B6 (sk) 1999-09-10
AU4332193A (en) 1994-01-04
SK155194A3 (en) 1997-01-08
MD1472F2 (en) 2000-05-31
ES2052458B1 (es) 1995-01-16
DE69308849D1 (de) 1997-04-17
FR2692146A1 (fr) 1993-12-17
FI111220B (fi) 2003-06-30
FR2692146B1 (fr) 1995-06-02
ZA934266B (en) 1996-02-09
RU94046268A (ru) 1996-10-10
CZ316594A3 (en) 1995-05-17
NZ253179A (en) 1996-05-28
CN1086130A (zh) 1994-05-04
MD1472G2 (ro) 2001-01-31
TJ230B (en) 1999-11-24
US5385739A (en) 1995-01-31
RU2103995C1 (ru) 1998-02-10
MX9303612A (es) 1994-04-29
EP0646006A1 (fr) 1995-04-05
CA2138149C (fr) 2003-08-19
AU669719B2 (en) 1996-06-20
WO1993025204A1 (fr) 1993-12-23
CZ287260B6 (en) 2000-10-11
MD960332A (en) 1998-03-31
GR1001535B (el) 1994-03-31
CA2138149A1 (fr) 1993-12-23
KR100193966B1 (ko) 1999-06-15
DE69308849T2 (de) 1997-09-04
JP3568950B2 (ja) 2004-09-22
JPH07508509A (ja) 1995-09-21
DK0646006T3 (da) 1997-10-13
CN1051225C (zh) 2000-04-12
ES2052458A1 (es) 1994-07-01
GEP20002015B (en) 2000-04-10

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