FI942963L - Imidatsokinatsoliiniyhdisteitä ja niiden valmistus ja käyttö - Google Patents
Imidatsokinatsoliiniyhdisteitä ja niiden valmistus ja käyttö Download PDFInfo
- Publication number
- FI942963L FI942963L FI942963A FI942963A FI942963L FI 942963 L FI942963 L FI 942963L FI 942963 A FI942963 A FI 942963A FI 942963 A FI942963 A FI 942963A FI 942963 L FI942963 L FI 942963L
- Authority
- FI
- Finland
- Prior art keywords
- preparation
- imidazoquinazoline
- compounds
- imidazoquinazoline compounds
- Prior art date
Links
- KJMFQJFNQYWQAV-UHFFFAOYSA-N 3h-imidazo[4,5-h]quinazoline Chemical class C1=NC=NC2=C(NC=N3)C3=CC=C21 KJMFQJFNQYWQAV-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK912042A DK204291D0 (da) | 1991-12-20 | 1991-12-20 | Heterocykliske forbindelser deres fremstilling og anvendelse |
PCT/DK1992/000385 WO1993013103A1 (en) | 1991-12-20 | 1992-12-18 | Imidazoquinazoline compounds and their preparation and use |
Publications (2)
Publication Number | Publication Date |
---|---|
FI942963L true FI942963L (fi) | 1994-06-20 |
FI942963A0 FI942963A0 (fi) | 1994-06-20 |
Family
ID=8109668
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI942963A FI942963A0 (fi) | 1991-12-20 | 1994-06-20 | Imidatsokinatsoliiniyhdisteitä ja niiden valmistus ja käyttö |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0619820A1 (fi) |
JP (1) | JPH07502278A (fi) |
AU (1) | AU673814B2 (fi) |
CA (1) | CA2125854A1 (fi) |
DK (1) | DK204291D0 (fi) |
FI (1) | FI942963A0 (fi) |
IL (1) | IL104099A (fi) |
NO (1) | NO942301L (fi) |
NZ (1) | NZ246558A (fi) |
TW (1) | TW211568B (fi) |
WO (1) | WO1993013103A1 (fi) |
ZA (1) | ZA929770B (fi) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK151890D0 (da) * | 1990-06-22 | 1990-06-22 | Ferrosan As | Heterocykliske forbindelser deres fremstilling og brug |
CN1052724C (zh) * | 1996-07-01 | 2000-05-24 | 瑞安大药厂股份有限公司 | 新的光学活性的2,3-二氢咪唑并[1,2-c]喹唑啉衍生物及其制备方法和用途 |
KR100864364B1 (ko) | 2005-12-13 | 2008-10-17 | 주식회사 엘지화학 | 신규한 이미다조퀴나졸린 유도체, 이의 제조방법 및 이를이용한 유기전기소자 |
EP2125750B1 (en) | 2007-02-26 | 2014-05-21 | Vitae Pharmaceuticals, Inc. | Cyclic urea and carbamate inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
AR069207A1 (es) | 2007-11-07 | 2010-01-06 | Vitae Pharmaceuticals Inc | Ureas ciclicas como inhibidores de la 11 beta - hidroxi-esteroide deshidrogenasa 1 |
CA2708303A1 (en) | 2007-12-11 | 2009-06-18 | Vitae Pharmaceuticals, Inc. | Cyclic urea inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1 |
EP2324017B1 (en) | 2008-07-25 | 2014-12-31 | Boehringer Ingelheim International GmbH | INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1 |
US8114868B2 (en) | 2008-07-25 | 2012-02-14 | Boehringer Ingelheim International Gmbh | Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 |
CA2744946A1 (en) | 2009-02-04 | 2010-08-12 | Boehringer Ingelheim International Gmbh | Cyclic inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1 |
US8680093B2 (en) | 2009-04-30 | 2014-03-25 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
JP5656986B2 (ja) | 2009-06-11 | 2015-01-21 | ヴァイティー ファーマシューティカルズ,インコーポレイテッド | 1,3−オキサジナン−2−オン構造に基づく11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状阻害剤 |
WO2011002910A1 (en) | 2009-07-01 | 2011-01-06 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
US8933072B2 (en) | 2010-06-16 | 2015-01-13 | Vitae Pharmaceuticals, Inc. | Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use |
WO2011161128A1 (en) | 2010-06-25 | 2011-12-29 | Boehringer Ingelheim International Gmbh | Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders |
EP2635268A1 (en) | 2010-11-02 | 2013-09-11 | Boehringer Ingelheim International GmbH | Pharmaceutical combinations for the treatment of metabolic disorders |
WO2022078480A1 (zh) * | 2020-10-16 | 2022-04-21 | 上海迪诺医药科技有限公司 | 三杂环衍生物、其药物组合物及应用 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1297099C (en) * | 1985-10-17 | 1992-03-10 | Frank Watjen | Quinazoline compounds and their preparation and use |
DK155524C (da) * | 1987-03-18 | 1989-09-11 | Ferrosan As | Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse |
DK443589D0 (da) * | 1989-09-08 | 1989-09-08 | Ferrosan As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
DK151890D0 (da) * | 1990-06-22 | 1990-06-22 | Ferrosan As | Heterocykliske forbindelser deres fremstilling og brug |
-
1991
- 1991-12-20 DK DK912042A patent/DK204291D0/da not_active Application Discontinuation
-
1992
- 1992-12-15 IL IL10409992A patent/IL104099A/en not_active IP Right Cessation
- 1992-12-17 ZA ZA929770A patent/ZA929770B/xx unknown
- 1992-12-18 CA CA002125854A patent/CA2125854A1/en not_active Abandoned
- 1992-12-18 AU AU33448/93A patent/AU673814B2/en not_active Ceased
- 1992-12-18 JP JP5511363A patent/JPH07502278A/ja active Pending
- 1992-12-18 NZ NZ246558A patent/NZ246558A/en unknown
- 1992-12-18 WO PCT/DK1992/000385 patent/WO1993013103A1/en not_active Application Discontinuation
- 1992-12-18 TW TW081110173A patent/TW211568B/zh active
- 1992-12-18 EP EP93902092A patent/EP0619820A1/en not_active Withdrawn
-
1994
- 1994-06-17 NO NO942301A patent/NO942301L/no unknown
- 1994-06-20 FI FI942963A patent/FI942963A0/fi not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NZ246558A (en) | 1995-07-26 |
WO1993013103A1 (en) | 1993-07-08 |
IL104099A (en) | 1996-07-23 |
AU673814B2 (en) | 1996-11-28 |
NO942301D0 (no) | 1994-06-17 |
NO942301L (no) | 1994-08-19 |
ZA929770B (en) | 1994-06-17 |
TW211568B (fi) | 1993-08-21 |
EP0619820A1 (en) | 1994-10-19 |
FI942963A0 (fi) | 1994-06-20 |
CA2125854A1 (en) | 1993-07-08 |
JPH07502278A (ja) | 1995-03-09 |
IL104099A0 (en) | 1993-05-13 |
DK204291D0 (da) | 1991-12-20 |
AU3344893A (en) | 1993-07-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |