[go: up one dir, main page]

FI941287A0 - Triatsolokinoksalin-1,4-dioneja ja niiden valmistus ja käyttö - Google Patents

Triatsolokinoksalin-1,4-dioneja ja niiden valmistus ja käyttö

Info

Publication number
FI941287A0
FI941287A0 FI941287A FI941287A FI941287A0 FI 941287 A0 FI941287 A0 FI 941287A0 FI 941287 A FI941287 A FI 941287A FI 941287 A FI941287 A FI 941287A FI 941287 A0 FI941287 A0 FI 941287A0
Authority
FI
Finland
Prior art keywords
triazoloquinoxaline
diones
preparation
Prior art date
Application number
FI941287A
Other languages
English (en)
Swedish (sv)
Other versions
FI106719B (fi
FI941287L (fi
Inventor
Poul Jacobsen
Flemming Elmelund Nielsen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of FI941287A0 publication Critical patent/FI941287A0/fi
Publication of FI941287L publication Critical patent/FI941287L/fi
Application granted granted Critical
Publication of FI106719B publication Critical patent/FI106719B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI941287A 1991-09-20 1994-03-18 Menetelmä terapeuttisesti käyttökelpoisten [1,2,4]triatsolo[4,3-a]kinoksaliini-1,4-dionien ja -4-onien valmistamiseksi FI106719B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DK911624A DK162491D0 (da) 1991-09-20 1991-09-20 Heterocycliske forbindelser, deres fremstilling og farmaceutiske praeparater indeholdende forbindelserne
DK162491 1991-09-20
DK9200271 1992-09-09
PCT/DK1992/000271 WO1993006103A1 (en) 1991-09-20 1992-09-09 Triazoloquinoxalin-1,4-diones and their preparation and use

Publications (3)

Publication Number Publication Date
FI941287A0 true FI941287A0 (fi) 1994-03-18
FI941287L FI941287L (fi) 1994-03-18
FI106719B FI106719B (fi) 2001-03-30

Family

ID=8106648

Family Applications (1)

Application Number Title Priority Date Filing Date
FI941287A FI106719B (fi) 1991-09-20 1994-03-18 Menetelmä terapeuttisesti käyttökelpoisten [1,2,4]triatsolo[4,3-a]kinoksaliini-1,4-dionien ja -4-onien valmistamiseksi

Country Status (13)

Country Link
US (1) US5504085A (fi)
EP (1) EP0633885A1 (fi)
JP (1) JPH07501791A (fi)
AU (1) AU663523B2 (fi)
CA (1) CA2119579A1 (fi)
DK (1) DK162491D0 (fi)
FI (1) FI106719B (fi)
IL (1) IL103160A (fi)
NO (1) NO302368B1 (fi)
NZ (1) NZ244398A (fi)
TW (1) TW210341B (fi)
WO (1) WO1993006103A1 (fi)
ZA (1) ZA927172B (fi)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1041931C (zh) * 1993-05-06 1999-02-03 诺沃-诺迪斯克有限公司 [1,2,4]三唑并[4,3-a]喹喔啉化合物,它们的制备及其应用
EP0750631B1 (en) * 1994-02-14 2000-04-05 Merrell Pharmaceuticals Inc. Novel mercaptoacetylamido 1,3,4,5-tetrahydro-benzo(c)azepin-3-one disulfide derivatives useful as inhibitors of enkephalinase and ace
FR2717812B1 (fr) * 1994-03-28 1996-05-10 Rhone Poulenc Rorer Sa Indeno[1,2-e]pyrazine-4-ones, leur préparation et les médicaments les contenant.
FR2717813B1 (fr) * 1994-03-28 1996-05-10 Rhone Poulenc Rorer Sa Dérivés d'imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, leur préparation et les médicaments les contenant .
FR2717805B1 (fr) * 1994-03-28 1996-05-10 Rhone Poulenc Rorer Sa Dérivés de 5H-indeno[1,2-b]pyrazine-2,3-dione, leur préparation et les médicaments les contenant .
FR2717814B1 (fr) * 1994-03-28 1996-04-26 Rhone Poulenc Rorer Sa Dérivés de 1,2,4-triazolo(4,3-a)pyrazine-4-one, leur préparation et les médicaments les contenant.
FR2722789B1 (fr) * 1994-07-20 1996-08-23 Rhone Poulenc Rorer Sa Derives d'acide imidazo (1,2-a)indeno(1,2-e) pyrazine-2-carboxylique, leur preparation et les medicaments les contenant
ATE190616T1 (de) * 1994-09-16 2000-04-15 Novo Nordisk As (1,2,4)triazolo(4,3-a)chinoxylinonderivate, ihre darstellung und verwendung als antagonisten von ampa-rezeptoren
HUT76802A (en) * 1994-09-16 1997-11-28 Novo Nordisk As [1,2,4]triazolo[4,3-a]quinoxalinone derivatives,process for their preparation and pharmaceutical compositions containing them
US5679680A (en) * 1995-02-16 1997-10-21 Warner-Lambert Company α-substituted hydrazides having calpain inhibitory activity
US5958926A (en) 1996-11-01 1999-09-28 Nitromed, Inc. Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
USRE37234E1 (en) * 1996-11-01 2001-06-19 Nitromed, Inc. Nitrosated and nitrosylated phosphodiestrase inhibitor compounds, compositions and their uses
IL125950A0 (en) * 1997-09-05 1999-04-11 Pfizer Prod Inc Methods of administering ampa receptor antagonists to treat dyskinesias associated with dopamine agonist therapy
US20040152694A1 (en) * 2003-02-04 2004-08-05 Istvan Kurucz Methods and compositions for treating inflammatory disorders of the airways
EP2103613B1 (en) * 2006-12-13 2016-02-17 ASKA Pharmaceutical Co., Ltd. Quinoxaline derivative
EP2338492A1 (en) 2009-12-24 2011-06-29 Universidad del Pais Vasco Methods and compositions for the treatment of alzheimer
CN103097393B (zh) * 2010-09-07 2015-09-16 安斯泰来制药株式会社 喹喔啉化合物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4400382A (en) * 1980-05-09 1983-08-23 Usv Pharmaceutical Corporation Thiazoloquinoxalin-1,4-diones for treating allergy
US4354027A (en) * 1980-05-19 1982-10-12 Usv Pharmaceutical Corporation Triazoloquinoxalin-4-ones
US4623725A (en) * 1982-10-18 1986-11-18 Pfizer Inc. [1,2,4]Triazolo[4,3-a]quinoxaline-4-amine derivatives
US4780464A (en) * 1986-12-08 1988-10-25 Warner-Lambert Company (1,2,4)triazolo(4,3-a)quinoxaline-4-amines
DK160941C (da) * 1988-06-28 1991-10-21 Novo Nordisk As Kondenserede 2,3-dihydroxypyraziner, fremgangsmaade til deres fremstilling og farmaceutiske praeparater, hvori forbindelserne indgaar
US4975430A (en) * 1989-06-16 1990-12-04 The State Of Oregon Acting By And Through The State Board Of Education On Behalf Of The Oregon Health Sciences University CNQX and its analogs as therapeutics for degenerative neural diseases
JP2550456B2 (ja) * 1990-11-06 1996-11-06 山之内製薬株式会社 縮合ピラジン誘導体
PT101004B (pt) * 1991-10-26 1999-10-29 Schering Ag Derivados da quinoxalina, processo para a sua preparacao e composicoes farmaceuticas que os contem
FR2690160A1 (fr) * 1992-04-15 1993-10-22 Rhone Poulenc Rorer Sa Application de dérivés d'acide 2H-1,2,4-benzothiadiazine-1,1-dioxyde-3-carboxylique à la préparation de médicaments, les produits nouveaux, leur préparation et les médicaments les contenant.

Also Published As

Publication number Publication date
WO1993006103A1 (en) 1993-04-01
ZA927172B (en) 1993-03-24
NO940989L (no) 1994-03-18
AU2660092A (en) 1993-04-27
IL103160A (en) 1999-08-17
TW210341B (fi) 1993-08-01
DK162491D0 (da) 1991-09-20
CA2119579A1 (en) 1993-04-01
FI106719B (fi) 2001-03-30
EP0633885A1 (en) 1995-01-18
IL103160A0 (en) 1993-02-21
FI941287L (fi) 1994-03-18
NO940989D0 (no) 1994-03-18
AU663523B2 (en) 1995-10-12
NO302368B1 (no) 1998-02-23
JPH07501791A (ja) 1995-02-23
NZ244398A (en) 1995-02-24
US5504085A (en) 1996-04-02

Similar Documents

Publication Publication Date Title
FI940904L (fi) Oksatsolidiinidionijohdannaiset, niiden valmistus ja käyttö
MX9204301A (es) Acilmercaptoalcanoildipeptidos, metodos de preparacion y su uso terapeutico.
FI941378L (fi) Bentsimidatsoliyhdisteitä, niiden käyttö ja valmistus
FI945281L (fi) Heterosykliset yhdisteet, niiden valmistus ja käyttö
FI943042L (fi) Suuontelossa hajoava valmiste ja sen valmistus
FI955235A0 (fi) Oksatsolidiinionijohdannaiset, niiden valmistus ja käyttö
FI945625L (fi) Indolokarbatsoli-imidit ja niiden käyttö
NL350016I2 (nl) 3-aryl-4-hydroxy-delta#3-dihydrofuranon-en 3-aryl-4-hydroxy-delta#3-dihydrothiofenon-derivaten.
FI892689L (fi) Uusi transaminaasi, sen valmistus ja käyttö
FI953666L (fi) Hetersykliset yhdisteet ja niiden valmistus ja käyttö
FI935887L (fi) Tiatzolidiinidionijohdannaiset, niiden valmistus ja käyttö
FI943912L (fi) Tienopyrimidiinijohdannaiset, niiden valmistus ja käyttö
FI962043L (fi) Substituoidut 5-rengas-heterosyklit, niiden valmistus ja niiden käyttö
FI935897L (fi) Pyridopyrimidiinijohdannaiset, niiden valmistus ja käyttö
FI941287L (fi) Triatsolokinoksalin-1,4-dioneja ja niiden valmistus ja käyttö
FI935801L (fi) Imidatsoliyhdisteitä, niiden valmistus ja käyttö
FI940696L (fi) Uudet pyratsiinijohdannaiset, niiden valmistus ja käyttö
FI944417L (fi) Atsoliyhdisteet, niiden valmistus ja käyttö
FI942963L (fi) Imidatsokinatsoliiniyhdisteitä ja niiden valmistus ja käyttö
FI954229L (fi) Heterosykliset yhdisteet, niiden käyttö ja valmistus
FI945227L (fi) Sykliset heksapeptidit, niiden valmistus ja käyttö
FI935654L (fi) Kondensoituneet heterosykliset yhdisteet, niiden valmistus ja käyttö
FI946076L (fi) Modifioituja Kluyveromyces-hiivoja, valmistus ja käyttö
MX9200706A (es) Composicion y uso.
FI941214L (fi) Bentsimidatsolin johdannaisia, niiden valmistus ja käyttö