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ES2133877T3 - Procedimiento para la fabricacion de derivados de la (4,5)-trans-oxazolidina. - Google Patents

Procedimiento para la fabricacion de derivados de la (4,5)-trans-oxazolidina.

Info

Publication number
ES2133877T3
ES2133877T3 ES96117478T ES96117478T ES2133877T3 ES 2133877 T3 ES2133877 T3 ES 2133877T3 ES 96117478 T ES96117478 T ES 96117478T ES 96117478 T ES96117478 T ES 96117478T ES 2133877 T3 ES2133877 T3 ES 2133877T3
Authority
ES
Spain
Prior art keywords
sup
trans
procedure
oxazolidine
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES96117478T
Other languages
English (en)
Inventor
Hans Hilpert
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
HOFFMANN LA ROCHE
F Hoffmann La Roche AG
Original Assignee
HOFFMANN LA ROCHE
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by HOFFMANN LA ROCHE, F Hoffmann La Roche AG filed Critical HOFFMANN LA ROCHE
Application granted granted Critical
Publication of ES2133877T3 publication Critical patent/ES2133877T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • C07D263/26—Oxygen atoms attached in position 2 with hetero atoms or acyl radicals directly attached to the ring nitrogen atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

LA PRESENTE INVENCION TRATA DE UN PROCEDIMIENTO PARA LA OBTENCION DE (4,5)-TRANS-2-OXO-OXAZOLIDINONAS DE FORMULA (I) EN DONDE R{SUP,1} ES UN GRUPO CARACTERIZADOR DE UN {AL}-AMINOACIDO, R{SUP,2} ES ALQUILO Y R{SUP,3} ES HIDROGENO, UN GRUPO PROTECTOR DE AMINA, AMIDA O URETANO O UN GRUPO DE FORMULA -C(O)-R{SUP,4}, SIENDO R{SUP,4} ALQUILO O UNO O VARIOS {AL}-AMINOACIDOS, QUE ESTAN UNIDOS UNOS CON OTROS MEDIANTE UNO O VARIOS ENLACES AMIDO, MEDIANTE ISOMERIZACION CON UNA BASE FUERTE A PARTIR DE LOS CORRESPONDIENTES COMPUESTOS CIS DE PARTIDA.
ES96117478T 1995-11-06 1996-10-31 Procedimiento para la fabricacion de derivados de la (4,5)-trans-oxazolidina. Expired - Lifetime ES2133877T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH313195 1995-11-06

Publications (1)

Publication Number Publication Date
ES2133877T3 true ES2133877T3 (es) 1999-09-16

Family

ID=4249292

Family Applications (1)

Application Number Title Priority Date Filing Date
ES96117478T Expired - Lifetime ES2133877T3 (es) 1995-11-06 1996-10-31 Procedimiento para la fabricacion de derivados de la (4,5)-trans-oxazolidina.

Country Status (9)

Country Link
US (1) US5670653A (es)
EP (1) EP0771792B1 (es)
JP (1) JP2907781B2 (es)
KR (1) KR100197459B1 (es)
CN (1) CN1152570A (es)
AT (1) ATE180775T1 (es)
DE (1) DE59602077D1 (es)
DK (1) DK0771792T3 (es)
ES (1) ES2133877T3 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1229934B1 (en) 1999-10-01 2014-03-05 Immunogen, Inc. Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents
EP1403257A4 (en) 2001-05-23 2004-10-13 Kaneka Corp METHOD FOR PRODUCING OXAZOLIDINONE DERIVATIVES OF BETA-HYDROXYETHYLAMINE COMPOUNDS AND FOR PRODUCING BETA-HYDROXYETHYLAMINE COMPOUNDS
KR100686117B1 (ko) * 2005-05-04 2007-02-26 엘지전자 주식회사 식기세척기

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5455353A (en) * 1993-03-24 1995-10-03 Hoffmann-La Roche Inc. 4-(benzyl-2-oxo-oxazolidin-5 ylmethyl)N tertbutyl-decahydroisoquinoline-3-carboxamides

Also Published As

Publication number Publication date
CN1152570A (zh) 1997-06-25
US5670653A (en) 1997-09-23
JPH09169744A (ja) 1997-06-30
KR970027061A (ko) 1997-06-24
DE59602077D1 (de) 1999-07-08
ATE180775T1 (de) 1999-06-15
EP0771792B1 (de) 1999-06-02
EP0771792A1 (de) 1997-05-07
DK0771792T3 (da) 1999-11-15
KR100197459B1 (ko) 1999-06-15
JP2907781B2 (ja) 1999-06-21

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