EA201792502A1 - Кабазитаксел и его применение для лечения рака - Google Patents
Кабазитаксел и его применение для лечения ракаInfo
- Publication number
- EA201792502A1 EA201792502A1 EA201792502A EA201792502A EA201792502A1 EA 201792502 A1 EA201792502 A1 EA 201792502A1 EA 201792502 A EA201792502 A EA 201792502A EA 201792502 A EA201792502 A EA 201792502A EA 201792502 A1 EA201792502 A1 EA 201792502A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- kabazitaxel
- applications
- cancer treatment
- cancer
- treatment
- Prior art date
Links
- 206010028980 Neoplasm Diseases 0.000 title abstract 2
- 201000011510 cancer Diseases 0.000 title abstract 2
- BMQGVNUXMIRLCK-OAGWZNDDSA-N cabazitaxel Chemical compound O([C@H]1[C@@H]2[C@]3(OC(C)=O)CO[C@@H]3C[C@@H]([C@]2(C(=O)[C@H](OC)C2=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)C=3C=CC=CC=3)C[C@]1(O)C2(C)C)C)OC)C(=O)C1=CC=CC=C1 BMQGVNUXMIRLCK-OAGWZNDDSA-N 0.000 title 1
- 208000000857 Hepatic Insufficiency Diseases 0.000 abstract 1
- 206010019663 Hepatic failure Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J1/00—Containers specially adapted for medical or pharmaceutical purposes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J2205/00—General identification or selection means
- A61J2205/30—Printed labels
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gastroenterology & Hepatology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
Abstract
Настоящее изобретение относится к соединению, характеризующемуся следующей формулой (I), которое может находиться в форме основания или в форме гидрата или сольвата, для применения в качестве лекарственного препарата при лечении рака у пациентов с печеночной недостаточностью.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP15305720.3A EP3093014A1 (en) | 2015-05-13 | 2015-05-13 | Cabazitaxel and its use for treating cancer |
PCT/EP2016/060759 WO2016180943A1 (en) | 2015-05-13 | 2016-05-12 | Cabazitaxel and its use for treating cancer |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201792502A1 true EA201792502A1 (ru) | 2018-02-28 |
Family
ID=53177311
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201792502A EA201792502A1 (ru) | 2015-05-13 | 2016-05-12 | Кабазитаксел и его применение для лечения рака |
Country Status (15)
Country | Link |
---|---|
US (1) | US20160331717A1 (ru) |
EP (3) | EP3093014A1 (ru) |
JP (1) | JP2018516890A (ru) |
KR (1) | KR20180006417A (ru) |
CN (1) | CN108135878A (ru) |
AU (1) | AU2016259775A1 (ru) |
CA (1) | CA2985408A1 (ru) |
EA (1) | EA201792502A1 (ru) |
ES (1) | ES2774101T3 (ru) |
IL (1) | IL255541A (ru) |
MX (1) | MX2017014463A (ru) |
PL (1) | PL3294285T3 (ru) |
PT (1) | PT3294285T (ru) |
TW (1) | TW201705950A (ru) |
WO (1) | WO2016180943A1 (ru) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3093014A1 (en) | 2015-05-13 | 2016-11-16 | Aventis Pharma S.A. | Cabazitaxel and its use for treating cancer |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5847170A (en) | 1995-03-27 | 1998-12-08 | Rhone-Poulenc Rorer, S.A. | Taxoids, their preparation and pharmaceutical compositions containing them |
MA23823A1 (fr) | 1995-03-27 | 1996-10-01 | Aventis Pharma Sa | Nouveaux taxoides, leur preparation et les compositions qui les contiennent |
ES2248684T3 (es) | 2003-07-02 | 2006-03-16 | Scheuten Glasgroep | Procedimiento para la fabricacion de un acristalamiento contra incendios. |
FR2859996B1 (fr) * | 2003-09-19 | 2006-02-03 | Aventis Pharma Sa | Solvat acetonique du dimethoxy docetaxel et son procede de preparation |
ES2862340T3 (es) | 2009-10-29 | 2021-10-07 | Sanofi Mature Ip | Nuevo uso antitumoral de cabazitaxel |
BR112012012210B8 (pt) * | 2009-11-23 | 2021-05-25 | Cerulean Pharma Inc | conjugado de (cdp)-taxano de polímero contendo ciclodextrina, composição, composição farmacêutica, forma de dosagem, kit e uso de um conjugado de cdp-taxano |
CN103826634A (zh) * | 2011-09-15 | 2014-05-28 | 诺华股份有限公司 | 4-氨基-5-氟-3-[6-(4-甲基哌嗪-1-基)-1h-苯并咪唑-2-基]-1h-喹啉-2-酮在治疗中度肝损伤患者癌症中的应用 |
EP3093014A1 (en) | 2015-05-13 | 2016-11-16 | Aventis Pharma S.A. | Cabazitaxel and its use for treating cancer |
-
2015
- 2015-05-13 EP EP15305720.3A patent/EP3093014A1/en not_active Ceased
-
2016
- 2016-05-12 JP JP2017558939A patent/JP2018516890A/ja active Pending
- 2016-05-12 US US15/153,128 patent/US20160331717A1/en not_active Abandoned
- 2016-05-12 CN CN201680040986.2A patent/CN108135878A/zh active Pending
- 2016-05-12 KR KR1020177035580A patent/KR20180006417A/ko not_active Withdrawn
- 2016-05-12 EP EP16721844.5A patent/EP3294285B1/en not_active Revoked
- 2016-05-12 EA EA201792502A patent/EA201792502A1/ru unknown
- 2016-05-12 EP EP19209255.9A patent/EP3643307A1/en not_active Withdrawn
- 2016-05-12 AU AU2016259775A patent/AU2016259775A1/en not_active Abandoned
- 2016-05-12 MX MX2017014463A patent/MX2017014463A/es unknown
- 2016-05-12 PL PL16721844T patent/PL3294285T3/pl unknown
- 2016-05-12 WO PCT/EP2016/060759 patent/WO2016180943A1/en active Application Filing
- 2016-05-12 ES ES16721844T patent/ES2774101T3/es active Active
- 2016-05-12 PT PT167218445T patent/PT3294285T/pt unknown
- 2016-05-12 CA CA2985408A patent/CA2985408A1/en not_active Abandoned
- 2016-05-13 TW TW105114982A patent/TW201705950A/zh unknown
-
2017
- 2017-11-09 IL IL255541A patent/IL255541A/en unknown
Also Published As
Publication number | Publication date |
---|---|
TW201705950A (zh) | 2017-02-16 |
IL255541A (en) | 2018-01-31 |
AU2016259775A1 (en) | 2018-01-04 |
CA2985408A1 (en) | 2016-11-17 |
EP3093014A1 (en) | 2016-11-16 |
US20160331717A1 (en) | 2016-11-17 |
PT3294285T (pt) | 2020-03-06 |
KR20180006417A (ko) | 2018-01-17 |
EP3294285A1 (en) | 2018-03-21 |
JP2018516890A (ja) | 2018-06-28 |
EP3294285B1 (en) | 2019-12-18 |
ES2774101T3 (es) | 2020-07-16 |
CN108135878A (zh) | 2018-06-08 |
WO2016180943A1 (en) | 2016-11-17 |
PL3294285T3 (pl) | 2020-05-18 |
MX2017014463A (es) | 2018-03-21 |
EP3643307A1 (en) | 2020-04-29 |
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