[go: up one dir, main page]

EA201100757A1 - Способ приготовления гранулята действующих веществ и полученный таким способом гранулят - Google Patents

Способ приготовления гранулята действующих веществ и полученный таким способом гранулят

Info

Publication number
EA201100757A1
EA201100757A1 EA201100757A EA201100757A EA201100757A1 EA 201100757 A1 EA201100757 A1 EA 201100757A1 EA 201100757 A EA201100757 A EA 201100757A EA 201100757 A EA201100757 A EA 201100757A EA 201100757 A1 EA201100757 A1 EA 201100757A1
Authority
EA
Eurasian Patent Office
Prior art keywords
active substances
granules
granulate
preparing
preparing granulate
Prior art date
Application number
EA201100757A
Other languages
English (en)
Inventor
Кристоф Лёбон
Паскаль Сюпли
Original Assignee
Дебрежа Э Ассосье Фарма
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40348849&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201100757(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Дебрежа Э Ассосье Фарма filed Critical Дебрежа Э Ассосье Фарма
Publication of EA201100757A1 publication Critical patent/EA201100757A1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Glanulating (AREA)
  • Fertilizers (AREA)
  • Seasonings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Fodder In General (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Настоящее изобретение относится к способу приготовления гранулята по меньшей мере из двух действующих веществ, включающему этап нанесения упомянутых действующих веществ опудриванием на твердую основу в виде частиц, притом что упомянутые действующие вещества не являются экстрактами растений.
EA201100757A 2008-11-14 2009-11-13 Способ приготовления гранулята действующих веществ и полученный таким способом гранулят EA201100757A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0857764A FR2938432B1 (fr) 2008-11-14 2008-11-14 Nouveau procede de preparation de granules de principes actifs, et granules tels qu'obtenus
PCT/FR2009/052180 WO2010055268A1 (fr) 2008-11-14 2009-11-13 Nouveau procédé de préparation de granulés de principes actifs, et granulés tels qu'obtenus

Publications (1)

Publication Number Publication Date
EA201100757A1 true EA201100757A1 (ru) 2011-12-30

Family

ID=40348849

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201100757A EA201100757A1 (ru) 2008-11-14 2009-11-13 Способ приготовления гранулята действующих веществ и полученный таким способом гранулят

Country Status (25)

Country Link
US (1) US20110280945A1 (ru)
EP (1) EP2349226A1 (ru)
JP (1) JP5608681B2 (ru)
KR (1) KR101585705B1 (ru)
CN (1) CN102223879A (ru)
AR (1) AR074330A1 (ru)
AU (1) AU2009315449B2 (ru)
BR (1) BRPI0916019A2 (ru)
CA (1) CA2743753A1 (ru)
CL (1) CL2011001115A1 (ru)
CO (1) CO6382108A2 (ru)
CU (1) CU20110107A7 (ru)
EA (1) EA201100757A1 (ru)
FR (1) FR2938432B1 (ru)
IL (1) IL212850A0 (ru)
MA (1) MA32789B1 (ru)
MX (1) MX2011005072A (ru)
NZ (1) NZ592857A (ru)
PE (1) PE20110945A1 (ru)
SG (1) SG195651A1 (ru)
TN (1) TN2011000235A1 (ru)
TW (1) TWI522113B (ru)
UA (1) UA103781C2 (ru)
WO (1) WO2010055268A1 (ru)
ZA (1) ZA201103543B (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2971422B1 (fr) 2011-02-11 2016-05-20 Debregeas Et Associes Pharma Granules d'acide gamma-hydroxybutyrique
US9241956B2 (en) * 2012-11-05 2016-01-26 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US20140127296A1 (en) * 2012-11-05 2014-05-08 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US11058635B1 (en) * 2020-10-15 2021-07-13 King Abdulaziz University Oral administration of 5-FU in a gelling nanosuspension for targeted delivery to treat colorectal cancers
KR20240157168A (ko) * 2023-04-24 2024-11-01 주식회사 케이티앤지 바인더를 사용하는 파우치 충진 물질의 제조 방법

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6327424A (ja) * 1986-07-17 1988-02-05 Shionogi & Co Ltd 徐放性製剤およびその製造法
JP2820829B2 (ja) * 1991-03-07 1998-11-05 武田薬品工業株式会社 有核散剤およびその製造方法
JPH08310969A (ja) * 1995-05-22 1996-11-26 Lion Corp 固形薬品組成物及びその製造方法
FR2790668B1 (fr) * 1999-03-12 2002-07-26 D B F Granules contenant une substance vegetale et leur procede de preparation
JP2002544220A (ja) * 1999-05-17 2002-12-24 デー.ベー.エフ. 植物物質を含有する顆粒及びその製造方法
MY148805A (en) * 2002-10-16 2013-05-31 Takeda Pharmaceutical Controlled release preparation
US9247765B2 (en) * 2004-01-14 2016-02-02 Omniactive Health Technologies Limited Stable beadlets of lipophilic nutrients
FR2880541B1 (fr) * 2005-01-10 2008-02-22 Amalric Veret Une nouvelle formule de plantes sous forme de micro-granules de xilitol pour renforcer les effets des plantes et leurs proprietes par une meilleure assimilation
US20060182796A1 (en) * 2005-02-03 2006-08-17 Abrika Pharmaceuticals, Inc. Taste masked pharmaceutical compositions
CA2661683C (en) * 2006-08-31 2015-11-24 Eurand, Inc Drug delivery systems comprising solid solutions of weakly basic drugs
ES2403103T3 (es) * 2007-02-14 2013-05-14 Dainichiseika Color & Chemicals Mfg. Co., Ltd. Agente dispersante para pigmento orgánico y su utilización
US20090004281A1 (en) * 2007-06-26 2009-01-01 Biovail Laboratories International S.R.L. Multiparticulate osmotic delivery system

Also Published As

Publication number Publication date
TWI522113B (zh) 2016-02-21
CN102223879A (zh) 2011-10-19
AU2009315449A1 (en) 2010-05-20
FR2938432A1 (fr) 2010-05-21
IL212850A0 (en) 2011-07-31
JP2012508786A (ja) 2012-04-12
MX2011005072A (es) 2011-10-03
TN2011000235A1 (fr) 2012-12-17
FR2938432B1 (fr) 2011-05-20
SG195651A1 (en) 2013-12-30
AU2009315449B2 (en) 2015-03-26
ZA201103543B (en) 2012-01-25
PE20110945A1 (es) 2012-02-01
CU20110107A7 (es) 2012-01-31
NZ592857A (en) 2013-07-26
KR101585705B1 (ko) 2016-01-15
EP2349226A1 (fr) 2011-08-03
CL2011001115A1 (es) 2011-11-11
MA32789B1 (fr) 2011-11-01
CA2743753A1 (fr) 2010-05-20
UA103781C2 (ru) 2013-11-25
AR074330A1 (es) 2011-01-05
CO6382108A2 (es) 2012-02-15
KR20110095888A (ko) 2011-08-25
JP5608681B2 (ja) 2014-10-15
US20110280945A1 (en) 2011-11-17
TW201029667A (en) 2010-08-16
BRPI0916019A2 (pt) 2015-11-10
WO2010055268A1 (fr) 2010-05-20

Similar Documents

Publication Publication Date Title
EA200970580A1 (ru) Таннат разагилина
CL2012002427A1 (es) Composiciones fertilizante que comprende un granulo del fertilizante de base, un recubrimiento de barrera y uno o mas micronutrientes que cubren al menos una parte de dicho recubrimiento de barrera; y su metodo de fabricacion.
DK1896006T3 (da) Fremstillingmetode for entacapon-holdige granuler til orale doseringsformet
EA200901157A1 (ru) Конденсированные кольцевые гетероциклические модуляторы киназы
EA201170742A1 (ru) Производные n-{[(1r,4s,6r)-3-(2-пиридинилкарбонил)-3-азабицикло[4.1.0]гепт-4-ил]метил}-2-гетероариламинов и их применения
BR112012023044A2 (pt) composições para saúde de planta compreendendo um pesticida solúvel em água e um agroquímico insolúvel em água.
EA201391318A1 (ru) Твердые формы 3-(5-амино-2-метил-4-оксо-4н-хиназолин-3-ил)пиперидин-2,6-диона и их фармацевтические композиции и применение
EA201100758A1 (ru) Гранулят гамма-гидроксимасляной кислоты
CY1111729T1 (el) Υπογλωσσιο επικαλυμμενο δισκιο
CL2008001897A1 (es) Proceso para la preparacion de 3-halometil-1-metil-1h-pirazol, utiles como intermediario en la produccion de fungicidas; compuestos derivados de 3-halometil-1-metil-1h-pirazol.
EA201170396A1 (ru) 2-оксо-1,2-дигидрохинолиновые модуляторы иммунной функции
WO2012010509A3 (de) Gelköder zur bekämpfung von kriechenden schadinsekten
BR112012001048A2 (pt) Composições adjuvantes agrícolas, composições de pesticidas, e métodos de utilização de tais composições.
EA201100757A1 (ru) Способ приготовления гранулята действующих веществ и полученный таким способом гранулят
EA200970126A1 (ru) Способ получения прегабалина и его энантиомера
ECSP13012666A (es) Formulacion en comprimidos difusibles y flotantes de un pesticida
EA201200616A1 (ru) Производные 2-оксо-1-пирролидинилимидазотиадиазола
GEP20156396B (en) Adjuvant comprising dimethylsulfoxide and a phosphate ester
HK1247125A1 (zh) 結晶化合物
HK1222325A1 (zh) 高效的胰酶藥物組合物
EA200901523A1 (ru) Композиция пролонгированного высвобождения, содержащая производное соматостатина в микрочастицах
WO2009059712A3 (de) Homogene und lagerstabile mischungen unterschiedlicher pflanzenschutzmittel-wirkstoff-granulatpartikel
EA200601608A1 (ru) Способ производства твёрдой фармацевтической композиции
TW200621684A (en) Methods for the manufacture of biphenyl amines
MY152388A (en) Composition and method for controlling plant diseases