[go: up one dir, main page]

CO6382108A2 - Nuevo procedimiento de preparacion de granulados de principios activos, y granulados tal como se los ha obtenido - Google Patents

Nuevo procedimiento de preparacion de granulados de principios activos, y granulados tal como se los ha obtenido

Info

Publication number
CO6382108A2
CO6382108A2 CO11059023A CO11059023A CO6382108A2 CO 6382108 A2 CO6382108 A2 CO 6382108A2 CO 11059023 A CO11059023 A CO 11059023A CO 11059023 A CO11059023 A CO 11059023A CO 6382108 A2 CO6382108 A2 CO 6382108A2
Authority
CO
Colombia
Prior art keywords
granulates
active principles
preparation
new procedure
active
Prior art date
Application number
CO11059023A
Other languages
English (en)
Inventor
Christophe Lebon
Pascal Suplie
Original Assignee
Debregeas Et Associes Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40348849&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6382108(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Debregeas Et Associes Pharma filed Critical Debregeas Et Associes Pharma
Publication of CO6382108A2 publication Critical patent/CO6382108A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Glanulating (AREA)
  • Fertilizers (AREA)
  • Fodder In General (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Seasonings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

La presente invención se refiere al campo de la ciencia médica, en particular preparaciones de uso médico en microcápsulas con compuestos orgánicos, un procedimiento de preparación de un granulado de, al menos, dos principios activos, que comprende una etapa de aplicación por polvificado de dichos principios activos sobre un soporte particular sólido, y dichos principios activos no son extractos de plantas. Los granulados obtenidos pueden ser utilizados en el campo farmacéutico.
CO11059023A 2008-11-14 2011-05-13 Nuevo procedimiento de preparacion de granulados de principios activos, y granulados tal como se los ha obtenido CO6382108A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0857764A FR2938432B1 (fr) 2008-11-14 2008-11-14 Nouveau procede de preparation de granules de principes actifs, et granules tels qu'obtenus

Publications (1)

Publication Number Publication Date
CO6382108A2 true CO6382108A2 (es) 2012-02-15

Family

ID=40348849

Family Applications (1)

Application Number Title Priority Date Filing Date
CO11059023A CO6382108A2 (es) 2008-11-14 2011-05-13 Nuevo procedimiento de preparacion de granulados de principios activos, y granulados tal como se los ha obtenido

Country Status (25)

Country Link
US (1) US20110280945A1 (es)
EP (1) EP2349226A1 (es)
JP (1) JP5608681B2 (es)
KR (1) KR101585705B1 (es)
CN (1) CN102223879A (es)
AR (1) AR074330A1 (es)
AU (1) AU2009315449B2 (es)
BR (1) BRPI0916019A2 (es)
CA (1) CA2743753A1 (es)
CL (1) CL2011001115A1 (es)
CO (1) CO6382108A2 (es)
CU (1) CU20110107A7 (es)
EA (1) EA201100757A1 (es)
FR (1) FR2938432B1 (es)
IL (1) IL212850A0 (es)
MA (1) MA32789B1 (es)
MX (1) MX2011005072A (es)
NZ (1) NZ592857A (es)
PE (1) PE20110945A1 (es)
SG (1) SG195651A1 (es)
TN (1) TN2011000235A1 (es)
TW (1) TWI522113B (es)
UA (1) UA103781C2 (es)
WO (1) WO2010055268A1 (es)
ZA (1) ZA201103543B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2971422B1 (fr) * 2011-02-11 2016-05-20 Debregeas Et Associes Pharma Granules d'acide gamma-hydroxybutyrique
US9241956B2 (en) * 2012-11-05 2016-01-26 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US20140127296A1 (en) * 2012-11-05 2014-05-08 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US11058635B1 (en) * 2020-10-15 2021-07-13 King Abdulaziz University Oral administration of 5-FU in a gelling nanosuspension for targeted delivery to treat colorectal cancers
KR20240157168A (ko) * 2023-04-24 2024-11-01 주식회사 케이티앤지 바인더를 사용하는 파우치 충진 물질의 제조 방법

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6327424A (ja) * 1986-07-17 1988-02-05 Shionogi & Co Ltd 徐放性製剤およびその製造法
JP2820829B2 (ja) * 1991-03-07 1998-11-05 武田薬品工業株式会社 有核散剤およびその製造方法
JPH08310969A (ja) * 1995-05-22 1996-11-26 Lion Corp 固形薬品組成物及びその製造方法
FR2790668B1 (fr) * 1999-03-12 2002-07-26 D B F Granules contenant une substance vegetale et leur procede de preparation
DE60026295T2 (de) * 1999-05-17 2006-10-12 D.B.F. Pflanzenmaterial enthaltendes granulat und verfahren zur herstellung
MY148805A (en) * 2002-10-16 2013-05-31 Takeda Pharmaceutical Controlled release preparation
US9247765B2 (en) * 2004-01-14 2016-02-02 Omniactive Health Technologies Limited Stable beadlets of lipophilic nutrients
FR2880541B1 (fr) * 2005-01-10 2008-02-22 Amalric Veret Une nouvelle formule de plantes sous forme de micro-granules de xilitol pour renforcer les effets des plantes et leurs proprietes par une meilleure assimilation
US20060182796A1 (en) * 2005-02-03 2006-08-17 Abrika Pharmaceuticals, Inc. Taste masked pharmaceutical compositions
CA2661683C (en) * 2006-08-31 2015-11-24 Eurand, Inc Drug delivery systems comprising solid solutions of weakly basic drugs
EP2110413B1 (en) * 2007-02-14 2013-03-20 Dainichiseika Color & Chemicals Mfg. Co., Ltd. Dispersing agent for organic pigment and use thereof
US20090004281A1 (en) * 2007-06-26 2009-01-01 Biovail Laboratories International S.R.L. Multiparticulate osmotic delivery system

Also Published As

Publication number Publication date
PE20110945A1 (es) 2012-02-01
AU2009315449B2 (en) 2015-03-26
JP5608681B2 (ja) 2014-10-15
CL2011001115A1 (es) 2011-11-11
CN102223879A (zh) 2011-10-19
NZ592857A (en) 2013-07-26
MA32789B1 (fr) 2011-11-01
FR2938432A1 (fr) 2010-05-21
EP2349226A1 (fr) 2011-08-03
TW201029667A (en) 2010-08-16
TN2011000235A1 (fr) 2012-12-17
AR074330A1 (es) 2011-01-05
EA201100757A1 (ru) 2011-12-30
JP2012508786A (ja) 2012-04-12
BRPI0916019A2 (pt) 2015-11-10
IL212850A0 (en) 2011-07-31
FR2938432B1 (fr) 2011-05-20
UA103781C2 (uk) 2013-11-25
TWI522113B (zh) 2016-02-21
CA2743753A1 (fr) 2010-05-20
KR20110095888A (ko) 2011-08-25
AU2009315449A1 (en) 2010-05-20
SG195651A1 (en) 2013-12-30
CU20110107A7 (es) 2012-01-31
MX2011005072A (es) 2011-10-03
US20110280945A1 (en) 2011-11-17
KR101585705B1 (ko) 2016-01-15
ZA201103543B (en) 2012-01-25
WO2010055268A1 (fr) 2010-05-20

Similar Documents

Publication Publication Date Title
ECSP11011183A (es) Compuestos orgánicos
ECSP11011184A (es) Compuestos orgánicos
CL2015001945A1 (es) (divisional de la solicitud n° 1567-2013) combinaciones de principios activos que comprenden piridiletilbenzamidas y otros principios activos.
ECSP13012482A (es) Derivados de 5-yodo-triazol
CL2009001240A1 (es) Compuestos derivados del acido l-glutamico y l-glutamina marcados con [f-18]; procedimiento de preparacion; composicion farmaceutica que comprende a los compuestos y su uso como agentes en el diagnostico de tumores.
ECSP11011181A (es) Compuestos orgánicos
BR112016007356A2 (pt) compostos herbicidas
UY31069A1 (es) Nuevos derivados de imidazoquinola, composiciones conteniendolos, proceso de preparacion y aplicaciones
CR20140365A (es) Compuestos de carbamato y preparación y uso de los mismos
BR112012019103A2 (pt) compostos de isoxazolina cetônica, composto cetônico, composição agrícola, composição veterinária, uso de um composto, método e material de propagação de planta
DOP2010000259A (es) Derivados heterociclicos de urea y metodos de uso de los mismos-211
UY32648A (es) Nuevos derivados de pirimidina y su uso en el tratamiento de enfermedades
CL2012001366A1 (es) Compuestos derivados de carboxamida n-((2-morfolino-5-ariltiazol-4-il)metil), moduladores de receptores nicotinicos alfa 7; composicion farmaceutica; proceso para prepararla; combinacion farmaceutica; y su uso para el tratamiento de la enfermedad de alzheimer, demencia, esquizofrenia, enfermedad de parkinson, entre otras.
UY33014A (es) Nuevos compuestos de diazinil-pirazolilo
CR11801A (es) Derivados de indazol sustituidos con fenilo y benzodioxinilo
AR081774A1 (es) Composiciones farmaceuticas de co-cristales de tramadol y coxibs
UA106631C2 (uk) Композиції з контрольованим вивільненням
CO6382108A2 (es) Nuevo procedimiento de preparacion de granulados de principios activos, y granulados tal como se los ha obtenido
UY32673A (es) Nuevas pirimidinas, composiciones farmaceuticas que las contienen, procedimientos de preparaciones y su aplicacion como medicamentos
CL2008003274A1 (es) Metod para el tratamiento de cultivos que comprende preparar una solucion de pulverizacion mezclando una composicion agroquimica, glicerol crudo derivado de la produccion de biodiesel y aplicar dicha solucion al acultivo y/o malezas y/o su habitat; la solucion de pulverizacion y uso de dicho glicerol para prepararla.
BRPI1007539A8 (pt) Composto, processo para a preparação do mesmo, composição herbicida, e, método para controlar gramíneas e ervas daninhas em culturas de plantas úteis
BR112013004662B8 (pt) Composto, composição farmacêutica, usos de um composto, e método para preparar uma composição farmacêutica
BR112012009310A2 (pt) composto, e, composição farmacêutica
UY31905A (es) Derivados de benzoxazinona, procesos de preparación, composiciones farmacéuticas conteniéndolos y aplicaciones.
CO6491117A2 (es) Derivados de n1-acil-5-fluoropirimidinona

Legal Events

Date Code Title Description
FC Application refused