DZ2887A1 - Dérivés d'azétidine, leur préparation et les médicaments les contenant. - Google Patents

Dérivés d'azétidine, leur préparation et les médicaments les contenant.

Info

Publication number: DZ2887A1
Authority: DZ; Algeria
Prior art keywords: preparation; drugs containing; azetidine derivatives; azetidine; derivatives
Prior art date: 1998-09-11

Application number

DZ990187A

Other languages

English (en)

Inventor

Daniel Achard

Herve Bouchard

Jean Bouquerel

Marc Capet

Serge Grisoni

Jean-Luc Malleron

Serge Mignani

Augustin Hittinger

Original Assignee

Rhone Poulenc Rorer Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-09-11

Filing date

1999-09-08

Publication date

2003-12-15

1999-09-08 Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa

2003-12-15 Application granted granted Critical

2003-12-15 Publication of DZ2887A1 publication Critical patent/DZ2887A1/fr

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Communicable Diseases (AREA)
Immunology (AREA)
Cardiology (AREA)
Oncology (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Psychology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Ophthalmology & Optometry (AREA)
Addiction (AREA)
Rheumatology (AREA)
Virology (AREA)
Tropical Medicine & Parasitology (AREA)
Obesity (AREA)
Hematology (AREA)
Child & Adolescent Psychology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Endocrinology (AREA)

DZ990187A 1998-09-11 1999-09-08 Dérivés d'azétidine, leur préparation et les médicaments les contenant. DZ2887A1 (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9811342A FR2783246B1 (fr)	1998-09-11	1998-09-11	Derives d'azetidine, leur preparation et les medicaments les contenant

Publications (1)

Publication Number	Publication Date
DZ2887A1 true DZ2887A1 (fr)	2003-12-15

Family

ID=9530327

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DZ990187A DZ2887A1 (fr)	1998-09-11	1999-09-08	Dérivés d'azétidine, leur préparation et les médicaments les contenant.

Country Status (26)

Country	Link
EP (1)	EP1112251B1 (fr)
JP (1)	JP4767413B2 (fr)
CN (1)	CN1149191C (fr)
AR (1)	AR021483A1 (fr)
AT (1)	ATE239703T1 (fr)
AU (1)	AU772025B2 (fr)
BR (1)	BR9913592A (fr)
CA (1)	CA2342739C (fr)
CO (1)	CO5150230A1 (fr)
CZ (1)	CZ301446B6 (fr)
DE (1)	DE69907698T2 (fr)
DK (1)	DK1112251T3 (fr)
DZ (1)	DZ2887A1 (fr)
ES (1)	ES2197666T3 (fr)
FR (1)	FR2783246B1 (fr)
HU (1)	HUP0103341A3 (fr)
MA (1)	MA26685A1 (fr)
MY (1)	MY119150A (fr)
PL (1)	PL198526B1 (fr)
PT (1)	PT1112251E (fr)
RU (1)	RU2230739C2 (fr)
TN (1)	TNSN99168A1 (fr)
TR (1)	TR200100693T2 (fr)
TW (1)	TW530046B (fr)
WO (1)	WO2000015609A1 (fr)
ZA (1)	ZA200102003B (fr)

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ATE478856T1 (de)	2004-01-28	2010-09-15	Hoffmann La Roche	Spirobenzodioxole und deren verwendung als cb1- antagonisten
ATE432275T1 (de)	2004-05-10	2009-06-15	Hoffmann La Roche	Pyrrol- bzw. imidazolamide zur behandlung von obesitas
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BRPI0609685A2 (pt)	2005-04-06	2010-04-20	Hoffmann La Roche	compostos, processo para a sua manufatura, composições farmacêuticas que os compreendem, método para tratamento e/ou profilaxia de enfermidades que estão associados com a modulação de receptores de cb1, e utilização dos mesmos
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BRPI0716134A2 (pt)	2006-09-07	2013-09-17	Nycomed Gmbh	tratamento de combinaÇço para diabetes mellitus
US7781593B2 (en)	2006-09-14	2010-08-24	Hoffmann-La Roche Inc.	5-phenyl-nicotinamide derivatives
JP5508258B2 (ja)	2007-06-04	2014-05-28	ベングリオンユニバーシティオブザネガフリサーチアンドディベロップメントオーソリティ	トリアリール化合物および前記化合物を含む組成物
EP2025674A1 (fr)	2007-08-15	2009-02-18	sanofi-aventis	Tetrahydronaphthaline substituée, son procédé de fabrication et son utilisation en tant que médicament
UY31968A (es)	2008-07-09	2010-01-29	Sanofi Aventis	Nuevos derivados heterocíclicos, sus procesos para su preparación, y sus usos terapéuticos
WO2010068601A1 (fr)	2008-12-08	2010-06-17	Sanofi-Aventis	Hydrate de fluoroglycoside hétéroaromatique cristallin, ses procédés de fabrication, ses procédés d'utilisation et compositions pharmaceutiques le contenant
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WO2012120055A1 (fr)	2011-03-08	2012-09-13	Sanofi	Dérivés oxathiazine di- et tri-substitués, procédé pour leur préparation, utilisation en tant que médicament, agent pharmaceutique contenant ces dérivés et utilisation
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1998
- 1998-09-11 FR FR9811342A patent/FR2783246B1/fr not_active Expired - Fee Related
1999
- 1999-09-01 TW TW088115056A patent/TW530046B/zh not_active IP Right Cessation
- 1999-09-07 MY MYPI99003867A patent/MY119150A/en unknown
- 1999-09-08 TN TNTNSN99168A patent/TNSN99168A1/fr unknown
- 1999-09-08 DZ DZ990187A patent/DZ2887A1/fr active
- 1999-09-08 MA MA25758A patent/MA26685A1/fr unknown
- 1999-09-09 EP EP99941728A patent/EP1112251B1/fr not_active Expired - Lifetime
- 1999-09-09 CA CA002342739A patent/CA2342739C/fr not_active Expired - Fee Related
- 1999-09-09 DK DK99941728T patent/DK1112251T3/da active
- 1999-09-09 AU AU55232/99A patent/AU772025B2/en not_active Ceased
- 1999-09-09 RU RU2001110080/04A patent/RU2230739C2/ru not_active IP Right Cessation
- 1999-09-09 BR BR9913592-2A patent/BR9913592A/pt not_active Application Discontinuation
- 1999-09-09 HU HU0103341A patent/HUP0103341A3/hu unknown
- 1999-09-09 PT PT99941728T patent/PT1112251E/pt unknown
- 1999-09-09 CN CNB99810762XA patent/CN1149191C/zh not_active Expired - Fee Related
- 1999-09-09 TR TR2001/00693T patent/TR200100693T2/xx unknown
- 1999-09-09 AT AT99941728T patent/ATE239703T1/de active
- 1999-09-09 WO PCT/FR1999/002147 patent/WO2000015609A1/fr not_active Application Discontinuation
- 1999-09-09 PL PL346530A patent/PL198526B1/pl not_active IP Right Cessation
- 1999-09-09 JP JP2000570149A patent/JP4767413B2/ja not_active Expired - Fee Related
- 1999-09-09 ES ES99941728T patent/ES2197666T3/es not_active Expired - Lifetime
- 1999-09-09 CZ CZ20010883A patent/CZ301446B6/cs not_active IP Right Cessation
- 1999-09-09 DE DE69907698T patent/DE69907698T2/de not_active Expired - Lifetime
- 1999-09-10 CO CO99057627A patent/CO5150230A1/es unknown
- 1999-09-10 AR ARP990104563A patent/AR021483A1/es active IP Right Grant
2001
- 2001-03-08 ZA ZA200102003A patent/ZA200102003B/en unknown

Also Published As

Publication number	Publication date
CZ301446B6 (cs)	2010-03-03
FR2783246B1 (fr)	2000-11-17
WO2000015609A1 (fr)	2000-03-23
BR9913592A (pt)	2001-06-12
MY119150A (en)	2005-04-30
CA2342739A1 (fr)	2000-03-23
TR200100693T2 (tr)	2001-07-23
JP4767413B2 (ja)	2011-09-07
HUP0103341A3 (en)	2002-10-28
TW530046B (en)	2003-05-01
DE69907698D1 (de)	2003-06-12
CN1149191C (zh)	2004-05-12
ATE239703T1 (de)	2003-05-15
AU772025B2 (en)	2004-04-08
DE69907698T2 (de)	2004-03-25
CN1316991A (zh)	2001-10-10
AU5523299A (en)	2000-04-03
CO5150230A1 (es)	2002-04-29
TNSN99168A1 (fr)	2005-11-10
EP1112251A1 (fr)	2001-07-04
DK1112251T3 (da)	2003-09-01
EP1112251B1 (fr)	2003-05-07
HUP0103341A2 (hu)	2002-02-28
CZ2001883A3 (en)	2001-06-13
ZA200102003B (en)	2002-08-28
MA26685A1 (fr)	2004-12-20
AR021483A1 (es)	2002-07-24
RU2230739C2 (ru)	2004-06-20
ES2197666T3 (es)	2004-01-01
JP2002525267A (ja)	2002-08-13
CA2342739C (fr)	2009-09-08
PT1112251E (pt)	2003-09-30
PL198526B1 (pl)	2008-06-30
PL346530A1 (en)	2002-02-11
FR2783246A1 (fr)	2000-03-17

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