DK533783D0 - 6alfa-methylcortikoider, deres fremstilling og anvendelse - Google Patents

6alfa-methylcortikoider, deres fremstilling og anvendelse

Info

Publication number: DK533783D0
Authority: DK; Denmark
Prior art keywords: 6alfa; preparation; corticoids; methyl; methyl corticoids
Prior art date: 1982-11-22

Application number

DK5337/83A

Other languages

English (en)

Other versions

DK533783A (da

DK159686B (da

DK159686C (da

Inventor

Klaus Annen

Henry Laurent

Helmut Hofmeister

Rudolf Weichert

Hans Wendt

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-11-22

Filing date

1983-11-22

Publication date

1983-11-22

1983-11-22 Application filed by Schering Ag filed Critical Schering Ag

1983-11-22 Publication of DK533783D0 publication Critical patent/DK533783D0/da

1984-05-23 Publication of DK533783A publication Critical patent/DK533783A/da

1990-11-19 Publication of DK159686B publication Critical patent/DK159686B/da

1991-04-15 Application granted granted Critical

1991-04-15 Publication of DK159686C publication Critical patent/DK159686C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0053—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa not substituted in position 16
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/008—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21
- C07J7/0085—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21 by an halogen atom

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pulmonology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines Containing Plant Substances (AREA)
Saccharide Compounds (AREA)
Peptides Or Proteins (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Manufacture Of Tobacco Products (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Detergent Compositions (AREA)
Seasonings (AREA)

DK533783A 1982-11-22 1983-11-22 Analogifremgangsmaade til fremstilling af 6alfa-methylcotikoider DK159686C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19823243482 DE3243482A1 (de)	1982-11-22	1982-11-22	Neue 6(alpha)-methylkortikoide, ihre herstellung und verwendung
DE3243482		1982-11-22

Publications (4)

Publication Number	Publication Date
DK533783D0 true DK533783D0 (da)	1983-11-22
DK533783A DK533783A (da)	1984-05-23
DK159686B DK159686B (da)	1990-11-19
DK159686C DK159686C (da)	1991-04-15

Family

ID=6178924

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK533783A DK159686C (da)	1982-11-22	1983-11-22	Analogifremgangsmaade til fremstilling af 6alfa-methylcotikoider

Country Status (22)

Country	Link
US (1)	US4645763A (da)
EP (1)	EP0110041B1 (da)
JP (1)	JPS59106500A (da)
AT (1)	ATE28651T1 (da)
AU (1)	AU2098983A (da)
BG (2)	BG43867A3 (da)
CA (1)	CA1303607C (da)
CS (1)	CS248712B2 (da)
DD (1)	DD219200A5 (da)
DE (2)	DE3243482A1 (da)
DK (1)	DK159686C (da)
ES (1)	ES8405421A1 (da)
GB (1)	GB2130587A (da)
GR (1)	GR79725B (da)
HU (1)	HU190746B (da)
IE (1)	IE56281B1 (da)
IL (1)	IL70160A (da)
NO (1)	NO157454C (da)
PL (3)	PL141686B1 (da)
PT (1)	PT77408B (da)
RO (2)	RO93593B (da)
ZA (1)	ZA838720B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60161914A (ja) *	1984-02-02	1985-08-23	Green Cross Corp:The	ステロイド脂肪酸エステル含有直腸投与製剤
JPS61274795A (ja) *	1985-05-30	1986-12-04	Toshiba Corp	曝気槽の溶存酸素濃度制御装置
US4968822A (en) *	1987-12-11	1990-11-06	Taisho Pharmaceutical Co., Ltd.	21-alkoxysteroid compounds
EP0523132A1 (en) *	1990-03-27	1993-01-20	Schering Corporation	PROCESS FOR 9$g(a)-HYDROXY STEROID DEHYDRATION
DE4333920A1 (de) *	1993-10-05	1995-04-13	Hoechst Ag	Corticoid-17,21-dicarbonsäureester sowie Corticosteroid-17-carbonsäureester-21-kohlensäureester, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
ITMI20011762A1 (it)	2001-08-10	2003-02-10	Cosmo Spa	Esteri di 17alfa,21-diidrossipregnene, loro uso come agenti anti-androgenetici e procedimenti per la loro preparazione
ITMI20071616A1 (it)	2007-08-03	2009-02-04	Cosmo Spa	Processo enzimatico per l'ottenimento di 17-alfa monoesteri del cortexolone e/o suoi 9,11-deidroderivati.
MX2010012976A (es)	2008-05-28	2011-05-31	Validus Genetics	Moduladores de nf-kb esteroides no hormonales para el tratamiento de enfermedades.
US9198921B2 (en)	2010-04-05	2015-12-01	Reveragen Biopharma, Inc.	Non-hormonal steroid modulators of NF-κB for treatment of disease
EP3108879A1 (en)	2015-06-25	2016-12-28	Cassiopea S.p.A.	High concentration formulation
US10799514B2 (en)	2015-06-29	2020-10-13	Reveragen Biopharma, Inc.	Non-hormonal steroid modulators of NF-kappa beta for treatment of disease
US11382922B2 (en)	2019-03-07	2022-07-12	Reveragen Biopharma, Inc.	Aqueous oral pharmaceutical suspension compositions

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3053832A (en) *	1957-04-29	1962-09-11	Schering Corp	Alkylated cortical steroids
GB921533A (en) *	1958-07-12	1963-03-20	Syntex Sa	Cyclopentanophenanthrene derivatives and process for the production thereof
GB1047518A (en) *	1963-06-11	1966-11-02	Glaxo Lab Ltd	17ª-monoesters of 11,17,21-trihydroxy steroid compounds
DE2645104C2 (de) *	1976-10-04	1986-04-24	Schering AG, 1000 Berlin und 4709 Bergkamen	11β-Hydroxy-1,4,8-pregnatrien-3,20-dion-Derivate und Verfahren zu ihrer Herstellung
US4243586A (en) *	1980-01-18	1981-01-06	E. R. Squibb & Sons, Inc.	Steroidal-17-spiro-dihydrofuranones
US4318853A (en) *	1980-01-31	1982-03-09	The Upjohn Company	9β,11β-Epoxy-5β-corticoids
US4336200A (en) *	1980-01-31	1982-06-22	The Upjohn Company	17α-Acyloxy-5β-corticoids
ATE12237T1 (de) *	1980-12-23	1985-04-15	Schering Ag	Neue 6-alpha-methylhydrocortison-derivate, ihre herstellung und verwendung.

1982
- 1982-11-22 DE DE19823243482 patent/DE3243482A1/de not_active Withdrawn
1983
- 1983-09-20 EP EP83109308A patent/EP0110041B1/de not_active Expired
- 1983-09-20 DE DE8383109308T patent/DE3372776D1/de not_active Expired
- 1983-09-20 AT AT83109308T patent/ATE28651T1/de not_active IP Right Cessation
- 1983-09-28 PT PT77408A patent/PT77408B/pt not_active IP Right Cessation
- 1983-10-13 ES ES526446A patent/ES8405421A1/es not_active Expired
- 1983-10-17 GB GB08327736A patent/GB2130587A/en not_active Withdrawn
- 1983-11-04 AU AU20989/83A patent/AU2098983A/en not_active Abandoned
- 1983-11-08 IL IL70160A patent/IL70160A/xx not_active IP Right Cessation
- 1983-11-18 DD DD83256872A patent/DD219200A5/de not_active IP Right Cessation
- 1983-11-21 PL PL1983250735A patent/PL141686B1/pl unknown
- 1983-11-21 PL PL1983244685A patent/PL138796B1/pl unknown
- 1983-11-21 HU HU834000A patent/HU190746B/hu not_active IP Right Cessation
- 1983-11-21 RO RO122112A patent/RO93593B/ro unknown
- 1983-11-21 GR GR73030A patent/GR79725B/el unknown
- 1983-11-21 NO NO834265A patent/NO157454C/no unknown
- 1983-11-21 CA CA000441605A patent/CA1303607C/en not_active Expired - Lifetime
- 1983-11-21 IE IE2708/83A patent/IE56281B1/en not_active IP Right Cessation
- 1983-11-21 RO RO83112614A patent/RO89343A/ro unknown
- 1983-11-21 PL PL25073483A patent/PL250734A1/xx unknown
- 1983-11-22 JP JP58218852A patent/JPS59106500A/ja active Granted
- 1983-11-22 DK DK533783A patent/DK159686C/da active
- 1983-11-22 ZA ZA838720A patent/ZA838720B/xx unknown
- 1983-11-22 BG BG070923A patent/BG43867A3/xx unknown
- 1983-11-22 BG BG063156A patent/BG42677A3/xx unknown
- 1983-11-22 US US06/554,418 patent/US4645763A/en not_active Expired - Lifetime
- 1983-11-22 CS CS838675A patent/CS248712B2/cs unknown

Also Published As

Publication number	Publication date
EP0110041A1 (de)	1984-06-13
IE56281B1 (en)	1991-06-05
RO89343A (ro)	1986-03-15
BG42677A3 (en)	1988-01-15
NO157454B (no)	1987-12-14
PT77408A (de)	1983-10-01
IL70160A0 (en)	1984-02-29
ES526446A0 (es)	1984-06-16
DK533783A (da)	1984-05-23
PT77408B (de)	1986-02-27
PL250735A1 (en)	1985-07-30
IE832708L (en)	1984-05-22
PL141686B1 (en)	1987-08-31
AU2098983A (en)	1984-05-31
PL138796B1 (en)	1986-11-29
PL244685A1 (en)	1985-04-24
IL70160A (en)	1988-03-31
PL250734A1 (en)	1985-07-30
ES8405421A1 (es)	1984-06-16
CS248712B2 (en)	1987-02-12
RO93593A (ro)	1987-12-31
HU190746B (en)	1986-10-28
EP0110041B1 (de)	1987-07-29
DE3243482A1 (de)	1984-05-24
DE3372776D1 (en)	1987-09-03
ATE28651T1 (de)	1987-08-15
NO834265L (no)	1984-05-23
BG43867A3 (en)	1988-08-15
ZA838720B (en)	1984-07-25
JPS59106500A (ja)	1984-06-20
JPH0415799B2 (da)	1992-03-19
GR79725B (da)	1984-10-31
NO157454C (no)	1988-03-23
RO93593B (ro)	1988-01-01
DD219200A5 (de)	1985-02-27
CA1303607C (en)	1992-06-16
DK159686B (da)	1990-11-19
GB2130587A (en)	1984-06-06
GB8327736D0 (en)	1983-11-16
US4645763A (en)	1987-02-24
DK159686C (da)	1991-04-15

Publication	Publication Date	Title
ES512381A0 (es)	1983-03-01	"procedimiento de preparacion de disacaridos".
DK533783A (da)	1984-05-23	6alfa-methylcortikoider, deres fremstilling og anvendelse
DK369482A (da)	1983-02-19	6alfa-methylprednisolonderivater, deres fremstilling og anvendelse
DK306385D0 (da)	1985-07-04	Phenylnaphthyridiner samt deres fremstilling og anvendelse
IE833006L (en)	1984-06-21	Substituted azabicycloalkanes.
DK440987D0 (da)	1987-08-24	Thyroninderivater, deres fremstilling og anvendelse
FI910059A0 (fi)	1991-01-04	Kemiska foereningar.
FI852429A0 (fi)	1985-06-19	Substituerade azabicykloheptaner, deras anvaendning, dessa foereningar innehaollande farmaceutiska preparat och foerfaranden foer framstaellning av dessa foereningar.
SE8206548L (sv)	1983-05-19	Bensylidenderivat
ES483271A1 (es)	1980-04-16	Un metodo para preparar tiofenocarboxamido-alcohil-mercapta-nos
ES526898A0 (es)	1984-07-01	Procedimiento para la preparacion de nuevas 7 -aciltio-1 ,2 -metilen-3-oxo-17 -pregn-4-en-21,17-carbolactonas
SE8303569D0 (sv)	1983-06-21	Polyprenylforeningar
SE7905468L (sv)	1979-12-23	(1-alkyl-5-nitro-2-imidazolyl)-vinyl-glyoxal-diacetaler, deras framstellning och anvendning