DK1680425T3 - 6-[(substitueret)phenyl]triazolopyrimidiner som anticancermidler - Google Patents

6-[(substitueret)phenyl]triazolopyrimidiner som anticancermidler

Info

Publication number: DK1680425T3
Authority: DK; Denmark
Prior art keywords: triazolopyrimidines; phenyl; substituted; anticancer agents; anticancer
Prior art date: 2003-09-24

Application number

DK04788820T

Other languages

English (en)

Inventor

Thai Hiep Nguyen

Yanzhong Wu

Wei Tong

Nan Zhang

Semiramis Ayral-Kaloustian

Original Assignee

Wyeth Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-09-24

Filing date

2004-09-17

Publication date

2007-03-19

2004-09-17 Application filed by Wyeth Corp filed Critical Wyeth Corp

2007-03-19 Application granted granted Critical

2007-03-19 Publication of DK1680425T3 publication Critical patent/DK1680425T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Oncology (AREA)
Hematology (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK04788820T 2003-09-24 2004-09-17 6-[(substitueret)phenyl]triazolopyrimidiner som anticancermidler DK1680425T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US50554403P	2003-09-24	2003-09-24
PCT/US2004/030515 WO2005030775A1 (en)	2003-09-24	2004-09-17	6-[(substituted)phenyl]triazolopyrimidines as anticancer agents

Publications (1)

Publication Number	Publication Date
DK1680425T3 true DK1680425T3 (da)	2007-03-19

Family

ID=34393032

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK04788820T DK1680425T3 (da)	2003-09-24	2004-09-17	6-[(substitueret)phenyl]triazolopyrimidiner som anticancermidler

Country Status (31)

Country	Link
US (1)	US7507739B2 (da)
EP (1)	EP1680425B1 (da)
JP (1)	JP2007506744A (da)
KR (1)	KR20060098368A (da)
CN (1)	CN100519559C (da)
AR (1)	AR045810A1 (da)
AU (1)	AU2004276240A1 (da)
BR (1)	BRPI0414700A (da)
CA (1)	CA2539252A1 (da)
CO (1)	CO5690598A2 (da)
CR (1)	CR8288A (da)
CY (1)	CY1106392T1 (da)
DE (1)	DE602004004295T8 (da)
DK (1)	DK1680425T3 (da)
EC (1)	ECSP066458A (da)
ES (1)	ES2279452T3 (da)
GT (1)	GT200400190A (da)
HK (1)	HK1090374A1 (da)
IL (1)	IL174281A0 (da)
MX (1)	MXPA06003206A (da)
NO (1)	NO20061318L (da)
PA (1)	PA8613301A1 (da)
PE (1)	PE20050433A1 (da)
PL (1)	PL1680425T3 (da)
PT (1)	PT1680425E (da)
RU (1)	RU2006107579A (da)
SA (1)	SA04250302A (da)
SI (1)	SI1680425T1 (da)
TW (1)	TW200512211A (da)
WO (1)	WO2005030775A1 (da)
ZA (1)	ZA200602387B (da)

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AU2004276240A1 (en)	2003-09-24	2005-04-07	Wyeth Holdings Corporation	6-[(substituted)phenyl]triazolopyrimidines as anticancer agents
US7419982B2 (en) *	2003-09-24	2008-09-02	Wyeth Holdings Corporation	Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
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CN101193884A (zh)	2005-06-13	2008-06-04	惠氏公司	微管蛋白抑制剂和其制备方法
WO2006138180A1 (en) *	2005-06-13	2006-12-28	Wyeth	Tubulin inhibitor and process for its preparation
US20090131708A1 (en) *	2005-06-27	2009-05-21	Basf Aktiengesellschaft	Method For Production of Substituted Phenylmalonate Esters, Intermediate Compounds and The Use Thereof for production of 5, 7-dihydroxy-6-(2,4,5-trifluorophenyl)-(1,2,4)triazolo(1,5-A)pyrimidines
JP2009519952A (ja) *	2005-12-16	2009-05-21	ワイス	トリアゾロピリミジン化合物の凍結乾燥組成物
JP2009519954A (ja) *	2005-12-16	2009-05-21	ワイス	抗癌剤として有用な６−［（置換）フェニル］トリアゾロピリミジンの二量体および付加物
BRPI0807458A2 (pt) *	2007-01-08	2014-06-03	Basf Se	Uso de compostos, agente, semente, método para combater fungos nocivos fitopatogênicos, e, composto
EP3219207A1 (en) *	2012-09-19	2017-09-20	The Trustees Of The University Of Pennsylvania	Heterocyclic compounds and their use for the treatment of neurodegenerative tauopathies
US11623927B2 (en)	2018-03-02	2023-04-11	The Trustees Of The University Of Pennsylvania	Substituted [1,2,4]triazolo[1,5-a]pyrimidines for stabilizing microtubules
CN114369098B (zh) *	2022-01-06	2023-03-10	苏州大学	一种三唑并嘧啶醇类化合物及其制备方法和应用

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US6268371B1 (en)	1998-09-10	2001-07-31	American Cyanamid Co.	Fungicidal mixtures
US5985883A (en)	1998-09-25	1999-11-16	American Cyanamid Company	Fungicidal trichlorophenyl-triazolopyrimidines
US6277856B1 (en)	1998-09-25	2001-08-21	American Cynamid Co.	Fungicidal mixtures
US5986135A (en)	1998-09-25	1999-11-16	American Cyanamid Company	Fungicidal trifluoromethylalkylamino-triazolopyrimidines
DE69908052T2 (de)	1998-09-25	2003-11-27	Basf Ag	Fungizide Mischungen
DE69914364T2 (de)	1998-09-25	2004-07-22	Basf Ag	Nicht-wässriges suspensionskonzentrat
US6242451B1 (en)	1998-09-25	2001-06-05	Klaus-Juergen Pees	Fungicidal trihalophenyl-triazolopyrimidines
JP2000103790A (ja)	1998-09-25	2000-04-11	American Cyanamid Co	殺菌・殺カビ性のトリハロフェニル―トリアゾロピリミジン類
US6521628B1 (en)	1999-01-29	2003-02-18	Basf Aktiengesellschaft	Fungicidal mixtures
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WO2001035738A2 (en)	1999-11-18	2001-05-25	Basf Corporation	Non-aqueous concentrated spreading oil composition
US6559151B2 (en)	2000-05-08	2003-05-06	Basf Aktiengesellschaft	6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
AU7306201A (en) *	2000-06-30	2002-01-14	American Home Prod	Substituted-triazolopyrimidines as anticancer agents
CZ295872B6 (cs)	2000-08-25	2005-11-16	Basf Aktiengesellschaft	Fungicidní prostředek
US6459602B1 (en) *	2000-10-26	2002-10-01	O2 Micro International Limited	DC-to-DC converter with improved transient response
JP2004513170A (ja)	2000-11-13	2004-04-30	ビーエーエスエフ　アクチェンゲゼルシャフト	７−（ｒ）−アミノトリアゾロピリミジン類、それらの製造及び植物病原性真菌を防除するためのそれらの使用
DE60013188T2 (de)	2000-12-06	2004-12-30	Basf Ag	Fungiizide 6-(trifluormethyl-phenyl)-triazolpyrimidine
DE10063115A1 (de)	2000-12-18	2002-06-27	Bayer Ag	Triazolopyrimidine
WO2002067679A1 (en)	2001-02-19	2002-09-06	Basf Aktiengesellschaft	Fungicidal mixtures
NZ528745A (en)	2001-04-11	2005-03-24	Basf Ag	5-halogen-6-phenyl-7-fluoralkylamino-triazolopyrimidines as fungicides and their preparation process
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AU2004276240A1 (en)	2003-09-24	2005-04-07	Wyeth Holdings Corporation	6-[(substituted)phenyl]triazolopyrimidines as anticancer agents

2004
- 2004-09-17 AU AU2004276240A patent/AU2004276240A1/en not_active Withdrawn
- 2004-09-17 ES ES04788820T patent/ES2279452T3/es not_active Expired - Lifetime
- 2004-09-17 MX MXPA06003206A patent/MXPA06003206A/es active IP Right Grant
- 2004-09-17 CN CNB2004800302006A patent/CN100519559C/zh not_active Expired - Fee Related
- 2004-09-17 BR BRPI0414700-6A patent/BRPI0414700A/pt not_active IP Right Cessation
- 2004-09-17 EP EP04788820A patent/EP1680425B1/en not_active Expired - Lifetime
- 2004-09-17 JP JP2006528075A patent/JP2007506744A/ja not_active Withdrawn
- 2004-09-17 PL PL04788820T patent/PL1680425T3/pl unknown
- 2004-09-17 DE DE602004004295T patent/DE602004004295T8/de active Active
- 2004-09-17 PT PT04788820T patent/PT1680425E/pt unknown
- 2004-09-17 SI SI200430195T patent/SI1680425T1/sl unknown
- 2004-09-17 KR KR1020067005785A patent/KR20060098368A/ko not_active Application Discontinuation
- 2004-09-17 WO PCT/US2004/030515 patent/WO2005030775A1/en active IP Right Grant
- 2004-09-17 DK DK04788820T patent/DK1680425T3/da active
- 2004-09-17 CA CA002539252A patent/CA2539252A1/en not_active Abandoned
- 2004-09-17 RU RU2006107579/04A patent/RU2006107579A/ru not_active Application Discontinuation
- 2004-09-21 TW TW093128500A patent/TW200512211A/zh unknown
- 2004-09-22 SA SA04250302A patent/SA04250302A/ar unknown
- 2004-09-23 PE PE2004000925A patent/PE20050433A1/es not_active Application Discontinuation
- 2004-09-23 AR ARP040103440A patent/AR045810A1/es not_active Application Discontinuation
- 2004-09-24 GT GT200400190A patent/GT200400190A/es unknown
- 2004-09-24 PA PA20048613301A patent/PA8613301A1/es unknown
- 2004-09-24 US US10/950,543 patent/US7507739B2/en not_active Expired - Fee Related
2006
- 2006-03-13 IL IL174281A patent/IL174281A0/en unknown
- 2006-03-14 CR CR8288A patent/CR8288A/es not_active Application Discontinuation
- 2006-03-23 NO NO20061318A patent/NO20061318L/no not_active Application Discontinuation
- 2006-03-23 ZA ZA200602387A patent/ZA200602387B/xx unknown
- 2006-03-24 EC EC2006006458A patent/ECSP066458A/es unknown
- 2006-04-21 CO CO06038133A patent/CO5690598A2/es not_active Application Discontinuation
- 2006-11-01 HK HK06112040A patent/HK1090374A1/xx not_active IP Right Cessation
2007
- 2007-03-16 CY CY20071100373T patent/CY1106392T1/el unknown

Also Published As

Publication number	Publication date
MXPA06003206A (es)	2006-06-23
PL1680425T3 (pl)	2007-05-31
SA04250302A (ar)	2005-12-03
DE602004004295T8 (de)	2007-09-20
RU2006107579A (ru)	2007-10-27
CN1867569A (zh)	2006-11-22
CY1106392T1 (el)	2011-10-12
CO5690598A2 (es)	2006-10-31
ES2279452T3 (es)	2007-08-16
AU2004276240A1 (en)	2005-04-07
GT200400190A (es)	2005-05-02
CN100519559C (zh)	2009-07-29
PT1680425E (pt)	2007-02-28
PE20050433A1 (es)	2005-07-21
HK1090374A1 (en)	2006-12-22
IL174281A0 (en)	2006-08-01
PA8613301A1 (es)	2005-11-25
DE602004004295D1 (de)	2007-02-22
NO20061318L (no)	2006-04-21
EP1680425A1 (en)	2006-07-19
EP1680425B1 (en)	2007-01-10
BRPI0414700A (pt)	2006-11-14
WO2005030775A1 (en)	2005-04-07
CA2539252A1 (en)	2005-04-07
ZA200602387B (en)	2008-11-26
JP2007506744A (ja)	2007-03-22
KR20060098368A (ko)	2006-09-18
CR8288A (es)	2006-10-04
DE602004004295T2 (de)	2007-06-06
AR045810A1 (es)	2005-11-16
ECSP066458A (es)	2006-09-18
US7507739B2 (en)	2009-03-24
US20050090508A1 (en)	2005-04-28
SI1680425T1 (sl)	2007-04-30
TW200512211A (en)	2005-04-01

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