DK1322651T3 - Bicykliske, heteroaromatiske forbindelser - Google Patents

Bicykliske, heteroaromatiske forbindelser

Info

Publication number: DK1322651T3
Authority: DK; Denmark
Prior art keywords: heteroaromatic compounds; bicyclic heteroaromatic; bicyclic; compounds; heteroaromatic
Prior art date: 2000-09-22

Application number

DK01982306T

Other languages

English (en)

Inventor

Cornelis Marius Timmers

Willem Frederik Johan Karstens

Original Assignee

Organon Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-09-22

Filing date

2001-09-17

Publication date

2008-06-02

2001-09-17 Application filed by Organon Nv filed Critical Organon Nv

2008-06-02 Application granted granted Critical

2008-06-02 Publication of DK1322651T3 publication Critical patent/DK1322651T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK01982306T 2000-09-22 2001-09-17 Bicykliske, heteroaromatiske forbindelser DK1322651T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP00203287		2000-09-22
PCT/EP2001/010743 WO2002024703A1 (en)	2000-09-22	2001-09-17	Bicyclic heteroaromatic compounds

Publications (1)

Publication Number	Publication Date
DK1322651T3 true DK1322651T3 (da)	2008-06-02

Family

ID=8172046

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK01982306T DK1322651T3 (da)	2000-09-22	2001-09-17	Bicykliske, heteroaromatiske forbindelser

Country Status (31)

Country	Link
US (2)	US7229990B2 (da)
EP (2)	EP1322651B1 (da)
JP (1)	JP4977940B2 (da)
KR (1)	KR100860040B1 (da)
CN (1)	CN1247594C (da)
AR (1)	AR030784A1 (da)
AT (1)	ATE384726T1 (da)
AU (2)	AU2002213929B2 (da)
BR (1)	BR0113987A (da)
CA (1)	CA2422054C (da)
CY (1)	CY1107308T1 (da)
CZ (1)	CZ297136B6 (da)
DE (1)	DE60132607T2 (da)
DK (1)	DK1322651T3 (da)
EC (1)	ECSP034523A (da)
ES (1)	ES2299524T3 (da)
HR (1)	HRP20030220B1 (da)
HU (1)	HU229422B1 (da)
IL (2)	IL154624A0 (da)
IS (1)	IS2531B (da)
MX (1)	MXPA03002478A (da)
NO (1)	NO328683B1 (da)
NZ (1)	NZ524444A (da)
PE (1)	PE20020537A1 (da)
PL (1)	PL207755B1 (da)
PT (1)	PT1322651E (da)
RU (1)	RU2271360C2 (da)
SK (1)	SK287554B6 (da)
TW (1)	TWI290143B (da)
WO (1)	WO2002024703A1 (da)
ZA (1)	ZA200301588B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PL207755B1 (pl) *	2000-09-22	2011-01-31	N V Organon	Bicykliczny związek heteroaromatyczny, zawierająca go kompozycja farmaceutyczna i jego zastosowania
TW200407127A (en)	2002-08-21	2004-05-16	Astrazeneca Ab	Chemical compounds
US7674822B2 (en)	2004-11-24	2010-03-09	Wyeth	PTP1b inhibitors
US7737155B2 (en) *	2005-05-17	2010-06-15	Schering Corporation	Nitrogen-containing heterocyclic compounds and methods of use thereof
WO2006124490A2 (en) *	2005-05-17	2006-11-23	Schering Corporation	Heterocycles as nicotinic acid receptor agonists for the treatment of dyslipidemia
AU2007254165A1 (en) *	2006-05-17	2007-11-29	Forschungsverbund Berlin E.V.	Pyrimidine low molecular weight ligands for modulating hormone receptors
EP2280969A1 (en)	2008-04-29	2011-02-09	F. Hoffmann-La Roche AG	Pyrimidinyl pyridone inhibitors of jnk.
CA2741030A1 (en) *	2008-10-20	2010-04-29	Marvin C. Gershengorn	Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
CA2789818A1 (en)	2010-04-08	2011-10-13	The United States Of America, As Represented By The Secretary, Departmen T Of Health And Human Services	Inverse agonists and neutral antagonists for the tsh receptor
EP2748166B1 (en)	2011-08-23	2018-07-11	Asana BioSciences, LLC	Pyrimido-pyridazinone compounds and use thereof
CN113680386B (zh) *	2021-08-23	2023-08-11	深圳湾实验室坪山生物医药研发转化中心	氮杂环卡宾-方酰胺双功能催化剂及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
RU2127736C1 (ru) *	1992-06-22	1999-03-20	Берингер Ингельгейм КГ	Производные анеллированного дигидропиридина или их соли с физиологически переносимыми кислотами и средство, блокирующее неселективные катионные каналы
TW276256B (da) *	1993-08-26	1996-05-21	Takeda Pharm Industry Co Ltd
CA2192820C (en) *	1994-06-16	2000-11-28	Yuhpyng L. Chen	Pyrazolo and pyrrolopyridines
AU712019B2 (en) *	1996-05-20	1999-10-28	Merck & Co., Inc.	Antagonists of gonadotropin releasing hormone
TW564247B (en) *	1999-04-08	2003-12-01	Akzo Nobel Nv	Bicyclic heteraromatic compound
PL207755B1 (pl) *	2000-09-22	2011-01-31	N V Organon	Bicykliczny związek heteroaromatyczny, zawierająca go kompozycja farmaceutyczna i jego zastosowania

2001
- 2001-09-17 PL PL360675A patent/PL207755B1/pl unknown
- 2001-09-17 MX MXPA03002478A patent/MXPA03002478A/es active IP Right Grant
- 2001-09-17 JP JP2002529113A patent/JP4977940B2/ja not_active Expired - Fee Related
- 2001-09-17 KR KR1020037004132A patent/KR100860040B1/ko not_active Expired - Fee Related
- 2001-09-17 PT PT01982306T patent/PT1322651E/pt unknown
- 2001-09-17 IL IL15462401A patent/IL154624A0/xx unknown
- 2001-09-17 AT AT01982306T patent/ATE384726T1/de active
- 2001-09-17 RU RU2003111463/04A patent/RU2271360C2/ru not_active IP Right Cessation
- 2001-09-17 CZ CZ20030828A patent/CZ297136B6/cs not_active IP Right Cessation
- 2001-09-17 AU AU2002213929A patent/AU2002213929B2/en not_active Ceased
- 2001-09-17 DE DE60132607T patent/DE60132607T2/de not_active Expired - Lifetime
- 2001-09-17 EP EP01982306A patent/EP1322651B1/en not_active Expired - Lifetime
- 2001-09-17 EP EP07113490A patent/EP1886999A3/en not_active Withdrawn
- 2001-09-17 BR BR0113987-8A patent/BR0113987A/pt not_active IP Right Cessation
- 2001-09-17 CA CA2422054A patent/CA2422054C/en not_active Expired - Fee Related
- 2001-09-17 WO PCT/EP2001/010743 patent/WO2002024703A1/en active IP Right Grant
- 2001-09-17 ES ES01982306T patent/ES2299524T3/es not_active Expired - Lifetime
- 2001-09-17 NZ NZ524444A patent/NZ524444A/en not_active IP Right Cessation
- 2001-09-17 US US10/381,248 patent/US7229990B2/en not_active Expired - Lifetime
- 2001-09-17 HR HR20030220A patent/HRP20030220B1/xx not_active IP Right Cessation
- 2001-09-17 HU HU0302648A patent/HU229422B1/hu not_active IP Right Cessation
- 2001-09-17 SK SK331-2003A patent/SK287554B6/sk not_active IP Right Cessation
- 2001-09-17 DK DK01982306T patent/DK1322651T3/da active
- 2001-09-17 AU AU1392902A patent/AU1392902A/xx active Pending
- 2001-09-17 CN CNB018160670A patent/CN1247594C/zh not_active Expired - Fee Related
- 2001-09-19 TW TW090123098A patent/TWI290143B/zh not_active IP Right Cessation
- 2001-09-21 PE PE2001000954A patent/PE20020537A1/es not_active Application Discontinuation
- 2001-09-21 AR ARP010104458A patent/AR030784A1/es active IP Right Grant
2003
- 2003-02-26 IL IL154624A patent/IL154624A/en not_active IP Right Cessation
- 2003-02-26 ZA ZA200301588A patent/ZA200301588B/en unknown
- 2003-02-28 IS IS6732A patent/IS2531B/is unknown
- 2003-03-21 EC EC2003004523A patent/ECSP034523A/es unknown
- 2003-03-21 NO NO20031314A patent/NO328683B1/no not_active IP Right Cessation
2007
- 2007-04-23 US US11/788,886 patent/US7618963B2/en not_active Expired - Lifetime
2008
- 2008-03-18 CY CY20081100301T patent/CY1107308T1/el unknown

Also Published As

Publication number	Publication date
HUP0302648A2 (hu)	2003-11-28
PL207755B1 (pl)	2011-01-31
CY1107308T1 (el)	2012-11-21
RU2271360C2 (ru)	2006-03-10
EP1322651A1 (en)	2003-07-02
DE60132607D1 (de)	2008-03-13
US7229990B2 (en)	2007-06-12
HU229422B1 (hu)	2013-12-30
CN1462273A (zh)	2003-12-17
DE60132607T2 (de)	2009-01-29
PL360675A1 (en)	2004-09-20
TWI290143B (en)	2007-11-21
HRP20030220A2 (en)	2003-06-30
US7618963B2 (en)	2009-11-17
NO20031314L (no)	2003-03-21
AU2002213929B2 (en)	2006-04-13
EP1886999A2 (en)	2008-02-13
US20070197527A1 (en)	2007-08-23
PE20020537A1 (es)	2002-06-20
NO328683B1 (no)	2010-04-26
CZ2003828A3 (cs)	2003-08-13
EP1886999A8 (en)	2010-08-04
ATE384726T1 (de)	2008-02-15
ECSP034523A (es)	2003-04-25
CZ297136B6 (cs)	2006-09-13
AR030784A1 (es)	2003-09-03
US20030225113A1 (en)	2003-12-04
KR100860040B1 (ko)	2008-09-25
HK1054942A1 (en)	2003-12-19
SK3312003A3 (en)	2003-08-05
CA2422054C (en)	2011-01-11
IL154624A0 (en)	2003-09-17
AU1392902A (en)	2002-04-02
KR20030040483A (ko)	2003-05-22
CA2422054A1 (en)	2002-03-28
SK287554B6 (sk)	2011-01-04
EP1322651B1 (en)	2008-01-23
HRP20030220B1 (en)	2011-10-31
JP2004509896A (ja)	2004-04-02
MXPA03002478A (es)	2004-05-05
IS2531B (is)	2009-07-15
BR0113987A (pt)	2003-08-12
JP4977940B2 (ja)	2012-07-18
EP1886999A3 (en)	2008-03-12
NO20031314D0 (no)	2003-03-21
PT1322651E (pt)	2008-02-28
IS6732A (is)	2003-02-28
CN1247594C (zh)	2006-03-29
ZA200301588B (en)	2004-06-22
WO2002024703A1 (en)	2002-03-28
ES2299524T3 (es)	2008-06-01
HUP0302648A3 (en)	2004-11-29
IL154624A (en)	2009-09-01
NZ524444A (en)	2004-03-26

Publication	Publication Date	Title
DK1259489T3 (da)	2006-10-09	Arylfusionerede, azapolycykliske forbindelser
NO20026196L (no)	2003-02-24	Kinazolinditosylatsalt-forbindelser
BR0214972B1 (pt)	2012-08-21	artigo absorvente.
IS6971A (is)	2003-09-29	Ný efnasambönd
NO20023516D0 (no)	2002-07-23	Antibakterielle 3-aminokinazolinon-2,4-dioner
DE50213548D1 (de)	2009-06-25	Substituierte 2-carba-3,5-dicyano-4-aryl-6-aminopylektive liganden
DK1322651T3 (da)	2008-06-02	Bicykliske, heteroaromatiske forbindelser
ATE372338T1 (de)	2007-09-15	Deshalogenverbindungen
NO20030303L (no)	2003-03-20	Kalsilytiske forbindelser
NO20023508L (no)	2002-07-23	Kalsilyttiske forbindelser
NO20031837D0 (no)	2003-04-24	Kalsilytiske forbindelser
BR0212092B1 (pt)	2012-05-15	artigo absorvente.
BR0213766B1 (pt)	2012-05-15	artigo absorvente.
ATE470655T1 (de)	2010-06-15	Substituierte 1,5-diaminopentan-3-ol-verbindungen
DE50209630D1 (de)	2007-04-19	Drehmaschine
DE60224192D1 (de)	2008-01-31	Antihaemorrhagische, betain-enthaltende zusammenseuzungen
SE0003477D0 (sv)	2000-09-28	Compounds
SE0101659D0 (sv)	2001-05-11	New compounds
SE0102056D0 (sv)	2001-06-08	New Compounds
SE0102386D0 (sv)	2001-07-03	New compounds
SE0103437D0 (sv)	2001-10-16	New compounds
SE0103461D0 (sv)	2001-10-16	New compounds
SE0104366D0 (sv)	2001-12-20	New compounds
SE0101958D0 (sv)	2001-06-05	New compounds
SE0100629D0 (sv)	2001-02-23	New compounds