DE69912282D1 - Verfahren zur herstellung eines indolderivates - Google Patents
Verfahren zur herstellung eines indolderivatesInfo
- Publication number
- DE69912282D1 DE69912282D1 DE69912282T DE69912282T DE69912282D1 DE 69912282 D1 DE69912282 D1 DE 69912282D1 DE 69912282 T DE69912282 T DE 69912282T DE 69912282 T DE69912282 T DE 69912282T DE 69912282 D1 DE69912282 D1 DE 69912282D1
- Authority
- DE
- Germany
- Prior art keywords
- indolder
- derivative
- producing
- carboxylate
- indole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- LAMUXTNQCICZQX-UHFFFAOYSA-N 3-chloropropan-1-ol Chemical compound OCCCCl LAMUXTNQCICZQX-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- SIKJAQJRHWYJAI-UHFFFAOYSA-N benzopyrrole Natural products C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 abstract 1
- PZOUSPYUWWUPPK-UHFFFAOYSA-N indole Natural products CC1=CC=CC2=C1C=CN2 PZOUSPYUWWUPPK-UHFFFAOYSA-N 0.000 abstract 1
- RKJUIXBNRJVNHR-UHFFFAOYSA-N indolenine Natural products C1=CC=C2CC=NC2=C1 RKJUIXBNRJVNHR-UHFFFAOYSA-N 0.000 abstract 1
- IJQYPUZBTYDSGN-UHFFFAOYSA-N methyl 2-(3-chloropropoxy)-1h-indole-3-carboxylate Chemical compound C1=CC=C2C(C(=O)OC)=C(OCCCCl)NC2=C1 IJQYPUZBTYDSGN-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9815481.8A GB9815481D0 (en) | 1998-07-16 | 1998-07-16 | Pharmaceuticals |
| GB9815481 | 1998-07-16 | ||
| PCT/EP1999/004944 WO2000003984A1 (en) | 1998-07-16 | 1999-07-13 | Process for the preparation of an indole derivate |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69912282D1 true DE69912282D1 (de) | 2003-11-27 |
| DE69912282T2 DE69912282T2 (de) | 2004-07-29 |
Family
ID=10835640
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69912282T Expired - Lifetime DE69912282T2 (de) | 1998-07-16 | 1999-07-13 | Verfahren zur herstellung eines indolderivates |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1097136B1 (de) |
| JP (1) | JP3842556B2 (de) |
| AT (1) | ATE252557T1 (de) |
| CA (1) | CA2337382C (de) |
| DE (1) | DE69912282T2 (de) |
| ES (1) | ES2209476T3 (de) |
| GB (1) | GB9815481D0 (de) |
| WO (1) | WO2000003984A1 (de) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0211230D0 (en) | 2002-05-16 | 2002-06-26 | Medinnova Sf | Treatment of heart failure |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK0922048T3 (da) * | 1996-08-16 | 2001-01-08 | Smithkline Beecham Plc | Fremgangsmåde til fremstilling af N-[(1-n-butyl-4-piperidinyl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a]-indol-10-carboxami |
-
1998
- 1998-07-16 GB GBGB9815481.8A patent/GB9815481D0/en not_active Ceased
-
1999
- 1999-07-13 EP EP99938234A patent/EP1097136B1/de not_active Expired - Lifetime
- 1999-07-13 JP JP2000560093A patent/JP3842556B2/ja not_active Expired - Fee Related
- 1999-07-13 WO PCT/EP1999/004944 patent/WO2000003984A1/en active IP Right Grant
- 1999-07-13 AT AT99938234T patent/ATE252557T1/de not_active IP Right Cessation
- 1999-07-13 DE DE69912282T patent/DE69912282T2/de not_active Expired - Lifetime
- 1999-07-13 ES ES99938234T patent/ES2209476T3/es not_active Expired - Lifetime
- 1999-07-13 CA CA002337382A patent/CA2337382C/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2337382A1 (en) | 2000-01-27 |
| WO2000003984A1 (en) | 2000-01-27 |
| JP2002520392A (ja) | 2002-07-09 |
| JP3842556B2 (ja) | 2006-11-08 |
| CA2337382C (en) | 2008-04-08 |
| ES2209476T3 (es) | 2004-06-16 |
| GB9815481D0 (en) | 1998-09-16 |
| DE69912282T2 (de) | 2004-07-29 |
| EP1097136A1 (de) | 2001-05-09 |
| ATE252557T1 (de) | 2003-11-15 |
| EP1097136B1 (de) | 2003-10-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |