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DE60004066D1 - Benzofurylpiperazine: 5-ht2c serotoninrezeptor agonisten - Google Patents

Benzofurylpiperazine: 5-ht2c serotoninrezeptor agonisten

Info

Publication number
DE60004066D1
DE60004066D1 DE60004066T DE60004066T DE60004066D1 DE 60004066 D1 DE60004066 D1 DE 60004066D1 DE 60004066 T DE60004066 T DE 60004066T DE 60004066 T DE60004066 T DE 60004066T DE 60004066 D1 DE60004066 D1 DE 60004066D1
Authority
DE
Germany
Prior art keywords
sup
benzofurylpiperazine
ht2c
receptor agonists
serotonine receptor
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60004066T
Other languages
English (en)
Other versions
DE60004066T2 (de
Inventor
Karin Briner
Paul Burkhart
Paul Burkholder
Eugene Cunningham
Joseph Fisher
Harlan Gritton
Christopher Miller
Thomas Mullaney
Robert Reinhard
Charles Thompson
Larry Winneroski
Yanping Xu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Application granted granted Critical
Publication of DE60004066D1 publication Critical patent/DE60004066D1/de
Publication of DE60004066T2 publication Critical patent/DE60004066T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
DE60004066T 1999-07-29 2000-07-21 Benzofurylpiperazine: 5-ht2c serotoninrezeptor agonisten Expired - Fee Related DE60004066T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14627099P 1999-07-29 1999-07-29
US146270P 1999-07-29
PCT/US2000/019543 WO2001009111A1 (en) 1999-07-29 2000-07-21 Benzofurylpiperazines and benzofurylhomopiperazines: serotonin agonists

Publications (2)

Publication Number Publication Date
DE60004066D1 true DE60004066D1 (de) 2003-08-28
DE60004066T2 DE60004066T2 (de) 2004-04-15

Family

ID=22516599

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60004066T Expired - Fee Related DE60004066T2 (de) 1999-07-29 2000-07-21 Benzofurylpiperazine: 5-ht2c serotoninrezeptor agonisten

Country Status (14)

Country Link
US (1) US6967201B1 (de)
EP (1) EP1204654B1 (de)
JP (1) JP2003506365A (de)
CN (1) CN1365359A (de)
AT (1) ATE245636T1 (de)
AU (1) AU768310B2 (de)
BR (1) BR0012752A (de)
CA (1) CA2378878A1 (de)
DE (1) DE60004066T2 (de)
DK (1) DK1204654T3 (de)
ES (1) ES2203498T3 (de)
MX (1) MXPA02000973A (de)
PT (1) PT1204654E (de)
WO (1) WO2001009111A1 (de)

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JP6772288B2 (ja) 2016-03-11 2020-10-21 ソルボンヌ・ユニヴェルシテＳｏｒｂｏｎｎｅ Ｕｎｉｖｅｒｓｉｔｅ 脊髄の治療および脊髄神経の治療のための体外式超音波発生治療デバイス、該デバイスを備える装置、および該装置を用いる方法
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Also Published As

Publication number Publication date
DE60004066T2 (de) 2004-04-15
AU6220200A (en) 2001-02-19
AU768310B2 (en) 2003-12-04
JP2003506365A (ja) 2003-02-18
MXPA02000973A (es) 2002-07-30
ATE245636T1 (de) 2003-08-15
WO2001009111A1 (en) 2001-02-08
PT1204654E (pt) 2003-11-28
ES2203498T3 (es) 2004-04-16
CN1365359A (zh) 2002-08-21
US6967201B1 (en) 2005-11-22
EP1204654B1 (de) 2003-07-23
DK1204654T3 (da) 2003-11-17
EP1204654A1 (de) 2002-05-15
BR0012752A (pt) 2002-04-02
CA2378878A1 (en) 2001-02-08

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