[go: up one dir, main page]

CY1116784T1 - Αντιμικροβιακες ενωσεις και μεθοδοι για χρηση αυτων - Google Patents

Αντιμικροβιακες ενωσεις και μεθοδοι για χρηση αυτων

Info

Publication number
CY1116784T1
CY1116784T1 CY20151100909T CY151100909T CY1116784T1 CY 1116784 T1 CY1116784 T1 CY 1116784T1 CY 20151100909 T CY20151100909 T CY 20151100909T CY 151100909 T CY151100909 T CY 151100909T CY 1116784 T1 CY1116784 T1 CY 1116784T1
Authority
CY
Cyprus
Prior art keywords
methods
antimicrobial compounds
protonated compounds
provides
antimicrobial activity
Prior art date
Application number
CY20151100909T
Other languages
English (en)
Inventor
Roderic M K Dale
Steven L Gatton
Amy Arrow
Terry Thompson
Original Assignee
Lakewood-Amedex, Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lakewood-Amedex, Inc filed Critical Lakewood-Amedex, Inc
Publication of CY1116784T1 publication Critical patent/CY1116784T1/el

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
    • A01N57/12—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing acyclic or cycloaliphatic radicals
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
    • A01N57/16—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing heterocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/02—Local antiseptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biotechnology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Materials For Medical Uses (AREA)
  • Apparatus For Disinfection Or Sterilisation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)
  • Cosmetics (AREA)

Abstract

Η παρούσα εφεύρεση παρέχει πρωτονιωμένες ενώσεις που έχουν αντιμικροβιακή δραστικότητα. Η εφεύρεση επίσης παρέχει αντιμικροβιακές συνθέσεις που περιλαμβάνουν πρωτονιωμένες ενώσεις της εφεύρεσης. Οι πρωτονιωμένες ενώσεις της εφεύρεσης παρέχουν αποτελεσματική αντιμικροβιακή δραστικότητα έναντι ανθεκτικών στελεχών βακτηριδίων και ευκαιριακών μυκήτων.
CY20151100909T 2001-05-03 2015-10-08 Αντιμικροβιακες ενωσεις και μεθοδοι για χρηση αυτων CY1116784T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/847,654 US20020032164A1 (en) 1998-12-30 2001-05-03 Antimicrobial compounds and methods for their use
EP10184218.5A EP2311466B1 (en) 2001-05-03 2002-05-03 Antimicrobial compounds and methods for their use

Publications (1)

Publication Number Publication Date
CY1116784T1 true CY1116784T1 (el) 2017-03-15

Family

ID=25301163

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20151100909T CY1116784T1 (el) 2001-05-03 2015-10-08 Αντιμικροβιακες ενωσεις και μεθοδοι για χρηση αυτων

Country Status (10)

Country Link
US (2) US20020032164A1 (el)
EP (2) EP2311466B1 (el)
JP (4) JP4347573B2 (el)
AU (1) AU2002305336B2 (el)
CA (2) CA2445381C (el)
CY (1) CY1116784T1 (el)
DK (1) DK2311466T3 (el)
ES (1) ES2549766T3 (el)
PT (1) PT2311466E (el)
WO (1) WO2002089581A1 (el)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020032164A1 (en) * 1998-12-30 2002-03-14 Dale Roderic M. K. Antimicrobial compounds and methods for their use
US6627215B1 (en) * 1998-12-30 2003-09-30 Oligos Etc. Inc. Devices for improved wound management
US7868162B2 (en) * 1998-12-30 2011-01-11 Lakewood-Amedex, Inc. Antimicrobial and antiviral compounds and methods for their use
CA2453362A1 (en) 2001-07-10 2003-01-23 Oligos Etc. Inc. Oligonucleotide-containing pharmacological compositions and their use
US8785403B2 (en) 2003-08-01 2014-07-22 Mitsubishi Tanabe Pharma Corporation Glucopyranoside compound
AU2004261264A1 (en) 2003-08-01 2005-02-10 Janssen Pharmaceutica N.V. Substituted indazole-O-glucosides
JP4130466B2 (ja) * 2003-08-01 2008-08-06 田辺三菱製薬株式会社 新規化合物
TW200727785A (en) * 2005-11-25 2007-08-01 Maruishi Pharma Gel composition for antibacterial sterilization
UY30730A1 (es) * 2006-12-04 2008-07-03 Mitsubishi Tanabe Pharma Corp Forma cristalina del hemihidrato de 1-(b (beta)-d-glucopiranosil) -4-metil-3-[5-(4-fluorofenil) -2-tienilmetil]benceno
ES2675045T3 (es) * 2007-05-04 2018-07-06 Symrise Ag Preparaciones activas sinérgicas que comprenden 1,2-decanodiol y además compuestos activos antimicrobianos
CN101801371B (zh) * 2007-09-10 2012-11-28 詹森药业有限公司 可用作sglt抑制剂的化合物的制备方法
CL2008003653A1 (es) 2008-01-17 2010-03-05 Mitsubishi Tanabe Pharma Corp Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica.
GB2460445B (en) * 2008-05-30 2012-07-11 Vernolix Ltd Treatment of ringworm
US9056850B2 (en) * 2008-10-17 2015-06-16 Janssen Pharmaceutica N.V. Process for the preparation of compounds useful as inhibitors of SGLT
US20110009347A1 (en) 2009-07-08 2011-01-13 Yin Liang Combination therapy for the treatment of diabetes
ES2416459T3 (es) 2009-07-10 2013-08-01 Janssen Pharmaceutica, N.V. Procedimiento de cristalización para 1-( -D-glucopiranosil)-4-metil-3-[5-(4-fluorofenil)-2-tienilmetil]benceno
LT2488515T (lt) * 2009-10-14 2017-03-10 Janssen Pharmaceutica Nv Junginių, naudotinų kaip sglt2 inhibitorių, paruošimo būdas
NZ703128A (en) 2010-05-11 2016-04-29 Janssen Pharmaceutica Nv Pharmaceutical formulations comprising 1 - (beta-d-glucopyranosyl) - 2 -thienylmethylbenzene derivatives as inhibitors of sglt
PL2697218T3 (pl) 2011-04-13 2016-11-30 Sposób wytwarzania związków użytecznych, jako inhibitory SGLT2
TWI542596B (zh) 2011-05-09 2016-07-21 健生藥品公司 （２ｓ,３ｒ,４ｒ,５ｓ,６ｒ）－２－（３－（（５－（４－氟苯基）噻吩－２－基）甲基）－４－甲基苯基）－６－（羥甲基）四氫－２ｈ－哌喃－３,４,５－三醇之ｌ－脯胺酸及檸檬酸共晶體
US20170071970A1 (en) 2015-09-15 2017-03-16 Janssen Pharmaceutica Nv Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders
US11795192B2 (en) 2017-03-10 2023-10-24 Lakewood Amedex, Inc. Antimicrobial compounds, compositions, and uses thereof
US11377468B2 (en) 2017-03-10 2022-07-05 Lakewood Amedex, Inc. Antimicrobial compounds, compositions, and uses thereof
KR102317158B1 (ko) 2017-03-10 2021-10-25 레이크우드 아메덱스, 인크. 항미생물 화합물, 조성물, 및 그의 용도
US12030908B2 (en) 2017-03-10 2024-07-09 Lakewood Amedex, Inc. Antimicrobial compounds, compositions, and uses thereof
AU2018282905B2 (en) 2017-06-12 2022-06-02 Lakewood Amedex, Inc Bisphosphocin gel formulations and uses thereof
WO2018237218A1 (en) 2017-06-23 2018-12-27 The Procter & Gamble Company COMPOSITION AND METHOD FOR ENHANCING SKIN APPEARANCE
CA3102288A1 (en) 2018-07-03 2020-01-09 The Procter & Gamble Company Method of treating a skin condition
CA3116157A1 (en) 2018-10-17 2020-04-23 Lakewood Amedex, Inc. Methods and compositions for treating oral mucositis
CZ2019769A3 (cs) * 2019-12-12 2021-09-22 Ăšstav organickĂ© chemie a biochemie AV ÄŚR, v. v. i. Lipofosfonoxiny třetí generace, jejich příprava a použití
US10959933B1 (en) 2020-06-01 2021-03-30 The Procter & Gamble Company Low pH skin care composition and methods of using the same
WO2021247496A1 (en) 2020-06-01 2021-12-09 The Procter & Gamble Company Method of improving penetration of a vitamin b3 compound into skin
KR20220009630A (ko) * 2020-07-16 2022-01-25 정준영 플라즈마를 이용한 마스크 폐기 처리기
CN115448967A (zh) * 2022-09-26 2022-12-09 泽同医药科技(南通)有限公司 一种吩噁嗪半乳烯糖碳苷化合物及其合成方法

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4105782A (en) 1975-03-07 1978-08-08 Yu Ruey J Treatment of acne and dandruff
DE2916318A1 (de) * 1979-04-23 1980-11-06 Hoechst Ag Waesserige desinfektionsloesung
US4421769A (en) 1981-09-29 1983-12-20 The Procter & Gamble Company Skin conditioning composition
US4908209A (en) * 1983-08-16 1990-03-13 Interface, Inc. Biocidal delivery system of phosphate ester and method of preparation thereof
JPS60209077A (ja) * 1984-03-27 1985-10-21 竹本油脂株式会社 繊維処理用油剤及び該油剤による合成繊維糸の処理方法
US4897355A (en) 1985-01-07 1990-01-30 Syntex (U.S.A.) Inc. N[ω,(ω-1)-dialkyloxy]- and N-[ω,(ω-1)-dialkenyloxy]-alk-1-yl-N,N,N-tetrasubstituted ammonium lipids and uses therefor
DE3542516A1 (de) 1985-12-02 1987-06-04 Henkel Kgaa Desinfektionsmittel
WO1989001023A1 (en) * 1987-08-03 1989-02-09 Interface Research Corporation Microbiocidal cleansing or disinfecting formulations and preparation thereof
US5153000A (en) * 1988-11-22 1992-10-06 Kao Corporation Phosphate, liposome comprising the phosphate as membrane constituent, and cosmetic and liposome preparation comprising the liposome
ZA902710B (en) 1989-05-22 1991-12-24 Univ Georgia Res Found Enzyme luminescence assay
US5153230A (en) 1989-10-06 1992-10-06 Perfective Cosmetics, Inc. Topical skin cream composition
US5264618A (en) 1990-04-19 1993-11-23 Vical, Inc. Cationic lipids for intracellular delivery of biologically active molecules
AU7979491A (en) 1990-05-03 1991-11-27 Vical, Inc. Intracellular delivery of biologically active substances by means of self-assembling lipid complexes
US5420330A (en) * 1990-09-07 1995-05-30 Pharmacia P-L Biochemicals Inc. Lipo-phosphoramidites
AU9097791A (en) * 1990-12-07 1992-07-08 Upjohn Company, The Phosphonic acid derivatives useful as antiinflammatory agents
US5681829A (en) * 1992-10-08 1997-10-28 Shaman Pharmaceuticals, Inc. Class of phosphocholine derivatives having antifungal activity
US5811568A (en) * 1992-10-08 1998-09-22 Shaman Pharmaceuticals, Inc. Process for the preparation of mono- and bis(phosphocholine) derivatives which have antifungal activity
AU5354494A (en) * 1992-10-08 1994-05-09 Shaman Pharmaceuticals, Inc. Novel class of phosphocholine derivatives having antifungal activity
DE4333385C2 (de) 1993-09-30 1997-01-30 Friedrich A Spruegel Flächendesinfektions- und Reinigungsmittel
FR2718022B1 (fr) 1994-04-01 1996-04-26 Roussel Uclaf Compositions cosmétiques ou dermatologiques et leur préparation.
FR2727289B1 (fr) * 1994-11-30 1999-03-05 Derives Resiniques Terpenique Composition desinfectante comprenant au moins un alcool terpenique et au moins un tensio-actif acide bactericide, et utilisation de tels tensio-actifs
US6071961A (en) * 1995-11-28 2000-06-06 Wider; Michael D. Antimicrobial composition and methods of use therefor
US5843998A (en) 1997-06-30 1998-12-01 Song; Jin Skin blemish treatment
US20020032164A1 (en) * 1998-12-30 2002-03-14 Dale Roderic M. K. Antimicrobial compounds and methods for their use
US6211349B1 (en) * 1998-12-30 2001-04-03 Oligos Etc., Inc. Protonated/acidified nucleic acids and methods of use
US6610314B2 (en) * 2001-03-12 2003-08-26 Kimberly-Clark Worldwide, Inc. Antimicrobial formulations

Also Published As

Publication number Publication date
JP5503900B2 (ja) 2014-05-28
JP4347573B2 (ja) 2009-10-21
CA2445381A1 (en) 2002-11-14
CA2445381C (en) 2013-09-17
CA2827671A1 (en) 2002-11-14
DK2311466T3 (en) 2015-10-19
EP2311466A3 (en) 2012-04-25
WO2002089581A1 (en) 2002-11-14
US20020032164A1 (en) 2002-03-14
US7176191B2 (en) 2007-02-13
EP1389909A1 (en) 2004-02-25
CA2827671C (en) 2016-07-05
PT2311466E (pt) 2015-10-27
JP2009179639A (ja) 2009-08-13
JP6097372B2 (ja) 2017-03-15
JP2005511482A (ja) 2005-04-28
EP2311466A2 (en) 2011-04-20
EP2311466B1 (en) 2015-07-08
ES2549766T3 (es) 2015-11-02
AU2002305336B2 (en) 2007-11-08
EP1389909B1 (en) 2012-07-18
US20050107344A1 (en) 2005-05-19
JP5883838B2 (ja) 2016-03-15
JP2016056177A (ja) 2016-04-21
JP2014055139A (ja) 2014-03-27
EP1389909A4 (en) 2005-03-30

Similar Documents

Publication Publication Date Title
CY1116784T1 (el) Αντιμικροβιακες ενωσεις και μεθοδοι για χρηση αυτων
EA200600602A1 (ru) Синергические фунгицидные комбинации биологически активных веществ
EP1431275A4 (en) DIARYL ETHER DERIVATIVE, ITS ADDITIONAL SALT AND IMMUNOSUPPRESSEUR
BR0307924A (pt) N-aril-2-oxazolidinona-5-carboxamidas e seus derivados
CY1108409T1 (el) Υβριδικα αντιβιοτικα οξαζολιδινονης-κινολονης
PT1453512E (pt) Derivados de acetileno tendo actividade antagonistica do mglur 5
NO20052787D0 (no) N-alkyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler
CY1110821T1 (el) Antibakthpiakoi πapaγontες τρικυκλικης tετραϋδροκινολινης
ATE455092T1 (de) Substituierte tetracyclin-verbindungen zur behandlung von malaria
CY1106247T1 (el) Θειοφαινο- και θειαζολοσουλφοναμιδες ως αντινεοπλαστικοι παραγοντες
NO20051082L (no) Antimikrobielle kinoloner, deres sammensetninger og anvendelser
MXPA04001686A (es) Combinaciones de productos activos fungicidas.
ATE511352T1 (de) Antimikrobielle zusammensetzungen
PT1289366E (pt) Combinacoes fungicidas de substancias activas
DE60321594D1 (de) Synergistische zusammensetzungen
UA83266C2 (en) Oxazole derivatives of tetracyclines
NO20052788L (no) N-sulfonyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler
ATE315380T1 (de) Epothilon zusammensetzungen
TR199901209T2 (xx) B�cek �ld�r�c� ve mitisidal kompozisyonlar
PL372769A1 (en) Cyanoguanidine prodrugs
PT1268475E (pt) Novos agentes bacterianos de benzosultam-oxazolidinona
BRPI0413744A (pt) n-aril-2-ciano-oxazolidinonas e seus derivados
ATE321760T1 (de) N-aryl-2-oxazolidinone und deren derivate
PT1387841E (pt) Novos derivados de azole ou de triazole, seu processo de preparacao e sua aplicacao como fungicidas
DE50212676D1 (de) Exopolysaccharidproduktion