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CY1113282T1 - Αντιικα νουκλεοζιτικα αναλογα - Google Patents

Αντιικα νουκλεοζιτικα αναλογα

Info

Publication number
CY1113282T1
CY1113282T1 CY20121100876T CY121100876T CY1113282T1 CY 1113282 T1 CY1113282 T1 CY 1113282T1 CY 20121100876 T CY20121100876 T CY 20121100876T CY 121100876 T CY121100876 T CY 121100876T CY 1113282 T1 CY1113282 T1 CY 1113282T1
Authority
CY
Cyprus
Prior art keywords
nucleozitic
antique
analogs
compounds
formula
Prior art date
Application number
CY20121100876T
Other languages
English (en)
Inventor
Yarlagadda S Babu
Pooran Chand
V Satish Kumar
Pravin L Kotian
Minwan Wu
Original Assignee
Biocryst Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biocryst Pharmaceuticals, Inc. filed Critical Biocryst Pharmaceuticals, Inc.
Publication of CY1113282T1 publication Critical patent/CY1113282T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/23—Heterocyclic radicals containing two or more heterocyclic rings condensed among themselves or condensed with a common carbocyclic ring system, not provided for in groups C07H19/14 - C07H19/22
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Η εφεύρεση παρουσιάζει ενώσεις του Τύπου (I), όπως περιγράφονται εδώ, καθώς και φαρμακευτικές συνθέσεις, οι οποίες περιέχουν τις ενώσεις, και συνθετικές μεθόδους και ενδιάμεσα, τα οποία είναι χρήσιμα για την παρασκευή των ενώσεων. Οι ενώσεις του Τύπου (I) είναι χρήσιμες ως αντιικοί παράγοντες και/ή ως αντικαρκινικοί παράγοντες.
CY20121100876T 2007-01-12 2012-09-25 Αντιικα νουκλεοζιτικα αναλογα CY1113282T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88027807P 2007-01-12 2007-01-12
EP08727625A EP2114980B1 (en) 2007-01-12 2008-01-11 Antiviral nucleoside analogs

Publications (1)

Publication Number Publication Date
CY1113282T1 true CY1113282T1 (el) 2016-04-13

Family

ID=39471795

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20121100876T CY1113282T1 (el) 2007-01-12 2012-09-25 Αντιικα νουκλεοζιτικα αναλογα

Country Status (20)

Country Link
US (1) US8440813B2 (el)
EP (2) EP2114980B1 (el)
JP (1) JP2010515760A (el)
CN (1) CN101611046A (el)
AU (1) AU2008206406A1 (el)
CA (1) CA2674589A1 (el)
CY (1) CY1113282T1 (el)
DK (1) DK2114980T3 (el)
ES (1) ES2390188T3 (el)
HK (1) HK1138286A1 (el)
HR (1) HRP20120758T1 (el)
IL (1) IL199664A0 (el)
MX (1) MX2009007333A (el)
NZ (2) NZ578556A (el)
PH (1) PH12012502284A1 (el)
PL (1) PL2114980T3 (el)
PT (1) PT2114980E (el)
SG (1) SG177974A1 (el)
SI (1) SI2114980T1 (el)
WO (1) WO2008089105A2 (el)

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Also Published As

Publication number Publication date
SG177974A1 (en) 2012-02-28
EP2114980A2 (en) 2009-11-11
PT2114980E (pt) 2012-09-25
WO2008089105A3 (en) 2008-09-12
MX2009007333A (es) 2009-08-31
EP2535345A1 (en) 2012-12-19
IL199664A0 (en) 2010-04-15
PH12012502284A1 (en) 2015-10-12
JP2010515760A (ja) 2010-05-13
PL2114980T3 (pl) 2012-11-30
WO2008089105A2 (en) 2008-07-24
EP2114980B1 (en) 2012-06-27
CA2674589A1 (en) 2008-07-24
HRP20120758T1 (hr) 2012-10-31
AU2008206406A1 (en) 2008-07-24
SI2114980T1 (sl) 2012-11-30
US20100015094A1 (en) 2010-01-21
ES2390188T3 (es) 2012-11-07
NZ598927A (en) 2013-09-27
NZ578556A (en) 2012-04-27
CN101611046A (zh) 2009-12-23
DK2114980T3 (da) 2012-09-24
US8440813B2 (en) 2013-05-14
HK1138286A1 (en) 2010-08-20

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