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CU20100119A7 - Compuestos orgánicos de aminotiazoles - Google Patents

Compuestos orgánicos de aminotiazoles

Info

Publication number
CU20100119A7
CU20100119A7 CU2010000119A CU20100119A CU20100119A7 CU 20100119 A7 CU20100119 A7 CU 20100119A7 CU 2010000119 A CU2010000119 A CU 2010000119A CU 20100119 A CU20100119 A CU 20100119A CU 20100119 A7 CU20100119 A7 CU 20100119A7
Authority
CU
Cuba
Prior art keywords
aminotiazols
organic compounds
diseases
prevention
improvement
Prior art date
Application number
CU2010000119A
Other languages
English (en)
Other versions
CU23908B1 (es
Inventor
Lewis Whitehead
Jennifer Leeds
Simon Bushell
Mathew J Lamarche
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40377437&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU20100119(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CU20100119A7 publication Critical patent/CU20100119A7/es
Publication of CU23908B1 publication Critical patent/CU23908B1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05—Dipeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/10—Anti-acne agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)

Abstract

La presente solicitud describe compuestos orgánicos de aminotiazoles que son útiles para el tratamiento, prevención y/o la mejora de enfermedades, en particular las infecciones bacterianas.
CU2010000119A 2007-12-12 2010-06-11 Compuestos orgánicos de aminotiazoles CU20100119A7 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1312207P 2007-12-12 2007-12-12
US2470908P 2008-01-30 2008-01-30
PCT/EP2008/067220 WO2009074605A1 (en) 2007-12-12 2008-12-10 Aminothiazoles and their uses

Publications (2)

Publication Number Publication Date
CU20100119A7 true CU20100119A7 (es) 2011-10-14
CU23908B1 CU23908B1 (es) 2013-06-28

Family

ID=40377437

Family Applications (1)

Application Number Title Priority Date Filing Date
CU2010000119A CU20100119A7 (es) 2007-12-12 2010-06-11 Compuestos orgánicos de aminotiazoles

Country Status (26)

Country Link
US (4) US8426356B2 (es)
EP (1) EP2229386B1 (es)
JP (2) JP5286366B2 (es)
KR (2) KR20120047335A (es)
CN (1) CN101945866B (es)
AR (1) AR069628A1 (es)
AU (1) AU2008334659A1 (es)
BR (1) BRPI0821138A2 (es)
CA (1) CA2708793C (es)
CL (1) CL2008003688A1 (es)
CO (1) CO6290661A2 (es)
CR (1) CR11469A (es)
CU (1) CU20100119A7 (es)
EA (2) EA201400280A1 (es)
EC (1) ECSP10010244A (es)
ES (1) ES2542878T3 (es)
GT (1) GT201000166A (es)
HN (1) HN2010001176A (es)
IL (1) IL206104A (es)
MA (1) MA31869B1 (es)
MY (1) MY156466A (es)
NZ (1) NZ585788A (es)
PE (1) PE20091108A1 (es)
TN (1) TN2010000254A1 (es)
TW (1) TWI430804B (es)
WO (1) WO2009074605A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR060977A1 (es) * 2006-05-31 2008-07-23 Novartis Ag Aminotiazoles y sus usos
JP5286366B2 (ja) * 2007-12-12 2013-09-11 ノバルティス アーゲー アミノチアゾール類およびその使用
WO2016081825A1 (en) 2014-11-21 2016-05-26 KamTek, Inc. Methods and compositions for treating clostridium difficile associated disease

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5202241A (en) 1988-09-09 1993-04-13 Gruppo Lepetit S.P.A. Antibiotic GE 2270
DE69016284T2 (de) 1989-07-04 1995-05-24 Lepetit Spa Antibiotikum GE 22270, Faktoren A1,A2,A3 und H.
ES2071143T3 (es) 1990-03-08 1995-06-16 Lepetit Spa Factores b1, b2, c1, c2, d1, d2, e y t del antibiotico ge 2270.
IL100572A (en) * 1991-01-03 1997-01-10 Lepetit Spa Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them
EP0529410B1 (en) 1991-08-30 1998-02-25 Biosearch Italia S.p.A. Antibiotic GE 2270 factor C2a
US5882900A (en) 1992-09-10 1999-03-16 Gruppo Lepetit S.P.A. Process for the selective increase of production of antibiotic GE 2270 factor a by adding vitamin B12 to nutrient medium
JPH08504782A (ja) 1992-12-22 1996-05-21 グルポ・レペチツト・エス・ピー・エイ 抗生物質ｇｅ３７４６８ａ、ｂ及びｃ
WO1996014427A1 (en) 1994-11-08 1996-05-17 Gruppo Lepetit S.P.A. Microbial transformation process for obtaining antibiotic ge 2270 factor d¿2?
ES2115424T3 (es) 1995-02-07 1998-06-16 Biosearch Italia Spa Derivados prolin-amidicos basicos de los antibioticos ge 2270 y similares a ge 2270.
JP3518606B2 (ja) 1995-02-07 2004-04-12 バイオサーチ・イタリア・ソチエタ・ペル・アチオニ Ｇｅ２２７０及びｇｅ２２７０−様抗生物質の塩基性オキサゾリン−アミド誘導体
HUP9901007A3 (en) 1996-02-14 1999-11-29 Vicuron Pharmaceuticals Inc Ki Derivatives of antibiotic ge2270 factors c2a, d2 and e
JPH1059997A (ja) 1996-08-22 1998-03-03 Microbial Chem Res Found アミチアマイシンアミド誘導体
JP4723857B2 (ja) 2002-06-17 2011-07-13 ヴィキュロン ファーマシューティカルズ インコーポレイテッド アクネの治療のためのｇｅ２２７０因子ａ３のアミド誘導体の使用
EP1793812A4 (en) 2004-09-22 2009-08-26 Merck & Co Inc ANTIBIOTIC COMPOUND
WO2007007399A1 (ja) * 2005-07-13 2007-01-18 Taisho Pharmaceutical Co., Ltd. チアゾール系化合物
AR060977A1 (es) * 2006-05-31 2008-07-23 Novartis Ag Aminotiazoles y sus usos
JP5230647B2 (ja) 2006-12-20 2013-07-10 ノバルティス アーゲー アミノチアゾール大環状分子、抗菌化合物としてのその使用およびその製造法
CN101772506B (zh) 2007-06-04 2014-02-12 诺华股份有限公司 大环化合物及其用途
JP5286366B2 (ja) * 2007-12-12 2013-09-11 ノバルティス アーゲー アミノチアゾール類およびその使用

Also Published As

Publication number Publication date
BRPI0821138A2 (pt) 2015-06-16
JP2013189468A (ja) 2013-09-26
GT201000166A (es) 2012-04-30
MA31869B1 (fr) 2010-11-01
CR11469A (es) 2010-07-09
TW200932256A (en) 2009-08-01
TN2010000254A1 (en) 2011-11-11
EA201000890A1 (ru) 2011-02-28
CA2708793C (en) 2016-06-21
EA020205B1 (ru) 2014-09-30
KR101187111B1 (ko) 2012-09-28
US20140274878A1 (en) 2014-09-18
US8426356B2 (en) 2013-04-23
CN101945866A (zh) 2011-01-12
CU23908B1 (es) 2013-06-28
PE20091108A1 (es) 2009-08-24
EA201400280A1 (ru) 2014-08-29
EP2229386B1 (en) 2015-06-03
ES2542878T3 (es) 2015-08-12
HN2010001176A (es) 2012-12-10
KR20120047335A (ko) 2012-05-11
NZ585788A (en) 2011-07-29
JP5286366B2 (ja) 2013-09-11
CL2008003688A1 (es) 2009-06-19
US20170015704A1 (en) 2017-01-19
CN101945866B (zh) 2013-06-19
ECSP10010244A (es) 2010-07-30
IL206104A0 (en) 2010-11-30
WO2009074605A1 (en) 2009-06-18
KR20100090809A (ko) 2010-08-17
CA2708793A1 (en) 2009-06-18
AR069628A1 (es) 2010-02-03
AU2008334659A1 (en) 2009-06-18
JP2011506394A (ja) 2011-03-03
TWI430804B (zh) 2014-03-21
IL206104A (en) 2015-03-31
MY156466A (en) 2016-02-26
US20130231275A1 (en) 2013-09-05
CO6290661A2 (es) 2011-06-20
US9492496B2 (en) 2016-11-15
US20090156628A1 (en) 2009-06-18
EP2229386A1 (en) 2010-09-22

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Legal Events

Date Code Title Description
FG Grant of patent
FD Lapse (for not paying fees)