CR8550A - Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo - Google Patents
Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfoniloInfo
- Publication number
- CR8550A CR8550A CR8550A CR8550A CR8550A CR 8550 A CR8550 A CR 8550A CR 8550 A CR8550 A CR 8550A CR 8550 A CR8550 A CR 8550A CR 8550 A CR8550 A CR 8550A
- Authority
- CR
- Costa Rica
- Prior art keywords
- preparation
- heteroarilalquilsulfonilo
- halogenuros
- aryl
- procedures
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
- C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
La presente invencion provee procedimientos de preparacion de halogenuros de arilalquilsulfonilo y halogenuros de heteroarilalquilsulfonilo de la formula Ar-R-SO2-X, que son utiles como intermediarios en la preparacion de agentes farmaceuticos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54760004P | 2004-02-25 | 2004-02-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR8550A true CR8550A (es) | 2007-02-05 |
Family
ID=34910921
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR8550A CR8550A (es) | 2004-02-25 | 2006-08-08 | Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo |
Country Status (24)
Country | Link |
---|---|
US (1) | US7321061B2 (es) |
EP (1) | EP1718605B1 (es) |
JP (1) | JP2007523954A (es) |
CN (1) | CN1922136A (es) |
AR (1) | AR048239A1 (es) |
AT (1) | ATE433955T1 (es) |
AU (1) | AU2005217619A1 (es) |
BR (1) | BRPI0507979A (es) |
CA (1) | CA2555247A1 (es) |
CO (1) | CO5720992A2 (es) |
CR (1) | CR8550A (es) |
DE (1) | DE602005014942D1 (es) |
EC (1) | ECSP066797A (es) |
ES (1) | ES2326746T3 (es) |
GT (1) | GT200500031A (es) |
IL (1) | IL177432A0 (es) |
NO (1) | NO20063611L (es) |
PA (1) | PA8624401A1 (es) |
PE (1) | PE20060018A1 (es) |
RU (1) | RU2006129650A (es) |
SV (1) | SV2005002015A (es) |
TW (1) | TW200602298A (es) |
WO (1) | WO2005082843A1 (es) |
ZA (1) | ZA200607097B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2466983C2 (ru) | 2005-07-21 | 2012-11-20 | Вайет | Способ синтеза сульфонилгалогенидов и сульфонамидов из солей сульфоновых кислот |
TW200824712A (en) * | 2006-10-31 | 2008-06-16 | Wyeth Corp | Liquid formulations of phospholipase enzyme inhibitors |
CL2007003146A1 (es) * | 2006-10-31 | 2008-01-25 | Wyeth Corp | Composición farmacéutica que comprende un compuesto derivado de indol y un sistema portador que comprende 15-25% de un mejorador de la viscosidad, 5-15% de un solubilizante, 10-50% de un diluyente y 1-10% de un estabilizante; proceso de preparación; y forma de dosificación. |
US20120116121A1 (en) * | 2009-07-30 | 2012-05-10 | Dow Global Technologies Llc | Process for the sulfochlorination of hydrocarbons |
CN102241613B (zh) * | 2011-05-09 | 2013-06-05 | 南通维立科化工有限公司 | 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法 |
CN102295587A (zh) * | 2011-05-26 | 2011-12-28 | 安徽丰乐农化有限责任公司 | 对甲基苯磺酰氯的制备新工艺 |
CN102976988B (zh) * | 2012-12-24 | 2014-06-18 | 三门峡奥科化工有限公司 | 2-萘硫酚的合成工艺 |
KR102122111B1 (ko) * | 2017-09-01 | 2020-06-11 | 주식회사 엘지화학 | 대체 용매의 선정 방법 |
CN111718286A (zh) * | 2020-07-23 | 2020-09-29 | 邓博天 | 一种带供电基团芳烃磺酰氯的工业化生产方法 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE48722C (de) * | Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 | Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid | ||
DE150313C (es) * | ||||
US2199568A (en) * | 1938-06-11 | 1940-05-07 | Gen Aniline & Film Corp | Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid |
US2507408A (en) | 1948-03-05 | 1950-05-09 | Rhone Poulenc Sa | 1-alkylsulfonyl-4-alkyl piperazines |
US2888486A (en) | 1953-11-20 | 1959-05-26 | Du Pont | Process for producing aromatic sulfonyl halides |
DE2545644A1 (de) * | 1975-10-11 | 1977-04-14 | Bayer Ag | Verfahren zur herstellung von sulfonsaeuren |
US4150049A (en) * | 1975-11-05 | 1979-04-17 | The Government Of The United States | Esters of aromatic sulfonic acids |
JPS5277030A (en) * | 1975-12-23 | 1977-06-29 | Toyo Pharma Kk | Production of novel benzyl sulphonic acid derivatives |
JPH09295962A (ja) * | 1996-03-08 | 1997-11-18 | Nagase & Co Ltd | 2,2−ジ置換−エタンスルホン酸誘導体およびその塩 |
DE19838516A1 (de) * | 1998-08-25 | 2000-03-09 | Degussa | Verfahren zur Herstellung von Sulfonylhalogeniden |
JP2000072739A (ja) * | 1998-09-01 | 2000-03-07 | Tanabe Seiyaku Co Ltd | スルホン酸類またはその塩の製法 |
DK1451154T3 (da) | 2001-12-03 | 2008-05-19 | Wyeth Corp | Inhibitorer af cytosolisk phospholipase A2 |
RU2466983C2 (ru) | 2005-07-21 | 2012-11-20 | Вайет | Способ синтеза сульфонилгалогенидов и сульфонамидов из солей сульфоновых кислот |
-
2005
- 2005-02-22 AR ARP050100642A patent/AR048239A1/es not_active Application Discontinuation
- 2005-02-23 PA PA20058624401A patent/PA8624401A1/es unknown
- 2005-02-23 EP EP05713940A patent/EP1718605B1/en not_active Expired - Lifetime
- 2005-02-23 AU AU2005217619A patent/AU2005217619A1/en not_active Abandoned
- 2005-02-23 DE DE602005014942T patent/DE602005014942D1/de not_active Expired - Lifetime
- 2005-02-23 PE PE2005000213A patent/PE20060018A1/es not_active Application Discontinuation
- 2005-02-23 AT AT05713940T patent/ATE433955T1/de not_active IP Right Cessation
- 2005-02-23 ES ES05713940T patent/ES2326746T3/es not_active Expired - Lifetime
- 2005-02-23 TW TW094105341A patent/TW200602298A/zh unknown
- 2005-02-23 BR BRPI0507979-9A patent/BRPI0507979A/pt not_active IP Right Cessation
- 2005-02-23 CN CNA2005800058622A patent/CN1922136A/zh active Pending
- 2005-02-23 GT GT200500031A patent/GT200500031A/es unknown
- 2005-02-23 RU RU2006129650/04A patent/RU2006129650A/ru not_active Application Discontinuation
- 2005-02-23 US US11/064,241 patent/US7321061B2/en not_active Expired - Fee Related
- 2005-02-23 SV SV2005002015A patent/SV2005002015A/es not_active Application Discontinuation
- 2005-02-23 WO PCT/US2005/005624 patent/WO2005082843A1/en active Application Filing
- 2005-02-23 CA CA002555247A patent/CA2555247A1/en not_active Abandoned
- 2005-02-23 JP JP2007500927A patent/JP2007523954A/ja active Pending
-
2006
- 2006-08-08 CR CR8550A patent/CR8550A/es not_active Application Discontinuation
- 2006-08-09 NO NO20063611A patent/NO20063611L/no not_active Application Discontinuation
- 2006-08-10 IL IL177432A patent/IL177432A0/en unknown
- 2006-08-23 CO CO06083312A patent/CO5720992A2/es not_active Application Discontinuation
- 2006-08-24 ZA ZA200607097A patent/ZA200607097B/xx unknown
- 2006-08-25 EC EC2006006797A patent/ECSP066797A/es unknown
Also Published As
Publication number | Publication date |
---|---|
SV2005002015A (es) | 2005-11-04 |
PE20060018A1 (es) | 2006-02-20 |
BRPI0507979A (pt) | 2007-07-24 |
WO2005082843A1 (en) | 2005-09-09 |
ATE433955T1 (de) | 2009-07-15 |
PA8624401A1 (es) | 2006-08-03 |
ECSP066797A (es) | 2006-11-16 |
CA2555247A1 (en) | 2005-09-09 |
AR048239A1 (es) | 2006-04-12 |
US20050187408A1 (en) | 2005-08-25 |
RU2006129650A (ru) | 2008-03-27 |
ZA200607097B (en) | 2009-08-26 |
JP2007523954A (ja) | 2007-08-23 |
AU2005217619A1 (en) | 2005-09-09 |
CO5720992A2 (es) | 2007-01-31 |
US7321061B2 (en) | 2008-01-22 |
DE602005014942D1 (de) | 2009-07-30 |
GT200500031A (es) | 2005-09-30 |
TW200602298A (en) | 2006-01-16 |
EP1718605A1 (en) | 2006-11-08 |
IL177432A0 (en) | 2006-12-10 |
NO20063611L (no) | 2006-09-21 |
EP1718605B1 (en) | 2009-06-17 |
ES2326746T3 (es) | 2009-10-19 |
CN1922136A (zh) | 2007-02-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal (granting procedure) |