[go: up one dir, main page]

ECSP066797A - Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo - Google Patents

Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo

Info

Publication number
ECSP066797A
ECSP066797A EC2006006797A ECSP066797A ECSP066797A EC SP066797 A ECSP066797 A EC SP066797A EC 2006006797 A EC2006006797 A EC 2006006797A EC SP066797 A ECSP066797 A EC SP066797A EC SP066797 A ECSP066797 A EC SP066797A
Authority
EC
Ecuador
Prior art keywords
preparation
heteroarilalquilsulfonilo
halogenures
aril
procedures
Prior art date
Application number
EC2006006797A
Other languages
English (en)
Inventor
Mousumi Ghosh
Mahmut Levent
Ronald S Mickalak
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ECSP066797A publication Critical patent/ECSP066797A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invención provee procedimientos de preparación de halogenuros de arilalquilsulfonilo y halogenuros de heteroarilalquilsulfonilo de la fórmula Ar-R-SO2-X, que son útiles como intermediarios en la preparación de agentes farmacéuticos.
EC2006006797A 2004-02-25 2006-08-25 Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo ECSP066797A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54760004P 2004-02-25 2004-02-25

Publications (1)

Publication Number Publication Date
ECSP066797A true ECSP066797A (es) 2006-11-16

Family

ID=34910921

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006006797A ECSP066797A (es) 2004-02-25 2006-08-25 Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo

Country Status (24)

Country Link
US (1) US7321061B2 (es)
EP (1) EP1718605B1 (es)
JP (1) JP2007523954A (es)
CN (1) CN1922136A (es)
AR (1) AR048239A1 (es)
AT (1) ATE433955T1 (es)
AU (1) AU2005217619A1 (es)
BR (1) BRPI0507979A (es)
CA (1) CA2555247A1 (es)
CO (1) CO5720992A2 (es)
CR (1) CR8550A (es)
DE (1) DE602005014942D1 (es)
EC (1) ECSP066797A (es)
ES (1) ES2326746T3 (es)
GT (1) GT200500031A (es)
IL (1) IL177432A0 (es)
NO (1) NO20063611L (es)
PA (1) PA8624401A1 (es)
PE (1) PE20060018A1 (es)
RU (1) RU2006129650A (es)
SV (1) SV2005002015A (es)
TW (1) TW200602298A (es)
WO (1) WO2005082843A1 (es)
ZA (1) ZA200607097B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2466983C2 (ru) 2005-07-21 2012-11-20 Вайет Способ синтеза сульфонилгалогенидов и сульфонамидов из солей сульфоновых кислот
TW200824712A (en) * 2006-10-31 2008-06-16 Wyeth Corp Liquid formulations of phospholipase enzyme inhibitors
CL2007003146A1 (es) * 2006-10-31 2008-01-25 Wyeth Corp Composición farmacéutica que comprende un compuesto derivado de indol y un sistema portador que comprende 15-25% de un mejorador de la viscosidad, 5-15% de un solubilizante, 10-50% de un diluyente y 1-10% de un estabilizante; proceso de preparación; y forma de dosificación.
US20120116121A1 (en) * 2009-07-30 2012-05-10 Dow Global Technologies Llc Process for the sulfochlorination of hydrocarbons
CN102241613B (zh) * 2011-05-09 2013-06-05 南通维立科化工有限公司 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法
CN102295587A (zh) * 2011-05-26 2011-12-28 安徽丰乐农化有限责任公司 对甲基苯磺酰氯的制备新工艺
CN102976988B (zh) * 2012-12-24 2014-06-18 三门峡奥科化工有限公司 2-萘硫酚的合成工艺
KR102122111B1 (ko) * 2017-09-01 2020-06-11 주식회사 엘지화학 대체 용매의 선정 방법
CN111718286A (zh) * 2020-07-23 2020-09-29 邓博天 一种带供电基团芳烃磺酰氯的工业化生产方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE48722C (de) * Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid
DE150313C (es) *
US2199568A (en) * 1938-06-11 1940-05-07 Gen Aniline & Film Corp Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid
US2507408A (en) 1948-03-05 1950-05-09 Rhone Poulenc Sa 1-alkylsulfonyl-4-alkyl piperazines
US2888486A (en) 1953-11-20 1959-05-26 Du Pont Process for producing aromatic sulfonyl halides
DE2545644A1 (de) * 1975-10-11 1977-04-14 Bayer Ag Verfahren zur herstellung von sulfonsaeuren
US4150049A (en) * 1975-11-05 1979-04-17 The Government Of The United States Esters of aromatic sulfonic acids
JPS5277030A (en) * 1975-12-23 1977-06-29 Toyo Pharma Kk Production of novel benzyl sulphonic acid derivatives
JPH09295962A (ja) * 1996-03-08 1997-11-18 Nagase & Co Ltd ２，２−ジ置換−エタンスルホン酸誘導体およびその塩
DE19838516A1 (de) * 1998-08-25 2000-03-09 Degussa Verfahren zur Herstellung von Sulfonylhalogeniden
JP2000072739A (ja) * 1998-09-01 2000-03-07 Tanabe Seiyaku Co Ltd スルホン酸類またはその塩の製法
DK1451154T3 (da) 2001-12-03 2008-05-19 Wyeth Corp Inhibitorer af cytosolisk phospholipase A2
RU2466983C2 (ru) 2005-07-21 2012-11-20 Вайет Способ синтеза сульфонилгалогенидов и сульфонамидов из солей сульфоновых кислот

Also Published As

Publication number Publication date
SV2005002015A (es) 2005-11-04
PE20060018A1 (es) 2006-02-20
BRPI0507979A (pt) 2007-07-24
WO2005082843A1 (en) 2005-09-09
ATE433955T1 (de) 2009-07-15
PA8624401A1 (es) 2006-08-03
CA2555247A1 (en) 2005-09-09
AR048239A1 (es) 2006-04-12
US20050187408A1 (en) 2005-08-25
CR8550A (es) 2007-02-05
RU2006129650A (ru) 2008-03-27
ZA200607097B (en) 2009-08-26
JP2007523954A (ja) 2007-08-23
AU2005217619A1 (en) 2005-09-09
CO5720992A2 (es) 2007-01-31
US7321061B2 (en) 2008-01-22
DE602005014942D1 (de) 2009-07-30
GT200500031A (es) 2005-09-30
TW200602298A (en) 2006-01-16
EP1718605A1 (en) 2006-11-08
IL177432A0 (en) 2006-12-10
NO20063611L (no) 2006-09-21
EP1718605B1 (en) 2009-06-17
ES2326746T3 (es) 2009-10-19
CN1922136A (zh) 2007-02-28

Similar Documents

Publication Publication Date Title
ECSP066797A (es) Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo
CR9223A (es) 18-metil-19-nor-17-pregn-4-en-21, 17-carbolactonas,asi como preparaciones farmaceuticas que las contienen
CR8919A (es) Analogos de tetrapeptidos
CY1109998T1 (el) Ενδυναμωτες υποδοχεων γλουταμινικου
CL2009000349A1 (es) Compuestos derivados de 4,5-dihidro-oxazol-2-ilamina; procedimiento de preparacion; composicion farmaceutica; y su uso para el tratamiento de la enfermedad de alzheimer.
NO20092611L (no) Krystallinsk faststoff Rasagilin base
TW200716647A (en) Synthesis of (R)-N-methylnaltrexone
CY1114271T1 (el) Αντισωματα εξουδετερωσης, ανθρωπινου κυτταρομεγαλοϊου και χρηση αυτων
SV2010003662A (es) Derivados de azetidina y ciclobutano como inhibidores de jak ref. x-19081
CY1113024T1 (el) Σπειροκυκλικα παραγωγα κυκλοεξανιου για τη θεραπεια της εξαρτησης ουσιων
UY29767A1 (es) Derivados de benzotiazolonas, procesos para su preparación, composiciones farmacéuticas que los contienen y aplicaciones
PA8667201A1 (es) Nuevos compuestos farmaceuticos
CR9786A (es) Compuestos de bencimidazol-tiofeno
TW200730518A (en) Crystalline forms of docetaxel and processes for their preparation
WO2010017387A3 (en) Lapatinib, salts thereof, processes and intermediates for their preparation
CY1122416T1 (el) Φαρμακα τα οποια περιεχουν κρυσταλλικες τροποποιησεις (1r,2r)-3-(3-δimeθyλamino-1-αιθυλο-2-μεθυλο-προπυλο)-φαινολης
DOP2006000087A (es) Compuestos heteroaromaticos acilaminobiciclicos y sus usos
UY33276A (es) Compuestos de amino-oxazinas y amino-dihidrotiazina como moduladores de beta-secretasa y métodos de uso
SE0401762D0 (sv) Novel compounds
ATE435209T1 (de) Verfahren zur herstellung von montelukast-natrium
ECSP11010956A (es) Compuestos enlazados con azufre para el tratamiento de enfermedades y trastornos oftalmicos
EA200701867A1 (ru) Хинолиноновые соединения в качестве агонистов рецептора 5-ht
UY29036A1 (es) Derivados de oxopiperidina, su preparacion y su aplicacion en terapeutica
MX367327B (es) Formulaciones, sales y polimorfos de transnorsertralina y usos de los mismos.
PA8659601A1 (es) Procedimiento para la preparacion de alcoholes aminoetoxibencilicos