CL2007003635A1 - Compuestos derivados de 6-amino-purin-8-ona; proceso de preparacion; composicion farmaceutica; proceso para preparar la composicion farmaceutica; y uso en el tratamiento de enfermedades alergicas, virales o cancer. - Google Patents
Compuestos derivados de 6-amino-purin-8-ona; proceso de preparacion; composicion farmaceutica; proceso para preparar la composicion farmaceutica; y uso en el tratamiento de enfermedades alergicas, virales o cancer.Info
- Publication number
- CL2007003635A1 CL2007003635A1 CL200703635A CL2007003635A CL2007003635A1 CL 2007003635 A1 CL2007003635 A1 CL 2007003635A1 CL 200703635 A CL200703635 A CL 200703635A CL 2007003635 A CL2007003635 A CL 2007003635A CL 2007003635 A1 CL2007003635 A1 CL 2007003635A1
- Authority
- CL
- Chile
- Prior art keywords
- pharmaceutical composition
- purin
- ona
- allergic
- viral
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 2
- 206010028980 Neoplasm Diseases 0.000 title 1
- 230000000172 allergic effect Effects 0.000 title 1
- 208000010668 atopic eczema Diseases 0.000 title 1
- 201000011510 cancer Diseases 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
- 230000003612 virological effect Effects 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P11/02—Nasal agents, e.g. decongestants
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Molecular Biology (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biotechnology (AREA)
- Rheumatology (AREA)
- Transplantation (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- AIDS & HIV (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86993006P | 2006-12-14 | 2006-12-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2007003635A1 true CL2007003635A1 (es) | 2008-08-22 |
Family
ID=39135145
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL200703635A CL2007003635A1 (es) | 2006-12-14 | 2007-12-14 | Compuestos derivados de 6-amino-purin-8-ona; proceso de preparacion; composicion farmaceutica; proceso para preparar la composicion farmaceutica; y uso en el tratamiento de enfermedades alergicas, virales o cancer. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8067411B2 (es) |
| EP (1) | EP2121693B1 (es) |
| JP (1) | JP5506393B2 (es) |
| AR (1) | AR064345A1 (es) |
| CL (1) | CL2007003635A1 (es) |
| PE (1) | PE20081480A1 (es) |
| TW (1) | TW200831105A (es) |
| UY (1) | UY30789A1 (es) |
| WO (1) | WO2008071976A1 (es) |
Families Citing this family (34)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4472693B2 (ja) * | 2004-03-26 | 2010-06-02 | 大日本住友製薬株式会社 | ９置換−８−オキソアデニン化合物 |
| TW200801003A (en) * | 2005-09-16 | 2008-01-01 | Astrazeneca Ab | Novel compounds |
| JPWO2007034817A1 (ja) * | 2005-09-22 | 2009-03-26 | 大日本住友製薬株式会社 | 新規アデニン化合物 |
| WO2008004948A1 (en) * | 2006-07-05 | 2008-01-10 | Astrazeneca Ab | 8-oxoadenine derivatives acting as modulators of tlr7 |
| TW200831105A (en) * | 2006-12-14 | 2008-08-01 | Astrazeneca Ab | Novel compounds |
| EP2125792B1 (en) * | 2007-02-19 | 2010-12-01 | GlaxoSmithKline LLC | Purine derivatives as immunomodulators |
| SI2132209T1 (sl) * | 2007-03-19 | 2014-05-30 | Astrazeneca Ab | Spojine 9-substituiranega-8-okso-adenina, kot modulatorji Toll-like receptorja (TLR7) |
| ES2373616T3 (es) * | 2007-03-19 | 2012-02-07 | Astrazeneca Ab | Compuestos de 8-oxo-adenina 9 sustituidos como moduladores del receptor de tipo toll (tlr7). |
| WO2008114819A1 (ja) * | 2007-03-20 | 2008-09-25 | Dainippon Sumitomo Pharma Co., Ltd. | 新規アデニン化合物 |
| TW200902018A (en) * | 2007-03-20 | 2009-01-16 | Dainippon Sumitomo Pharma Co | Novel adenine compound |
| KR20100016289A (ko) | 2007-05-08 | 2010-02-12 | 아스트라제네카 아베 | 면역-조정 특성의 이미다조퀴놀린 |
| WO2009005687A1 (en) | 2007-06-29 | 2009-01-08 | Gilead Sciences, Inc. | Purine derivatives and their use as modulators of toll-like receptor 7 |
| PE20091236A1 (es) * | 2007-11-22 | 2009-09-16 | Astrazeneca Ab | Derivados de pirimidina como immunomoduladores de tlr7 |
| UY31531A1 (es) | 2007-12-17 | 2009-08-03 | Sales derivadas de 8-oxoadenina composiciones farmacéuticas que las contienen y su uso en terapia como moduladores de receptor tipo toll (tlr) | |
| KR20100125245A (ko) * | 2008-01-17 | 2010-11-30 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 아데닌 화합물의 제조 방법 |
| JPWO2009091031A1 (ja) * | 2008-01-17 | 2011-05-26 | 大日本住友製薬株式会社 | アデニン化合物の製造方法 |
| UA103195C2 (uk) | 2008-08-11 | 2013-09-25 | Глаксосмитклайн Ллк | Похідні пурину для застосування у лікуванні алергій, запальних та інфекційних захворювань |
| PE20120106A1 (es) | 2008-12-09 | 2012-02-20 | Gilead Sciences Inc | Moduladores de receptores tipo toll |
| GB0908772D0 (en) * | 2009-05-21 | 2009-07-01 | Astrazeneca Ab | New salts 756 |
| AP3103A (en) | 2009-10-22 | 2015-01-31 | Gilead Sciences Inc | Derivatives of purine or deazapurine useful for the treatment of (inter alia)viral infections |
| WO2011068233A1 (en) * | 2009-12-03 | 2011-06-09 | Dainippon Sumitomo Pharma Co., Ltd. | Imidazoquinolines which act via toll - like receptors (tlr) |
| US20110150836A1 (en) * | 2009-12-22 | 2011-06-23 | Gilead Sciences, Inc. | Methods of treating hbv and hcv infection |
| CN103370317B (zh) | 2010-12-16 | 2015-10-07 | 阿斯利康(瑞典)有限公司 | 可用于治疗的咪唑并[4,5-c]喹啉-1-基衍生物 |
| EP2651943B1 (en) * | 2010-12-17 | 2017-03-22 | Sumitomo Dainippon Pharma Co., Ltd. | Purine derivatives |
| BR112014001425A2 (pt) | 2011-07-22 | 2017-11-21 | Glaxosmithkline Llc | forma de dosagem farmacêutica, composição farmacêutica, e, composto (i) ou sal farmaceuticamente aceitável do mesmo |
| CA2871589C (en) | 2012-05-18 | 2020-12-22 | Seiji Hori | Pyrimidine carboxylic acid derivatives and their use as tlr7 agonists |
| US9555036B2 (en) | 2012-08-24 | 2017-01-31 | Glaxosmithkline Llc | Pyrazolopyrimidine compounds |
| KR20150085080A (ko) | 2012-11-20 | 2015-07-22 | 글락소스미스클라인 엘엘씨 | 신규 화합물 |
| EP2922547B1 (en) | 2012-11-20 | 2017-03-08 | Glaxosmithkline LLC | Novel compounds |
| SG11201503282RA (en) | 2012-11-20 | 2015-06-29 | Glaxosmithkline Llc | Novel compounds |
| US20170001988A1 (en) * | 2013-11-27 | 2017-01-05 | The United States Of America, As Represented By The Secretary, Department Of Health And Human | Piperidine and piperazine derivatives and their use in treating viral infections and cancer |
| SI3166607T1 (sl) | 2014-07-11 | 2023-01-31 | Gilead Sciences, Inc. | Modulatorji toličnih receptorjev za zdravljenje HIV-a |
| EP3194401B1 (en) | 2014-09-16 | 2020-10-21 | Gilead Sciences, Inc. | Solid forms of a toll-like receptor modulator |
| JP7442192B2 (ja) * | 2018-03-03 | 2024-03-04 | 国立大学法人 東京大学 | がん特異的酵素活性を利用したプロドラッグ型抗がん剤 |
Family Cites Families (78)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1375162A (es) | 1970-10-22 | 1974-11-27 | ||
| GB1546937A (en) | 1976-07-29 | 1979-05-31 | Beecham Group Ltd | 2,4-diaminopyrimidine derivatives |
| SE8404768L (sv) | 1983-09-27 | 1985-03-28 | Ceskoslovenska Akademie Ved | 9-(aminoalkyl)-8-hydroxiadeniner och sett for deras framstellning |
| ZA848968B (en) | 1983-11-18 | 1986-06-25 | Riker Laboratories Inc | 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c)quinolin-4-amines |
| IL73534A (en) | 1983-11-18 | 1990-12-23 | Riker Laboratories Inc | 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds |
| IL78643A0 (en) | 1985-05-02 | 1986-08-31 | Wellcome Found | Purine derivatives,their preparation and pharmaceutical compositions containing them |
| DE3603577A1 (de) | 1986-02-06 | 1987-08-13 | Joachim K Prof Dr Seydel | Neue substituierte 2,4-diamino-5-benzylpyrimidine, deren herstellung und deren verwendung als arzneimittel mit antibakterieller wirksamkeit |
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-
2007
- 2007-12-06 TW TW096146507A patent/TW200831105A/zh unknown
- 2007-12-13 EP EP07848528A patent/EP2121693B1/en not_active Not-in-force
- 2007-12-13 UY UY30789A patent/UY30789A1/es unknown
- 2007-12-13 PE PE2007001780A patent/PE20081480A1/es not_active Application Discontinuation
- 2007-12-13 AR ARP070105613A patent/AR064345A1/es unknown
- 2007-12-13 JP JP2009540862A patent/JP5506393B2/ja not_active Expired - Fee Related
- 2007-12-13 WO PCT/GB2007/004786 patent/WO2008071976A1/en active Application Filing
- 2007-12-13 US US11/955,984 patent/US8067411B2/en not_active Expired - Fee Related
- 2007-12-14 CL CL200703635A patent/CL2007003635A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US8067411B2 (en) | 2011-11-29 |
| US20080300244A1 (en) | 2008-12-04 |
| JP5506393B2 (ja) | 2014-05-28 |
| WO2008071976A1 (en) | 2008-06-19 |
| TW200831105A (en) | 2008-08-01 |
| EP2121693B1 (en) | 2012-08-08 |
| EP2121693A1 (en) | 2009-11-25 |
| PE20081480A1 (es) | 2008-12-07 |
| AR064345A1 (es) | 2009-04-01 |
| JP2010513257A (ja) | 2010-04-30 |
| UY30789A1 (es) | 2008-07-31 |
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