BRPI0412999A - 2-aminotetralina substituìda para tratamento de depressão - Google Patents
2-aminotetralina substituìda para tratamento de depressãoInfo
- Publication number
- BRPI0412999A BRPI0412999A BRPI0412999-7A BRPI0412999A BRPI0412999A BR PI0412999 A BRPI0412999 A BR PI0412999A BR PI0412999 A BRPI0412999 A BR PI0412999A BR PI0412999 A BRPI0412999 A BR PI0412999A
- Authority
- BR
- Brazil
- Prior art keywords
- aminotetraline
- substituted
- depression treatment
- depression
- treatment
- Prior art date
Links
- LCGFVWKNXLRFIF-UHFFFAOYSA-N 1,2,3,4-tetrahydronaphthalen-2-amine Chemical class C1=CC=C2CC(N)CCC2=C1 LCGFVWKNXLRFIF-UHFFFAOYSA-N 0.000 title 1
- 208000020401 Depressive disease Diseases 0.000 title 1
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Organic Chemistry (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Abstract
"2-AMINOTETRALINA SUBSTITUìDA PARA TRATAMENTO DE DEPRESSãO". A invenção refere-se ao uso de um composto da fórmula geral (I) e aos seus sais farmaceuticamente aceitáveis, racematos ou enantiómeros puros para a produção de um medicamento usado para tratar depressão. Os substituintes são definidos como na descrição.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10334187A DE10334187A1 (de) | 2003-07-26 | 2003-07-26 | Substituierte 2-Aminotetraline zur Behandlung von Depressionen |
PCT/EP2004/008169 WO2005009425A1 (de) | 2003-07-26 | 2004-07-22 | Substituierte 2-aminotetraline zur behandlung von depressionen |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0412999A true BRPI0412999A (pt) | 2006-10-03 |
Family
ID=34088861
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0412999-7A BRPI0412999A (pt) | 2003-07-26 | 2004-07-22 | 2-aminotetralina substituìda para tratamento de depressão |
Country Status (19)
Country | Link |
---|---|
US (1) | US20070072917A1 (pt) |
EP (1) | EP1648433B1 (pt) |
JP (1) | JP2007500155A (pt) |
KR (1) | KR101160699B1 (pt) |
CN (1) | CN1832734B (pt) |
AT (1) | ATE373474T1 (pt) |
AU (1) | AU2004258698A1 (pt) |
BR (1) | BRPI0412999A (pt) |
CA (1) | CA2532804C (pt) |
DE (2) | DE10334187A1 (pt) |
EA (1) | EA009870B1 (pt) |
ES (1) | ES2291914T3 (pt) |
IL (1) | IL173062A (pt) |
IS (1) | IS2696B (pt) |
MX (1) | MXPA06000865A (pt) |
NO (1) | NO20060847L (pt) |
UA (1) | UA83233C2 (pt) |
WO (1) | WO2005009425A1 (pt) |
ZA (1) | ZA200600343B (pt) |
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DE10041478A1 (de) | 2000-08-24 | 2002-03-14 | Sanol Arznei Schwarz Gmbh | Neue pharmazeutische Zusammensetzung |
US20030027793A1 (en) * | 2001-05-08 | 2003-02-06 | Thomas Lauterback | Transdermal treatment of parkinson's disease |
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US8246980B2 (en) * | 2002-07-30 | 2012-08-21 | Ucb Pharma Gmbh | Transdermal delivery system |
DE10234673B4 (de) | 2002-07-30 | 2007-08-16 | Schwarz Pharma Ag | Heißschmelz-TTS zur Verabreichung von Rotigotin und Verfahren zu seiner Herstellung sowie Verwendung von Rotigotin bei der Herstellung eines TTS im Heißschmelzverfahren |
US8246979B2 (en) * | 2002-07-30 | 2012-08-21 | Ucb Pharma Gmbh | Transdermal delivery system for the administration of rotigotine |
US8211462B2 (en) | 2002-07-30 | 2012-07-03 | Ucb Pharma Gmbh | Hot-melt TTS for administering rotigotine |
PT1426049E (pt) | 2002-12-02 | 2005-09-30 | Sanol Arznei Schwarz Gmbh | Administracao iontoforetica de rotigotina para o tratamento da doenca de parkinson |
DE10261696A1 (de) * | 2002-12-30 | 2004-07-15 | Schwarz Pharma Ag | Vorrichtung zur transdermalen Verabreichung von Rotigotin-Base |
DE10334188B4 (de) * | 2003-07-26 | 2007-07-05 | Schwarz Pharma Ag | Verwendung von Rotigotin zur Behandlung von Depressionen |
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MY165575A (en) * | 2007-11-28 | 2018-04-05 | Ucb Pharma Gmbh | Polymorphic form of rotigotine |
EP2281559A1 (en) * | 2009-06-26 | 2011-02-09 | UCB Pharma GmbH | Pharmaceutical composition comprising rotigotine salts (acid or Na), especially for iontophoresis |
PL3257504T3 (pl) * | 2009-12-22 | 2024-10-21 | UCB Biopharma SRL | Poliwinylopirolidon do stabilizacji stałej dyspersji niekrystalicznej postaci rotygotyny |
-
2003
- 2003-07-26 DE DE10334187A patent/DE10334187A1/de not_active Ceased
-
2004
- 2004-07-22 AU AU2004258698A patent/AU2004258698A1/en not_active Abandoned
- 2004-07-22 JP JP2006521477A patent/JP2007500155A/ja active Pending
- 2004-07-22 DE DE502004005033T patent/DE502004005033D1/de not_active Expired - Lifetime
- 2004-07-22 AT AT04763387T patent/ATE373474T1/de not_active IP Right Cessation
- 2004-07-22 CA CA2532804A patent/CA2532804C/en not_active Expired - Fee Related
- 2004-07-22 BR BRPI0412999-7A patent/BRPI0412999A/pt not_active IP Right Cessation
- 2004-07-22 CN CN2004800216477A patent/CN1832734B/zh not_active Expired - Fee Related
- 2004-07-22 KR KR1020067001812A patent/KR101160699B1/ko not_active Expired - Fee Related
- 2004-07-22 EA EA200600223A patent/EA009870B1/ru not_active IP Right Cessation
- 2004-07-22 UA UAA200600562A patent/UA83233C2/ru unknown
- 2004-07-22 US US10/565,713 patent/US20070072917A1/en not_active Abandoned
- 2004-07-22 EP EP04763387A patent/EP1648433B1/de not_active Expired - Lifetime
- 2004-07-22 MX MXPA06000865A patent/MXPA06000865A/es active IP Right Grant
- 2004-07-22 WO PCT/EP2004/008169 patent/WO2005009425A1/de active IP Right Grant
- 2004-07-22 ES ES04763387T patent/ES2291914T3/es not_active Expired - Lifetime
-
2006
- 2006-01-10 IL IL173062A patent/IL173062A/en not_active IP Right Cessation
- 2006-01-10 ZA ZA200600343A patent/ZA200600343B/xx unknown
- 2006-01-12 IS IS8230A patent/IS2696B/is unknown
- 2006-02-21 NO NO20060847A patent/NO20060847L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
ES2291914T3 (es) | 2008-03-01 |
CA2532804C (en) | 2012-09-25 |
KR20060052898A (ko) | 2006-05-19 |
DE502004005033D1 (de) | 2007-10-31 |
EA200600223A1 (ru) | 2006-08-25 |
JP2007500155A (ja) | 2007-01-11 |
DE10334187A1 (de) | 2005-03-03 |
CN1832734A (zh) | 2006-09-13 |
WO2005009425A1 (de) | 2005-02-03 |
EA009870B1 (ru) | 2008-04-28 |
EP1648433A1 (de) | 2006-04-26 |
AU2004258698A1 (en) | 2005-02-03 |
US20070072917A1 (en) | 2007-03-29 |
EP1648433B1 (de) | 2007-09-19 |
KR101160699B1 (ko) | 2012-06-28 |
IS2696B (is) | 2010-11-15 |
NO20060847L (no) | 2006-02-21 |
CN1832734B (zh) | 2010-09-29 |
MXPA06000865A (es) | 2006-05-04 |
HK1091121A1 (en) | 2007-01-12 |
UA83233C2 (ru) | 2008-06-25 |
CA2532804A1 (en) | 2005-02-03 |
IL173062A0 (en) | 2006-06-11 |
ZA200600343B (en) | 2006-11-29 |
IL173062A (en) | 2011-12-29 |
IS8230A (is) | 2006-01-12 |
ATE373474T1 (de) | 2007-10-15 |
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