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BRPI0410638A - derivados de azitromicina - Google Patents

derivados de azitromicina

Info

Publication number
BRPI0410638A
BRPI0410638A BRPI0410638-5A BRPI0410638A BRPI0410638A BR PI0410638 A BRPI0410638 A BR PI0410638A BR PI0410638 A BRPI0410638 A BR PI0410638A BR PI0410638 A BRPI0410638 A BR PI0410638A
Authority
BR
Brazil
Prior art keywords
azithromycin
derivatives
azithromycin derivatives
azyromycin
manufacture
Prior art date
Application number
BRPI0410638-5A
Other languages
English (en)
Inventor
Albert Codony
Jose Diago
Rafael Garcia
Jordi Rifa
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of BRPI0410638A publication Critical patent/BRPI0410638A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

"DERIVADOS DE AZITROMICINA". A invenção refere-se a derivados de azitromicina, processos para fabricação dos mesmos, e composições farmacêuticas dos mesmos de preferência junto com azitromicina.
BRPI0410638-5A 2003-04-17 2004-04-16 derivados de azitromicina BRPI0410638A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US46360003P 2003-04-17 2003-04-17
US51128203P 2003-10-15 2003-10-15
PCT/EP2004/004053 WO2004092736A2 (en) 2003-04-17 2004-04-16 Derivatives of azithromycin

Publications (1)

Publication Number Publication Date
BRPI0410638A true BRPI0410638A (pt) 2006-06-13

Family

ID=33303125

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0410638-5A BRPI0410638A (pt) 2003-04-17 2004-04-16 derivados de azitromicina

Country Status (6)

Country Link
US (1) US7410952B2 (pt)
EP (1) EP1622922A2 (pt)
BR (1) BRPI0410638A (pt)
CA (1) CA2521462A1 (pt)
WO (1) WO2004092736A2 (pt)
ZA (1) ZA200507475B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011015219A1 (en) 2009-08-06 2011-02-10 Shifa Pharmed Industrial Group Co. Process for the purification of azithromycin by separation from its thermal degradation products and/or isomers
WO2012038372A1 (en) * 2010-09-20 2012-03-29 Novartis Ag Novel process for the preparation of 9-deoxo-9a-aza- 9a-homoerythromycin a modified in the c-4'' of the cladinose ring by an epoxide group
CN104558069B (zh) * 2014-12-31 2017-01-04 广东东阳光药业有限公司 大环内酯杂质的合成方法
CN104829662B (zh) * 2015-03-30 2017-11-07 石药集团欧意药业有限公司 一种阿奇霉素有关物质的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725385A (en) * 1970-11-02 1973-04-03 Abbott Lab Process for the demethylation of 3-amino macrolides
IT1306205B1 (it) * 1999-01-15 2001-05-30 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
EP1446010B1 (en) * 2001-10-18 2009-04-15 Teva Pharmaceutical Industries Ltd. Stabilized azithromycin compositions
CA2520192A1 (en) 2003-03-25 2004-10-14 Teva Pharmaceutical Industries Ltd. Degradation products of azithromycin, and methods for their identification

Also Published As

Publication number Publication date
WO2004092736A2 (en) 2004-10-28
CA2521462A1 (en) 2004-10-28
WO2004092736A3 (en) 2005-01-06
ZA200507475B (en) 2008-03-26
US7410952B2 (en) 2008-08-12
US20070043214A1 (en) 2007-02-22
EP1622922A2 (en) 2006-02-08

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Legal Events

Date Code Title Description
B08F Application fees: application dismissed [chapter 8.6 patent gazette]

Free format text: REFERENTE A 10A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2259 DE 22/04/2014.