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BR9916051A - Processo estereosseletivo para produzir agentes antineoplásticos - Google Patents

Processo estereosseletivo para produzir agentes antineoplásticos

Info

Publication number
BR9916051A
BR9916051A BR9916051-0A BR9916051A BR9916051A BR 9916051 A BR9916051 A BR 9916051A BR 9916051 A BR9916051 A BR 9916051A BR 9916051 A BR9916051 A BR 9916051A
Authority
BR
Brazil
Prior art keywords
antineoplastic agents
stereoselective process
produce antineoplastic
produce
stereoselective
Prior art date
Application number
BR9916051-0A
Other languages
English (en)
Inventor
James Abraham Aikins
Barbara Shreve Briggs
Tony Yantao Zhang
Milton Joseph Junior Zmijewski
Original Assignee
Lilly Co Eli
Univ Hawaii
Univ Wayne State
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli, Univ Hawaii, Univ Wayne State filed Critical Lilly Co Eli
Publication of BR9916051A publication Critical patent/BR9916051A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C07D273/08Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00 having two nitrogen atoms and more than one oxygen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Patente de Invenção: <B>"PROCESSO ESTEREOSSELETIVO PARA PRODUZIR AGENTES ANTINEOPLáSTICOS"<D>. Esta invenção fornece processos para preparar compostos de criptoficina de fórmula (II).
BR9916051-0A 1998-10-16 1999-10-15 Processo estereosseletivo para produzir agentes antineoplásticos BR9916051A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10466498P 1998-10-16 1998-10-16
PCT/US1999/024410 WO2000023429A2 (en) 1998-10-16 1999-10-15 Stereoselective process for producing cryptophycins

Publications (1)

Publication Number Publication Date
BR9916051A true BR9916051A (pt) 2001-08-14

Family

ID=22301706

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9916051-0A BR9916051A (pt) 1998-10-16 1999-10-15 Processo estereosseletivo para produzir agentes antineoplásticos

Country Status (10)

Country Link
EP (1) EP1127055A2 (pt)
JP (1) JP2002527509A (pt)
KR (1) KR20010099699A (pt)
AU (1) AU1123200A (pt)
BR (1) BR9916051A (pt)
CA (1) CA2347246A1 (pt)
HU (1) HUP0104027A3 (pt)
IL (1) IL142565A0 (pt)
TR (1) TR200101084T2 (pt)
WO (1) WO2000023429A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20120149895A1 (en) * 2009-04-01 2012-06-14 Lek Pharmaceuticals D.D. Process for dimethylation of active methylene groups
FR2947269B1 (fr) 2009-06-29 2013-01-18 Sanofi Aventis Nouveaux composes anticancereux
CN102140068B (zh) * 2010-01-30 2015-03-11 浙江华海药业股份有限公司 阿利吉仑中间体3-氨基-2,2-二甲基丙酰胺的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP737A (en) * 1995-03-07 1999-03-15 Univ Hawaii New cryptophycins from synthesis.
AU2058197A (en) * 1996-02-27 1997-09-16 Eli Lilly And Company Pharmaceutical compounds
CA2264557A1 (en) * 1996-09-06 1998-03-12 Eli Lilly And Company Process and novel intermediates
KR20000075671A (ko) * 1997-02-26 2000-12-26 피터 지. 스트링거 제약 화합물의 제조 방법

Also Published As

Publication number Publication date
TR200101084T2 (tr) 2001-09-21
AU1123200A (en) 2000-05-08
HUP0104027A3 (en) 2002-08-28
HUP0104027A2 (hu) 2002-03-28
EP1127055A2 (en) 2001-08-29
CA2347246A1 (en) 2000-04-27
KR20010099699A (ko) 2001-11-09
WO2000023429A2 (en) 2000-04-27
IL142565A0 (en) 2002-03-10
JP2002527509A (ja) 2002-08-27
WO2000023429A3 (en) 2000-07-27

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]