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BR0313796A - Processo para preparação de monoalquilaminocetonas - Google Patents

Processo para preparação de monoalquilaminocetonas

Info

Publication number
BR0313796A
BR0313796A BR0313796-1A BR0313796A BR0313796A BR 0313796 A BR0313796 A BR 0313796A BR 0313796 A BR0313796 A BR 0313796A BR 0313796 A BR0313796 A BR 0313796A
Authority
BR
Brazil
Prior art keywords
preparation
monoalkylaminoketones
monoalkylamino
ketones
formula
Prior art date
Application number
BR0313796-1A
Other languages
English (en)
Inventor
Kai Fabian
Claus-Peter Niesert
Joachim Kralik
Karl-Heinz Gluesenkamp
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31502148&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0313796(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of BR0313796A publication Critical patent/BR0313796A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C221/00—Preparation of compounds containing amino groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
    • C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
    • C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Furan Compounds (AREA)

Abstract

"PROCESSO PARA PREPARAçãO DE MONOALQUILAMINOCETONAS". A presente invenção refere-se a monoalquilaminocetonas da fórmula (I), onde R¬ 1¬ e R¬ 2¬ têm os significados indicados.
BR0313796-1A 2002-08-27 2003-08-01 Processo para preparação de monoalquilaminocetonas BR0313796A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10240026A DE10240026A1 (de) 2002-08-27 2002-08-27 Verfahren zur Herstellung von Monoalkylaminoketonen
PCT/EP2003/008514 WO2004020391A1 (de) 2002-08-27 2003-08-01 Verfahren zur herstellung von monoalkylaminoketonen

Publications (1)

Publication Number Publication Date
BR0313796A true BR0313796A (pt) 2005-09-27

Family

ID=31502148

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0313796-1A BR0313796A (pt) 2002-08-27 2003-08-01 Processo para preparação de monoalquilaminocetonas

Country Status (15)

Country Link
US (1) US7579484B2 (pt)
EP (1) EP1532101A1 (pt)
JP (1) JP4593275B2 (pt)
KR (1) KR101017885B1 (pt)
CN (1) CN100368384C (pt)
AU (1) AU2003260348B2 (pt)
BR (1) BR0313796A (pt)
CA (1) CA2497028A1 (pt)
DE (1) DE10240026A1 (pt)
HK (1) HK1081532A1 (pt)
MX (1) MXPA05002117A (pt)
PL (1) PL373599A1 (pt)
RU (1) RU2340595C2 (pt)
WO (1) WO2004020391A1 (pt)
ZA (1) ZA200502457B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004005239A1 (en) 2002-07-09 2004-01-15 Lonza Ag PROCESS FOR THE PREPARATION OF N-MONOSUBSTITUTED β-AMINO ALCOHOLS
DE10302595A1 (de) * 2003-01-22 2004-07-29 Basf Ag 3-Methylamino-1-(2-thienyl)-1-proganon, seine Herstellung und Verwendung
CN103214452B (zh) * 2013-05-07 2014-08-06 浙江丽晶化学有限公司 N-甲基-3-羟基-3-（2-噻吩基）-丙胺的制备方法
CN109134427B (zh) * 2018-10-24 2020-06-30 浙江乐普药业股份有限公司 一种3-甲氨基-1-(2-噻吩基)-1-丙酮盐酸盐的合成方法
CN114790146B (zh) * 2022-05-19 2024-03-29 河南省科学院高新技术研究中心 一种3-(甲基氨基)-1-芳香基丙酮的制备方法

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3859305A (en) * 1970-03-10 1975-01-07 Degussa Indole aminoketones
DE2017468A1 (en) * 1970-04-11 1971-11-04 Deutsche Gold- U. Silber-Scheideanstalt, Vorm. Roessler, 6000 Frankfurt Phenylalkylaminoalkyl-pyrazoles antiphlogistic
DE2063901A1 (en) * 1970-12-28 1972-07-20 Deutsche Gold- Und Silber-Scheideanstalt Vormals Roessler, 6000 Frankfurt Phenylalkylaminoalkylthiazoles - as antiphlogistics
DE2353873A1 (de) * 1973-10-26 1975-05-07 Inst Toxikologii Beta-ketoderivate der linearen und cyclischen beta-phenylaethylamine, deren salze und verfahren zu deren herstellung
DD122967A1 (de) * 1975-07-10 1976-11-12 Lothar Luecke Hylamin-derivate
US4948813A (en) * 1987-11-30 1990-08-14 E. I. Du Pont De Nemours And Company Benzylketone phospholipase A2 inhibitors
US5075339A (en) * 1989-07-28 1991-12-24 Du Pont Merck Pharmaceutical Company Benzylketone phospholipase A2 inhibitors
JPH0625178B2 (ja) * 1989-08-04 1994-04-06 三井東圧化学株式会社 アミノケトン誘導体及びその用途
JPH05503517A (ja) 1989-12-18 1993-06-10 バージニア・コモンウェルス・ユニバーシティ シグマレセプターリガンド及びその用途
JPH0570412A (ja) * 1991-09-13 1993-03-23 Fuji Yakuhin Kogyo Kk 光学活性なβ−アミノアルコールの製造方法
EP0571685A1 (en) * 1992-05-27 1993-12-01 Novo Nordisk A/S Aryloxyheteroarylpropylamines, their preparation and use
ATE224366T1 (de) 1997-10-31 2002-10-15 Hoffmann La Roche D-prolinderivate
JP2000264867A (ja) * 1999-03-18 2000-09-26 Nippon Shokubai Co Ltd 有機アミド化合物およびその製造法
NO992278L (no) * 1999-05-11 2000-11-13 Rf Procom As FremgangsmÕte for forhindring av tilstopping rørledninger med gasshydrater
BR0116721A (pt) * 2001-01-04 2003-12-23 Ferrer Int Processo para a preparação de (±)-trans-4-p-fluorofenil-3-hidroximetil-1-metilpiperi dina
US20050256318A1 (en) 2002-07-09 2005-11-17 Dominique Michel Process for the preparation of n-monosubstituted beta-amino alcohols
WO2004005239A1 (en) * 2002-07-09 2004-01-15 Lonza Ag PROCESS FOR THE PREPARATION OF N-MONOSUBSTITUTED β-AMINO ALCOHOLS

Also Published As

Publication number Publication date
DE10240026A1 (de) 2004-03-11
PL373599A1 (en) 2005-09-05
AU2003260348A1 (en) 2004-03-19
KR101017885B1 (ko) 2011-03-04
US7579484B2 (en) 2009-08-25
HK1081532A1 (en) 2006-05-19
CA2497028A1 (en) 2004-03-11
EP1532101A1 (de) 2005-05-25
JP2005536557A (ja) 2005-12-02
WO2004020391A1 (de) 2004-03-11
RU2340595C2 (ru) 2008-12-10
JP4593275B2 (ja) 2010-12-08
RU2005108974A (ru) 2005-10-27
MXPA05002117A (es) 2005-05-23
ZA200502457B (en) 2005-10-25
US20060122405A1 (en) 2006-06-08
AU2003260348B2 (en) 2009-09-03
KR20050059104A (ko) 2005-06-17
CN100368384C (zh) 2008-02-13
CN1678564A (zh) 2005-10-05

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Legal Events

Date Code Title Description
B06G Technical and formal requirements: other requirements [chapter 6.7 patent gazette]

Free format text: BASEADO NO ART. 216 1 DA LPI, APRESENTE COPIA AUTENTICADA DA PROCURACAO PARA QUE ESTA SEJA ACEITA.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2160 DE 29/05/2012.