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YU57900A - Sinteza karbamatno ketolidnih antibiotika - Google Patents

Sinteza karbamatno ketolidnih antibiotika

Info

Publication number
YU57900A
YU57900A YU57900A YUP57900A YU57900A YU 57900 A YU57900 A YU 57900A YU 57900 A YU57900 A YU 57900A YU P57900 A YUP57900 A YU P57900A YU 57900 A YU57900 A YU 57900A
Authority
YU
Yugoslavia
Prior art keywords
synthesis
antibiotics
ketolide antibiotics
carbamate ketolide
carbamate
Prior art date
Application number
YU57900A
Other languages
English (en)
Inventor
Kaneko Takushi
Wiliam Robert McLaughlin
Wiliam Thomas Mcmilan
David Harold Ripin
Brian Clement Vanderplas
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of YU57900A publication Critical patent/YU57900A/sh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Pronalazak se odnosi na postupak za proizvodnju makrolidnog antinibotika formule: u kojoj R1, R2, R3, R4, R5 su kako je definisano ranije. Ovi antibiotici su korisna antibakterijska i antiprotozojska sredstva kod sisara, uključujući čoveka, kao i kod riba i ptica. Pronalazak takodje obuhvata nova jedinjenja, proizvedenih prilikom pripreme makrolidnog antibiotika.[Invention refers to the procedure for the production of macrolide antibiotic of formula: wherein R1, R2, R3, R4, R5 are as previously defined. These antibiotics are useful antibacterical antiprotosoic means with mammals including men, such as fish and birds. The invention also includes new compounds, produced during the preparation of macrolide antibiotics.
YU57900A 1999-09-29 2000-09-22 Sinteza karbamatno ketolidnih antibiotika YU57900A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15655499P 1999-09-29 1999-09-29

Publications (1)

Publication Number Publication Date
YU57900A true YU57900A (sh) 2003-02-28

Family

ID=22560054

Family Applications (1)

Application Number Title Priority Date Filing Date
YU57900A YU57900A (sh) 1999-09-29 2000-09-22 Sinteza karbamatno ketolidnih antibiotika

Country Status (18)

Country Link
EP (1) EP1088828A3 (sh)
JP (1) JP2001151792A (sh)
KR (1) KR20010050704A (sh)
CN (1) CN1289778A (sh)
AR (1) AR023273A1 (sh)
AU (1) AU6129300A (sh)
BR (1) BR0004537A (sh)
CA (1) CA2321336C (sh)
CZ (1) CZ20003567A3 (sh)
HU (1) HUP0003834A3 (sh)
ID (1) ID27331A (sh)
IL (1) IL138633A0 (sh)
IN (2) IN187119B (sh)
PL (1) PL342917A1 (sh)
RU (1) RU2188827C2 (sh)
TR (1) TR200002787A2 (sh)
YU (1) YU57900A (sh)
ZA (1) ZA200005139B (sh)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050171342A1 (en) 2002-02-15 2005-08-04 Michael Burnet Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
WO2003070173A2 (en) 2002-02-15 2003-08-28 Sympore Gmbh Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
AU2003211113B2 (en) 2002-02-15 2007-08-09 Merckle Gmbh Antibiotic conjugates
CN102199180B (zh) * 2011-04-12 2014-07-09 连云港杰瑞药业有限公司 一种卡培他滨的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2727969B1 (fr) * 1994-12-09 1997-01-17 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
ID24529A (id) * 1997-06-11 2000-07-20 Pfizer Prod Inc Turunan-turunan 9-oksima eritromisin
HN1998000159A (es) * 1997-10-29 1999-02-09 Monsanto Co Derivados de 9- amino - 3 ceto eritromicina
AP1060A (en) * 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.

Also Published As

Publication number Publication date
AR023273A1 (es) 2002-09-04
IN188930B (sh) 2002-11-23
PL342917A1 (en) 2001-04-09
HU0003834D0 (en) 2000-09-28
RU2188827C2 (ru) 2002-09-10
IN187119B (sh) 2002-02-09
EP1088828A2 (en) 2001-04-04
HUP0003834A3 (en) 2001-07-30
JP2001151792A (ja) 2001-06-05
ZA200005139B (en) 2002-03-26
HUP0003834A2 (hu) 2001-05-28
AU6129300A (en) 2001-04-05
KR20010050704A (ko) 2001-06-15
BR0004537A (pt) 2001-04-17
TR200002787A2 (tr) 2001-04-20
IL138633A0 (en) 2001-10-31
CN1289778A (zh) 2001-04-04
CZ20003567A3 (cs) 2002-01-16
EP1088828A3 (en) 2001-04-11
CA2321336A1 (en) 2001-03-29
ID27331A (id) 2001-03-29
CA2321336C (en) 2005-03-15

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