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WO2003080614A3 - Triazolopyrimidine als fungizide - Google Patents

Triazolopyrimidine als fungizide Download PDF

Info

Publication number
WO2003080614A3
WO2003080614A3 PCT/EP2003/002413 EP0302413W WO03080614A3 WO 2003080614 A3 WO2003080614 A3 WO 2003080614A3 EP 0302413 W EP0302413 W EP 0302413W WO 03080614 A3 WO03080614 A3 WO 03080614A3
Authority
WO
WIPO (PCT)
Prior art keywords
optionally substituted
cycloalkyl
novel
relates
dialkylamino
Prior art date
Application number
PCT/EP2003/002413
Other languages
English (en)
French (fr)
Other versions
WO2003080614A2 (de
Inventor
Christiane Boie
Ralf Dunkel
Hans-Ludwig Elbe
Herbert Gayer
Olaf Gebauer
Bernd-Wieland Krueger
Ulrich Heinemann
Arnd Voerste
Oliver Guth
Ronald Ebbert
Ulrike Wachendorff-Neumann
Astrid Mauler-Machnik
Original Assignee
Bayer Cropscience Ag
Christiane Boie
Ralf Dunkel
Hans-Ludwig Elbe
Herbert Gayer
Olaf Gebauer
Bernd-Wieland Krueger
Ulrich Heinemann
Arnd Voerste
Oliver Guth
Ronald Ebbert
Ulrike Wachendorff-Neumann
Astrid Mauler-Machnik
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag, Christiane Boie, Ralf Dunkel, Hans-Ludwig Elbe, Herbert Gayer, Olaf Gebauer, Bernd-Wieland Krueger, Ulrich Heinemann, Arnd Voerste, Oliver Guth, Ronald Ebbert, Ulrike Wachendorff-Neumann, Astrid Mauler-Machnik filed Critical Bayer Cropscience Ag
Priority to AU2003212322A priority Critical patent/AU2003212322A1/en
Priority to JP2003578368A priority patent/JP2005528364A/ja
Priority to EP03708201A priority patent/EP1490370A2/de
Priority to US10/508,402 priority patent/US20050222173A1/en
Publication of WO2003080614A2 publication Critical patent/WO2003080614A2/de
Publication of WO2003080614A3 publication Critical patent/WO2003080614A3/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Neue Triazolopyrimidine der Formel (I),in welcherR1 für Amino, für jeweils gegebenenfalls substituiertes Alkyl, Alkenyl, Alkinyl, Cycloalkyl, Alkoxy, Alkenyloxy, Alkinyloxy, Cycloalkyloxy, Alkylamino, Dialkylamino, Alkenylamino, Alkinylamino, Cycloalkylamino, N-Cycloalkyl-N-Alkylamino, Alkylidenamino oder Heterocyclyl steht,R2 für Wasserstoff oder für jeweils gegebenenfalls substituiertes Alkyl, Alkenyl, Alkinyl oder Cycloalkyl steht, oderR1 und R2 gemeinsam mit dem Stickstoffatom, an das sie gebunden sind, einen gegebenenfalls substituierten heterocyclischen Ring bilden,R3 für gegebenenfalls einfach bis vierfach substituiertes Aryl steht,R4 für Halogen, Cyano oder für jeweils gegebenenfalls substituiertes Alkoxy oder Dialkylamino steht undX für Halogen steht, ein Verfahren zur Herstellung dieser neuen Stoffe und deren Verwendung zur Bekämpfung von unerwünschten Mikroorganismen.Neue Zwischenprodukte der Formeln (II), (IV) und (VIa), sowie Verfahren zu deren Herstellung.
PCT/EP2003/002413 2002-03-22 2003-03-10 Triazolopyrimidine als fungizide WO2003080614A2 (de)

Priority Applications (4)

Application Number Priority Date Filing Date Title
AU2003212322A AU2003212322A1 (en) 2002-03-22 2003-03-10 Triazolopyrimidines used as fungicides
JP2003578368A JP2005528364A (ja) 2002-03-22 2003-03-10 トリアゾロピリミジン類
EP03708201A EP1490370A2 (de) 2002-03-22 2003-03-10 Triazolopyrimidine
US10/508,402 US20050222173A1 (en) 2002-03-22 2003-03-10 Triazolopyrimidines

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10212886.3 2002-03-22
DE10212886A DE10212886A1 (de) 2002-03-22 2002-03-22 Triazolopyrimidine

Publications (2)

Publication Number Publication Date
WO2003080614A2 WO2003080614A2 (de) 2003-10-02
WO2003080614A3 true WO2003080614A3 (de) 2004-01-08

Family

ID=27798089

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2003/002413 WO2003080614A2 (de) 2002-03-22 2003-03-10 Triazolopyrimidine als fungizide

Country Status (7)

Country Link
US (1) US20050222173A1 (de)
EP (1) EP1490370A2 (de)
JP (1) JP2005528364A (de)
AU (1) AU2003212322A1 (de)
DE (1) DE10212886A1 (de)
PL (1) PL372462A1 (de)
WO (1) WO2003080614A2 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200533670A (en) * 2003-12-19 2005-10-16 Basf Ag 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
UY28986A1 (es) * 2004-06-25 2006-01-31 Basf Ag Compuestos de triazolopirimidina y su uso en el control de hongos daninos
EP2131658A2 (de) * 2007-01-30 2009-12-16 Basf Se Verfahren für verbessertes pflanzenwachstum
WO2012007416A1 (en) 2010-07-13 2012-01-19 Bayer Pharma Aktiengesellschaft Bicyclic pyrimidines
CN114634455B (zh) * 2020-12-15 2023-10-24 苏州华先医药科技有限公司 一种合成5-溴-1h-3-氨基-1,2,4-三氮唑的方法

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0550113A2 (de) * 1991-12-30 1993-07-07 Shell Internationale Researchmaatschappij B.V. Triazolopyrimidinderivate mit fungizider Aktivität
EP0834513A2 (de) * 1996-10-07 1998-04-08 American Cyanamid Company Pentafluorophenylazolopyrimidine
WO1998046608A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluoromethylalkylamino-triazolopyrimidines
WO1998046607A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
WO2002002536A1 (en) * 2000-07-06 2002-01-10 Bayer Cropscience K.K. Novel tetrazole derivatives
WO2002088126A1 (de) * 2001-04-30 2002-11-07 Bayer Cropscience Ag Triazolopyrimidine
WO2002088127A2 (de) * 2001-04-27 2002-11-07 Bayer Cropscience Ag Triazolopyrimidine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL108747A (en) * 1993-03-04 1999-03-12 Shell Int Research Mushroom-killing preparations containing a history of 6 metamorphoses of 5 - 7 Dihalo - 1, 2 - 4 Triazlo [A-1,5] Pyrimidine Certain such new compounds and their preparation
TW258648B (de) * 1993-03-04 1995-10-01 Shell Internat Res Schappej Bv
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0550113A2 (de) * 1991-12-30 1993-07-07 Shell Internationale Researchmaatschappij B.V. Triazolopyrimidinderivate mit fungizider Aktivität
EP0834513A2 (de) * 1996-10-07 1998-04-08 American Cyanamid Company Pentafluorophenylazolopyrimidine
WO1998046608A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluoromethylalkylamino-triazolopyrimidines
WO1998046607A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
WO2002002536A1 (en) * 2000-07-06 2002-01-10 Bayer Cropscience K.K. Novel tetrazole derivatives
WO2002088127A2 (de) * 2001-04-27 2002-11-07 Bayer Cropscience Ag Triazolopyrimidine
WO2002088126A1 (de) * 2001-04-30 2002-11-07 Bayer Cropscience Ag Triazolopyrimidine

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
KOFMAN ET AL., RUSS. J. ORG. CHEM., vol. 29, no. 11, 1993, pages 1942 - 1943, XP009012611 *

Also Published As

Publication number Publication date
EP1490370A2 (de) 2004-12-29
WO2003080614A2 (de) 2003-10-02
AU2003212322A8 (en) 2003-10-08
PL372462A1 (en) 2005-07-25
US20050222173A1 (en) 2005-10-06
AU2003212322A1 (en) 2003-10-08
DE10212886A1 (de) 2003-10-02
JP2005528364A (ja) 2005-09-22

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