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UY34220A - Indazoles, composiciones farmacéuticas y uso de los mismos - Google Patents

Indazoles, composiciones farmacéuticas y uso de los mismos

Info

Publication number
UY34220A
UY34220A UY0001034220A UY34220A UY34220A UY 34220 A UY34220 A UY 34220A UY 0001034220 A UY0001034220 A UY 0001034220A UY 34220 A UY34220 A UY 34220A UY 34220 A UY34220 A UY 34220A
Authority
UY
Uruguay
Prior art keywords
indazols
same
pharmaceutical compositions
página
sgdd
Prior art date
Application number
UY0001034220A
Other languages
English (en)
Inventor
Florian Michel Wakenhut
Jotham Wadsworth Coe
Christoph Martin Dehnhardt
Jones Peter
Steven Wade Kortum
Yogesh Anil Sabnis
Gavin Alistair Whitlock
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46826868&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY34220(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of UY34220A publication Critical patent/UY34220A/es

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Toxicology (AREA)
  • Obesity (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)

Abstract

La presente invención se refiere a los compuestos de fórmula I, a sales farmacéuticamente aceptables y a un solvatos farmacéuticamente aceptables de dichos compuestos y sales, donde los sustituyentes se definen en la presente; a composiciones que contienen tales compuestos; y a los usos de tales compuestos en el tratamiento de varias enfermedades, en particular asma y COPD.
UY0001034220A 2011-07-27 2012-07-26 Indazoles, composiciones farmacéuticas y uso de los mismos UY34220A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161512144P 2011-07-27 2011-07-27

Publications (1)

Publication Number Publication Date
UY34220A true UY34220A (es) 2013-02-28

Family

ID=46826868

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034220A UY34220A (es) 2011-07-27 2012-07-26 Indazoles, composiciones farmacéuticas y uso de los mismos

Country Status (30)

Country Link
US (2) US8575336B2 (es)
EP (1) EP2736907B1 (es)
JP (1) JP5579351B1 (es)
KR (1) KR20140026627A (es)
CN (1) CN103717599B (es)
AP (1) AP2014007372A0 (es)
AR (1) AR087348A1 (es)
AU (1) AU2012288491A1 (es)
BR (1) BR112014001801A2 (es)
CA (1) CA2841882A1 (es)
CL (1) CL2014000122A1 (es)
CO (1) CO6862160A2 (es)
CR (1) CR20140042A (es)
CU (1) CU20140009A7 (es)
DO (1) DOP2014000016A (es)
EA (1) EA201490357A1 (es)
EC (1) ECSP14013222A (es)
GT (1) GT201400016A (es)
IL (1) IL230662A0 (es)
MA (1) MA35285B1 (es)
MD (1) MD20140002A2 (es)
MX (1) MX2014001004A (es)
NI (1) NI201400005A (es)
PE (1) PE20141059A1 (es)
PH (1) PH12014500199A1 (es)
TN (1) TN2014000033A1 (es)
TW (1) TWI462922B (es)
UA (1) UA108442C2 (es)
UY (1) UY34220A (es)
WO (1) WO2013014567A1 (es)

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US8575336B2 (en) 2011-07-27 2013-11-05 Pfizer Limited Indazoles
EA201650029A1 (ru) * 2014-05-14 2017-09-29 Пфайзер Инк. Пиразолопиридины и пиразолопиримидины
WO2016139212A1 (en) 2015-03-04 2016-09-09 F. Hoffmann-La Roche Ag Triazolopyridine compounds and methods of use thereof
DK3286181T3 (da) 2015-04-22 2021-04-06 Rigel Pharmaceuticals Inc Pyrazolforbindelser og fremgangsmåde til fremstilling og anvendelse af forbindelserne
US10100049B2 (en) 2015-11-03 2018-10-16 Theravance Biopharma R&D Ip, Llc JAK kinase inhibitor compounds for treatment of respiratory disease
DK3371185T3 (da) 2015-11-03 2020-11-30 Topivert Pharma Ltd 4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridin og 1,4,5,6,7,8-hexahydroimidazo[4,5-d]azepinderivater som janus-kinase-inhibitorer
PL3712152T3 (pl) 2015-11-03 2021-08-02 Topivert Pharma Limited Pochodne 4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pirydyny i 1,4,5,6,7,8-heksahydroimidazo[4,5-d]azepiny jako inhibitory kinaz janusowych
TW201720828A (zh) 2015-11-23 2017-06-16 赫孚孟拉羅股份公司 治療性化合物及組合物以及其使用方法
US20170157215A1 (en) 2015-12-04 2017-06-08 Jomoco, Corp. Compositions and methods to mitigate or prevent an immune response to an immunogenic therapeutic molecule in non-human primates
WO2017140825A1 (en) 2016-02-18 2017-08-24 F. Hoffmann-La Roche Ag Therapeutic compounds, compositions and methods of use thereof
WO2017191098A1 (en) 2016-05-05 2017-11-09 F. Hoffmann-La Roche Ag Pyrazole derivatives, compositions and therapeutic use thereof
DK3464266T3 (da) * 2016-06-01 2021-11-22 Bayer Animal Health Gmbh Substituerede indazoler, der er anvendelige til behandling og forebyggelse af allergiske og/eller inflammatoriske sygdomme hos dyr
CN109890817B (zh) 2016-09-06 2022-06-17 豪夫迈·罗氏有限公司 8-(氮杂环丁烷-1-基)-[1,2,4]三唑并[1,5-a]吡啶基化合物、其组合物和应用方法
MX2019007339A (es) 2016-12-29 2019-09-06 Hoffmann La Roche Compuestos de pirazolopirimidina y metodos de uso de los mismos.
BR112019018649A2 (pt) * 2017-03-09 2020-04-07 Theravance Biopharma R&D Ip Llc inibidores jak derivados da fusão de imidazopiperidina
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