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UY32247A - Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicaciones - Google Patents

Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicaciones

Info

Publication number
UY32247A
UY32247A UY0001032247A UY32247A UY32247A UY 32247 A UY32247 A UY 32247A UY 0001032247 A UY0001032247 A UY 0001032247A UY 32247 A UY32247 A UY 32247A UY 32247 A UY32247 A UY 32247A
Authority
UY
Uruguay
Prior art keywords
compounds
aminociclohexilo
applications
new
same
Prior art date
Application number
UY0001032247A
Other languages
English (en)
Inventor
Cronin Mark
Geng Bolin
Reck Folkert
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY32247A publication Critical patent/UY32247A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53831,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

La presente invención se refiere a compuestos de Fórmula (I): y sales farmacéuticamente aceptables de los mismos, a su uso en el tratamiento de infecciones bacterianas y a sus métodos de preparación.
UY0001032247A 2008-11-14 2009-11-13 Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicaciones UY32247A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11470608P 2008-11-14 2008-11-14
US16384809P 2009-03-26 2009-03-26

Publications (1)

Publication Number Publication Date
UY32247A true UY32247A (es) 2010-06-30

Family

ID=41463108

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032247A UY32247A (es) 2008-11-14 2009-11-13 Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicaciones

Country Status (20)

Country Link
US (1) US20110288084A1 (es)
EP (1) EP2370444A1 (es)
JP (1) JP2012508789A (es)
KR (1) KR20110093797A (es)
CN (1) CN102216308A (es)
AR (1) AR074340A1 (es)
AU (1) AU2009315425A1 (es)
BR (1) BRPI0921148A2 (es)
CA (1) CA2742520A1 (es)
CO (1) CO6382113A2 (es)
CR (1) CR20110256A (es)
CU (1) CU20110108A7 (es)
EA (1) EA201100754A1 (es)
EC (1) ECSP11011053A (es)
IL (1) IL211941A0 (es)
MX (1) MX2011005106A (es)
TW (1) TW201022279A (es)
UY (1) UY32247A (es)
WO (1) WO2010055348A1 (es)
ZA (1) ZA201104395B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2840060A1 (en) * 2011-06-27 2013-01-03 Kyorin Pharmaceutical Co., Ltd. Bridged bicyclic compounds for the treatment of bacterial infections
AR096135A1 (es) * 2013-05-02 2015-12-09 Actelion Pharmaceuticals Ltd Derivados de la quinolona
UY36851A (es) 2015-08-16 2017-03-31 Glaxosmithkline Ip Dev Ltd Compuestos para uso en aplicaciones antibacterianas
TW201711999A (zh) 2015-09-03 2017-04-01 佛瑪治療公司 ﹝6,6﹞稠合雙環組蛋白脫乙醯基酶8(hdac8)抑制劑
SMT202000335T1 (it) * 2016-06-08 2020-07-08 Acraf Nuovi composti antibatterici
US10912780B2 (en) 2017-06-08 2021-02-09 Bugworks Research, Inc. Heterocyclic compounds useful as anti-bacterial agents and method for production thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY150958A (en) * 2005-06-16 2014-03-31 Astrazeneca Ab Compounds for the treatment of multi-drug resistant bacterial infections
NZ573032A (en) * 2006-05-26 2010-12-24 Taisho Pharmaceutical Co Ltd Antimicrobial heretocyclic compound and intermediates for its production
CL2007003693A1 (es) * 2006-12-22 2008-06-27 Actelion Pharmaceuticals Ltd Compuestos derivados de pirido [3,2-b] [1,4] tiazina; composicion farmaceutica que contiene dichos compuestos; y su uso en el tratamiento de infecciones bacterianas.

Also Published As

Publication number Publication date
CR20110256A (es) 2011-07-04
US20110288084A1 (en) 2011-11-24
ECSP11011053A (es) 2011-06-30
CU20110108A7 (es) 2012-01-31
BRPI0921148A2 (pt) 2016-02-23
CO6382113A2 (es) 2012-02-15
JP2012508789A (ja) 2012-04-12
CN102216308A (zh) 2011-10-12
WO2010055348A1 (en) 2010-05-20
ZA201104395B (en) 2012-03-28
EP2370444A1 (en) 2011-10-05
TW201022279A (en) 2010-06-16
AR074340A1 (es) 2011-01-12
CA2742520A1 (en) 2010-05-20
EA201100754A1 (ru) 2012-01-30
IL211941A0 (en) 2011-06-30
AU2009315425A1 (en) 2010-05-20
MX2011005106A (es) 2011-05-30
KR20110093797A (ko) 2011-08-18

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20181127