UY32247A - Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicaciones - Google Patents
Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicacionesInfo
- Publication number
- UY32247A UY32247A UY0001032247A UY32247A UY32247A UY 32247 A UY32247 A UY 32247A UY 0001032247 A UY0001032247 A UY 0001032247A UY 32247 A UY32247 A UY 32247A UY 32247 A UY32247 A UY 32247A
- Authority
- UY
- Uruguay
- Prior art keywords
- compounds
- aminociclohexilo
- applications
- new
- same
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Peptides Or Proteins (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
La presente invención se refiere a compuestos de Fórmula (I): y sales farmacéuticamente aceptables de los mismos, a su uso en el tratamiento de infecciones bacterianas y a sus métodos de preparación.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11470608P | 2008-11-14 | 2008-11-14 | |
US16384809P | 2009-03-26 | 2009-03-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY32247A true UY32247A (es) | 2010-06-30 |
Family
ID=41463108
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001032247A UY32247A (es) | 2008-11-14 | 2009-11-13 | Nuevos compuestos de aminociclohexilo, composiciones farmacéuticas de los mismos y aplicaciones |
Country Status (20)
Country | Link |
---|---|
US (1) | US20110288084A1 (es) |
EP (1) | EP2370444A1 (es) |
JP (1) | JP2012508789A (es) |
KR (1) | KR20110093797A (es) |
CN (1) | CN102216308A (es) |
AR (1) | AR074340A1 (es) |
AU (1) | AU2009315425A1 (es) |
BR (1) | BRPI0921148A2 (es) |
CA (1) | CA2742520A1 (es) |
CO (1) | CO6382113A2 (es) |
CR (1) | CR20110256A (es) |
CU (1) | CU20110108A7 (es) |
EA (1) | EA201100754A1 (es) |
EC (1) | ECSP11011053A (es) |
IL (1) | IL211941A0 (es) |
MX (1) | MX2011005106A (es) |
TW (1) | TW201022279A (es) |
UY (1) | UY32247A (es) |
WO (1) | WO2010055348A1 (es) |
ZA (1) | ZA201104395B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2840060A1 (en) * | 2011-06-27 | 2013-01-03 | Kyorin Pharmaceutical Co., Ltd. | Bridged bicyclic compounds for the treatment of bacterial infections |
AR096135A1 (es) * | 2013-05-02 | 2015-12-09 | Actelion Pharmaceuticals Ltd | Derivados de la quinolona |
UY36851A (es) | 2015-08-16 | 2017-03-31 | Glaxosmithkline Ip Dev Ltd | Compuestos para uso en aplicaciones antibacterianas |
TW201711999A (zh) | 2015-09-03 | 2017-04-01 | 佛瑪治療公司 | ﹝6,6﹞稠合雙環組蛋白脫乙醯基酶8(hdac8)抑制劑 |
SMT202000335T1 (it) * | 2016-06-08 | 2020-07-08 | Acraf | Nuovi composti antibatterici |
US10912780B2 (en) | 2017-06-08 | 2021-02-09 | Bugworks Research, Inc. | Heterocyclic compounds useful as anti-bacterial agents and method for production thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY150958A (en) * | 2005-06-16 | 2014-03-31 | Astrazeneca Ab | Compounds for the treatment of multi-drug resistant bacterial infections |
NZ573032A (en) * | 2006-05-26 | 2010-12-24 | Taisho Pharmaceutical Co Ltd | Antimicrobial heretocyclic compound and intermediates for its production |
CL2007003693A1 (es) * | 2006-12-22 | 2008-06-27 | Actelion Pharmaceuticals Ltd | Compuestos derivados de pirido [3,2-b] [1,4] tiazina; composicion farmaceutica que contiene dichos compuestos; y su uso en el tratamiento de infecciones bacterianas. |
-
2009
- 2009-11-12 TW TW098138483A patent/TW201022279A/zh unknown
- 2009-11-13 EA EA201100754A patent/EA201100754A1/ru unknown
- 2009-11-13 CA CA2742520A patent/CA2742520A1/en not_active Abandoned
- 2009-11-13 EP EP09753199A patent/EP2370444A1/en not_active Withdrawn
- 2009-11-13 US US13/128,596 patent/US20110288084A1/en not_active Abandoned
- 2009-11-13 CN CN2009801457755A patent/CN102216308A/zh active Pending
- 2009-11-13 WO PCT/GB2009/051532 patent/WO2010055348A1/en active Application Filing
- 2009-11-13 UY UY0001032247A patent/UY32247A/es not_active Application Discontinuation
- 2009-11-13 JP JP2011543815A patent/JP2012508789A/ja active Pending
- 2009-11-13 KR KR1020117010967A patent/KR20110093797A/ko not_active Application Discontinuation
- 2009-11-13 AU AU2009315425A patent/AU2009315425A1/en not_active Abandoned
- 2009-11-13 MX MX2011005106A patent/MX2011005106A/es not_active Application Discontinuation
- 2009-11-13 BR BRPI0921148A patent/BRPI0921148A2/pt not_active Application Discontinuation
- 2009-11-13 AR ARP090104378A patent/AR074340A1/es unknown
-
2011
- 2011-03-24 IL IL211941A patent/IL211941A0/en unknown
- 2011-05-11 CO CO11058050A patent/CO6382113A2/es not_active Application Discontinuation
- 2011-05-13 EC EC2011011053A patent/ECSP11011053A/es unknown
- 2011-05-13 CU CU20110108A patent/CU20110108A7/es unknown
- 2011-05-13 CR CR20110256A patent/CR20110256A/es not_active Application Discontinuation
- 2011-06-13 ZA ZA2011/04395A patent/ZA201104395B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CR20110256A (es) | 2011-07-04 |
US20110288084A1 (en) | 2011-11-24 |
ECSP11011053A (es) | 2011-06-30 |
CU20110108A7 (es) | 2012-01-31 |
BRPI0921148A2 (pt) | 2016-02-23 |
CO6382113A2 (es) | 2012-02-15 |
JP2012508789A (ja) | 2012-04-12 |
CN102216308A (zh) | 2011-10-12 |
WO2010055348A1 (en) | 2010-05-20 |
ZA201104395B (en) | 2012-03-28 |
EP2370444A1 (en) | 2011-10-05 |
TW201022279A (en) | 2010-06-16 |
AR074340A1 (es) | 2011-01-12 |
CA2742520A1 (en) | 2010-05-20 |
EA201100754A1 (ru) | 2012-01-30 |
IL211941A0 (en) | 2011-06-30 |
AU2009315425A1 (en) | 2010-05-20 |
MX2011005106A (es) | 2011-05-30 |
KR20110093797A (ko) | 2011-08-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20181127 |