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UY30843A1 - Derivados de isoquinolona sustituidos con ciloalquilamina - Google Patents

Derivados de isoquinolona sustituidos con ciloalquilamina

Info

Publication number
UY30843A1
UY30843A1 UY30843A UY30843A UY30843A1 UY 30843 A1 UY30843 A1 UY 30843A1 UY 30843 A UY30843 A UY 30843A UY 30843 A UY30843 A UY 30843A UY 30843 A1 UY30843 A1 UY 30843A1
Authority
UY
Uruguay
Prior art keywords
ciloalquilamina
isoquinolone derivatives
derivatives replaced
isoquinolone
replaced
Prior art date
Application number
UY30843A
Other languages
English (en)
Inventor
Dr Katrin Lorenz
Dr John Weston
Dr Matthias Lohn
Dr Armin Hofmeister
Dr Joachim Brendel
Dr Oliver Plettenburg
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38565513&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY30843(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY30843A1 publication Critical patent/UY30843A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Pregnancy & Childbirth (AREA)
  • Epidemiology (AREA)

Abstract

La invencion se refiere a derivados de isoquinolona sustituidos en la posicion 6, de formula (I) utiles para el tratamiento y/o prevencion de enfermedades asociadas con la Rhoquinasa y/o la fosforilacion mediada por la Rho-quinasa de la fosfatasa de la cadena ligera de miosina, y a composiciones que contienen tales compuestos
UY30843A 2006-12-27 2007-12-26 Derivados de isoquinolona sustituidos con ciloalquilamina UY30843A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06026899 2006-12-27

Publications (1)

Publication Number Publication Date
UY30843A1 true UY30843A1 (es) 2008-07-31

Family

ID=38565513

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30843A UY30843A1 (es) 2006-12-27 2007-12-26 Derivados de isoquinolona sustituidos con ciloalquilamina

Country Status (31)

Country Link
US (1) US8742116B2 (es)
EP (1) EP2125745B1 (es)
JP (1) JP5405314B2 (es)
KR (1) KR101474228B1 (es)
CN (1) CN101595094B (es)
AR (1) AR064492A1 (es)
AU (1) AU2007338407B2 (es)
BR (1) BRPI0722064A2 (es)
CA (1) CA2673917C (es)
CL (1) CL2007003821A1 (es)
CO (1) CO6210726A2 (es)
CR (1) CR10813A (es)
DO (1) DOP2009000164A (es)
EC (1) ECSP099467A (es)
ES (1) ES2625266T3 (es)
GT (1) GT200900179A (es)
HK (1) HK1139390A1 (es)
IL (1) IL199540A (es)
MA (1) MA31075B1 (es)
MX (1) MX2009005966A (es)
MY (1) MY155009A (es)
NI (1) NI200900108A (es)
NO (1) NO20092422L (es)
NZ (1) NZ577980A (es)
RU (1) RU2457203C2 (es)
SV (1) SV2009003318A (es)
TN (1) TN2009000269A1 (es)
TW (1) TWI434689B (es)
UY (1) UY30843A1 (es)
WO (1) WO2008077551A1 (es)
ZA (1) ZA200903551B (es)

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