UY29624A1 - NON-STEROID PROGESTERONE RECEPTOR MODULATORS - Google Patents
NON-STEROID PROGESTERONE RECEPTOR MODULATORSInfo
- Publication number
- UY29624A1 UY29624A1 UY29624A UY29624A UY29624A1 UY 29624 A1 UY29624 A1 UY 29624A1 UY 29624 A UY29624 A UY 29624A UY 29624 A UY29624 A UY 29624A UY 29624 A1 UY29624 A1 UY 29624A1
- Authority
- UY
- Uruguay
- Prior art keywords
- receptor modulators
- progesterone receptor
- prevention
- compounds
- steroid progesterone
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/02—1,2-Oxazines; Hydrogenated 1,2-oxazines
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Pregnancy & Childbirth (AREA)
- Gynecology & Obstetrics (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se refiere a moduladores no esteroides de receptor de progesterona de la fórmula general, a su uso para la preparación de medicamentos y a las composiciones farmacéuticas que contienen estos compuestos. Los compuestos de la invención son apropiados para la terapia y la prevención de enfermedades ginecológicas, como endometriosos, leiomiomas del útero, sangrados disfuncionales y dismenorrea y para el tratamiento y la prevención de tumores hormona-dependientes y para el control de la fertilidad femenina, así como para la terapia de sustitución hormonal.The present invention relates to non-steroidal progesterone receptor modulators of the general formula, their use for the preparation of medicaments and the pharmaceutical compositions containing these compounds. The compounds of the invention are suitable for the therapy and prevention of gynecological diseases, such as endometrious, uterine leiomyomas, dysfunctional bleeding and dysmenorrhea and for the treatment and prevention of hormone-dependent tumors and for the control of female fertility, as well. As for hormone replacement therapy.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005030292A DE102005030292A1 (en) | 2005-06-24 | 2005-06-24 | Nonsteroidal progesterone receptor modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY29624A1 true UY29624A1 (en) | 2007-01-31 |
Family
ID=37199176
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY29624A UY29624A1 (en) | 2005-06-24 | 2006-06-26 | NON-STEROID PROGESTERONE RECEPTOR MODULATORS |
Country Status (22)
| Country | Link |
|---|---|
| EP (1) | EP1902049A2 (en) |
| JP (1) | JP2008543910A (en) |
| KR (1) | KR20080030622A (en) |
| CN (1) | CN101248066A (en) |
| AR (1) | AR054519A1 (en) |
| AU (1) | AU2006261048A1 (en) |
| BR (1) | BRPI0611903A2 (en) |
| CA (1) | CA2611897A1 (en) |
| CR (1) | CR9598A (en) |
| DE (1) | DE102005030292A1 (en) |
| DO (1) | DOP2006000148A (en) |
| EA (1) | EA200702524A1 (en) |
| EC (1) | ECSP078044A (en) |
| GT (1) | GT200600271A (en) |
| IL (1) | IL188021A0 (en) |
| MX (1) | MX2008000072A (en) |
| NO (1) | NO20080440L (en) |
| PE (1) | PE20070125A1 (en) |
| TW (1) | TW200740778A (en) |
| UY (1) | UY29624A1 (en) |
| WO (1) | WO2006136461A2 (en) |
| ZA (1) | ZA200800690B (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UY30805A1 (en) * | 2006-12-21 | 2008-07-31 | Bayer Schering Pharma Ag | NON-STEROID MODULATORS OF PROGESTERONE RECEPTORS |
| DE102007032800A1 (en) * | 2007-07-10 | 2009-01-15 | Bayer Schering Pharma Aktiengesellschaft | Nonsteroidal progesterone receptor modulators |
| DE102007058747A1 (en) | 2007-12-05 | 2009-06-10 | Bayer Schering Pharma Aktiengesellschaft | Nonsteroidal progesterone receptor modulators |
| JP2011519916A (en) * | 2008-07-02 | 2011-07-14 | ファーマコステック カンパニー リミテッド | Method for producing amide derivative |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19856475A1 (en) * | 1998-11-27 | 2000-05-31 | Schering Ag | Nonsteroidal anti-inflammatories |
| EP1344776A1 (en) * | 2002-03-11 | 2003-09-17 | Schering Aktiengesellschaft | 5- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -phtalide and 6- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -4-methyl-2,3-benzoxazin-1-one derivatives with progesterone receptor modulating activity for use in fertility control, hormone replacement therapy and the treatment of gynecological disorders |
| EA200600148A1 (en) * | 2003-07-01 | 2006-08-25 | Шеринг Акциенгезельшафт | HETEROCYCLICALLY SUBSTITUTED DERIVATIVES OF PENTANOL, METHOD OF THEIR RECOVERY AND THEIR APPLICATION AS INFLAMMATION INHIBITORS |
-
2005
- 2005-06-24 DE DE102005030292A patent/DE102005030292A1/en not_active Ceased
-
2006
- 2006-06-22 BR BRPI0611903-4A patent/BRPI0611903A2/en not_active Application Discontinuation
- 2006-06-22 EA EA200702524A patent/EA200702524A1/en unknown
- 2006-06-22 JP JP2008517444A patent/JP2008543910A/en active Pending
- 2006-06-22 EP EP06762404A patent/EP1902049A2/en not_active Withdrawn
- 2006-06-22 WO PCT/EP2006/006531 patent/WO2006136461A2/en active Application Filing
- 2006-06-22 AU AU2006261048A patent/AU2006261048A1/en not_active Abandoned
- 2006-06-22 CA CA002611897A patent/CA2611897A1/en not_active Abandoned
- 2006-06-22 CN CNA2006800308707A patent/CN101248066A/en active Pending
- 2006-06-22 KR KR1020087001793A patent/KR20080030622A/en not_active Application Discontinuation
- 2006-06-22 MX MX2008000072A patent/MX2008000072A/en not_active Application Discontinuation
- 2006-06-23 TW TW095122742A patent/TW200740778A/en unknown
- 2006-06-26 PE PE2006000733A patent/PE20070125A1/en not_active Application Discontinuation
- 2006-06-26 DO DO2006000148A patent/DOP2006000148A/en unknown
- 2006-06-26 UY UY29624A patent/UY29624A1/en not_active Application Discontinuation
- 2006-06-27 AR ARP060102750A patent/AR054519A1/en unknown
- 2006-06-28 GT GT200600271A patent/GT200600271A/en unknown
-
2007
- 2007-12-10 IL IL188021A patent/IL188021A0/en unknown
- 2007-12-17 CR CR9598A patent/CR9598A/en not_active Application Discontinuation
- 2007-12-21 EC EC2007008044A patent/ECSP078044A/en unknown
-
2008
- 2008-01-23 NO NO20080440A patent/NO20080440L/en not_active Application Discontinuation
- 2008-01-23 ZA ZA200800690A patent/ZA200800690B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1902049A2 (en) | 2008-03-26 |
| KR20080030622A (en) | 2008-04-04 |
| BRPI0611903A2 (en) | 2010-10-05 |
| ECSP078044A (en) | 2008-01-23 |
| NO20080440L (en) | 2008-03-25 |
| JP2008543910A (en) | 2008-12-04 |
| AU2006261048A1 (en) | 2006-12-28 |
| CA2611897A1 (en) | 2006-12-28 |
| TW200740778A (en) | 2007-11-01 |
| WO2006136461A2 (en) | 2006-12-28 |
| WO2006136461A3 (en) | 2007-03-15 |
| IL188021A0 (en) | 2008-03-20 |
| CN101248066A (en) | 2008-08-20 |
| DE102005030292A1 (en) | 2007-01-11 |
| EA200702524A1 (en) | 2008-06-30 |
| AR054519A1 (en) | 2007-06-27 |
| MX2008000072A (en) | 2008-03-24 |
| PE20070125A1 (en) | 2007-02-14 |
| GT200600271A (en) | 2007-02-05 |
| DOP2006000148A (en) | 2007-07-15 |
| CR9598A (en) | 2008-04-09 |
| ZA200800690B (en) | 2009-09-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20160831 |