SK287645B6 - Tableta obsahujúca cetirizín a pseudoefedrín a jej použitie - Google Patents

Tableta obsahujúca cetirizín a pseudoefedrín a jej použitie Download PDF

Info

Publication number: SK287645B6
Authority: SK; Slovakia
Prior art keywords: cetirizine; pseudoephedrine; tablet; tablet according; segment
Prior art date: 2001-06-28

Application number

SK1550-2003A

Other languages

English (en)

Slovak (sk)

Other versions

SK15502003A3 (sk

Inventor

Domenico Fanara

Anthony Guichaux

Monique Berwaer

Michel Deleers

Original Assignee

Ucb, Farchim, S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-06-28

Filing date

2002-06-10

Publication date

2011-05-06

2002-06-10 Application filed by Ucb, Farchim, S.A. filed Critical Ucb, Farchim, S.A.

2004-05-04 Publication of SK15502003A3 publication Critical patent/SK15502003A3/sk

2011-05-06 Publication of SK287645B6 publication Critical patent/SK287645B6/sk

Links

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KWGRBVOPPLSCSI-WCBMZHEXSA-N pseudoephedrine Chemical compound CN[C@@H](C)[C@@H](O)C1=CC=CC=C1 KWGRBVOPPLSCSI-WCBMZHEXSA-N 0.000 title claims abstract description 101
KWGRBVOPPLSCSI-UHFFFAOYSA-N d-ephedrine Natural products CNC(C)C(O)C1=CC=CC=C1 KWGRBVOPPLSCSI-UHFFFAOYSA-N 0.000 title claims abstract description 100
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235000019447 hydroxyethyl cellulose Nutrition 0.000 description 1
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IQSHMXAZFHORGY-UHFFFAOYSA-N methyl prop-2-enoate;2-methylprop-2-enoic acid Chemical compound COC(=O)C=C.CC(=C)C(O)=O IQSHMXAZFHORGY-UHFFFAOYSA-N 0.000 description 1
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NGVDGCNFYWLIFO-UHFFFAOYSA-N pyridoxal 5'-phosphate Chemical compound CC1=NC=C(COP(O)(O)=O)C(C=O)=C1O NGVDGCNFYWLIFO-UHFFFAOYSA-N 0.000 description 1
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CVHZOJJKTDOEJC-UHFFFAOYSA-N saccharin Chemical compound C1=CC=C2C(=O)NS(=O)(=O)C2=C1 CVHZOJJKTDOEJC-UHFFFAOYSA-N 0.000 description 1
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ZLGIYFNHBLSMPS-ATJNOEHPSA-N shellac Chemical compound OCCCCCC(O)C(O)CCCCCCCC(O)=O.C1C23[C@H](C(O)=O)CCC2[C@](C)(CO)[C@@H]1C(C(O)=O)=C[C@@H]3O ZLGIYFNHBLSMPS-ATJNOEHPSA-N 0.000 description 1
235000013874 shellac Nutrition 0.000 description 1
239000011734 sodium Substances 0.000 description 1
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239000001509 sodium citrate Substances 0.000 description 1
NLJMYIDDQXHKNR-UHFFFAOYSA-K sodium citrate Chemical compound O.O.[Na+].[Na+].[Na+].[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O NLJMYIDDQXHKNR-UHFFFAOYSA-K 0.000 description 1
229920003109 sodium starch glycolate Polymers 0.000 description 1
239000008109 sodium starch glycolate Substances 0.000 description 1
229940079832 sodium starch glycolate Drugs 0.000 description 1
235000010339 sodium tetraborate Nutrition 0.000 description 1
239000011343 solid material Substances 0.000 description 1
239000000600 sorbitol Substances 0.000 description 1
238000013112 stability test Methods 0.000 description 1
239000007858 starting material Substances 0.000 description 1
239000008117 stearic acid Substances 0.000 description 1
239000007939 sustained release tablet Substances 0.000 description 1
239000003765 sweetening agent Substances 0.000 description 1
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239000000454 talc Substances 0.000 description 1
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229940124597 therapeutic agent Drugs 0.000 description 1
239000004408 titanium dioxide Substances 0.000 description 1
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239000000196 tragacanth Substances 0.000 description 1
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150000003626 triacylglycerols Chemical class 0.000 description 1
QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical class [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
BSVBQGMMJUBVOD-UHFFFAOYSA-N trisodium borate Chemical compound [Na+].[Na+].[Na+].[O-]B([O-])[O-] BSVBQGMMJUBVOD-UHFFFAOYSA-N 0.000 description 1
239000003981 vehicle Substances 0.000 description 1
125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 description 1
239000000341 volatile oil Substances 0.000 description 1
229940045860 white wax Drugs 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents

Landscapes

Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Pulmonology (AREA)
Otolaryngology (AREA)
Oncology (AREA)
Ophthalmology & Optometry (AREA)
Communicable Diseases (AREA)
Emergency Medicine (AREA)
Immunology (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medical Preparation Storing Or Oral Administration Devices (AREA)
Medicines Containing Plant Substances (AREA)

SK1550-2003A 2001-06-28 2002-06-10 Tableta obsahujúca cetirizín a pseudoefedrín a jej použitie SK287645B6 (sk)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US30125001P	2001-06-28	2001-06-28
EP01115807		2001-06-28
PCT/EP2002/006342 WO2003002098A1 (en)	2001-06-28	2002-06-10	Tablet comprising cetirizine and pseudoephedrine

Publications (2)

Publication Number	Publication Date
SK15502003A3 SK15502003A3 (sk)	2004-05-04
SK287645B6 true SK287645B6 (sk)	2011-05-06

Family

ID=56290291

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK1550-2003A SK287645B6 (sk)	2001-06-28	2002-06-10	Tableta obsahujúca cetirizín a pseudoefedrín a jej použitie

Country Status (22)

Country	Link
EP (1)	EP1404304B1 (zh)
JP (1)	JP4041460B2 (zh)
KR (1)	KR100926410B1 (zh)
CN (1)	CN100490809C (zh)
AT (1)	ATE432068T1 (zh)
AU (1)	AU2002345024B2 (zh)
BR (1)	BR0210650A (zh)
CA (1)	CA2451519C (zh)
CZ (1)	CZ20033454A3 (zh)
DK (1)	DK1404304T3 (zh)
EE (1)	EE05357B1 (zh)
ES (1)	ES2324769T3 (zh)
HU (1)	HU229803B1 (zh)
MX (1)	MXPA03010430A (zh)
NZ (1)	NZ530289A (zh)
PL (1)	PL206069B1 (zh)
PT (1)	PT1404304E (zh)
RO (1)	RO122476B1 (zh)
RU (1)	RU2286784C2 (zh)
SI (1)	SI1404304T1 (zh)
SK (1)	SK287645B6 (zh)
WO (1)	WO2003002098A1 (zh)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7014867B2 (en) *	2001-06-28	2006-03-21	Ucb Farchim Sa	Tablet comprising cetirizine and pseudoephedrine
KR100698400B1 (ko)	2004-04-14	2007-03-23	이은주	탈모증 및 전립선비대증 치료를 위한 약제학적 조성물
WO2007141743A2 (en) *	2006-06-06	2007-12-13	Ranbaxy Laboratories Limited	A tablet dosage form comprising cetirizine and pseudoephedrine
KR20090101362A (ko)	2006-12-26	2009-09-25	파마시클릭스, 인코포레이티드	병용 치료에 있어서 히스톤 디아세틸라제 억제제 이용 및 생체표지 감시 방법
US8439033B2 (en)	2007-10-09	2013-05-14	Microdose Therapeutx, Inc.	Inhalation device
MY187036A (en)	2010-01-05	2021-08-27	Microdose Therapeutx Inc	Inhalation device and method
KR101193495B1 (ko)	2010-02-01	2012-10-23	한미사이언스 주식회사	슈도에페드린 및 레보세티리진을 포함하는 경구용 복합 조성물
EP2799071B1 (en)	2010-06-16	2018-10-17	Inflammatory Response Research, Inc.	Levocetirizine and montelukast for the treatment of influenza and common cold
CN102302497A (zh) *	2011-05-18	2012-01-04	天圣制药集团股份有限公司	一种治疗过敏性鼻炎的制剂及其制备方法
KR20130009553A (ko)	2011-07-15	2013-01-23	한미약품 주식회사	몬테루카스트 또는 이의 약학적으로 허용가능한 염 및 레보세티리진 또는 이의 약학적으로 허용가능한 염을 함유하는 캡슐 제제
ES2627820T3 (es)	2011-09-13	2017-07-31	Pharmacyclics, Inc.	Formulaciones de inhibidor de histona desacetilasa en combinación con bendamustina y usos de las mismas
KR101372324B1 (ko) *	2012-02-09	2014-03-13	동국대학교 경주캠퍼스 산학협력단	알러지성 비염 치료를 위한 한방 치료제 및 슈도에페드린을 함유한 복합서방형의 약제학적 조성물
JP6441888B2 (ja)	2013-03-13	2018-12-19	インフラマトリー・レスポンス・リサーチ・インコーポレイテッド	自己免疫性障害の処置におけるレボセチリジン及びモンテルカストの使用
RU2672871C2 (ru)	2013-03-13	2018-11-20	Инфламматори Респонс Ресёрч, Инк.	Применение левоцетиризина и монтелукаста при лечении травматических повреждений
KR20160125283A (ko)	2013-03-13	2016-10-31	인플래머토리 리스폰스 리서치, 아이엔씨.	레보세티리진 및 몬테루카스트의 혈관염의 치료 용도
EP3193875B1 (en)	2014-09-15	2022-02-16	Inflammatory Response Research, Inc.	Levocetirizine and montelukast in the treatment of inflammation mediated conditions
WO2016140630A1 (en)	2015-03-05	2016-09-09	PHARMACTIVE ILAÇ SANAYI VE TlCARET A. Ş.	An effervescent composition comprising levocetirizine and pseudoephedrine
EP4099977A1 (en) *	2020-02-03	2022-12-14	Johnson & Johnson Consumer Inc.	A single layer chewable tablet comprising cetirizine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0811374A1 (en) *	1996-05-29	1997-12-10	Pfizer Inc.	Combination dosage form comprising cetirizine and pseudoephedrine
BE1011045A3 (fr) *	1997-03-14	1999-04-06	Ucb Sa	Compositions pharmaceutiques pour la liberation controlee de substances actives.
US6267986B1 (en) *	1999-09-24	2001-07-31	Ranbaxy Laboratories Limited	Process for the preparation of a controlled drug delivery system containing pseudoephedrine and a long acting antihistamine

2002
- 2002-06-10 HU HU0400386A patent/HU229803B1/hu unknown
- 2002-06-10 DK DK02743173T patent/DK1404304T3/da active
- 2002-06-10 JP JP2003508337A patent/JP4041460B2/ja not_active Expired - Fee Related
- 2002-06-10 EE EEP200400005A patent/EE05357B1/xx unknown
- 2002-06-10 CZ CZ20033454A patent/CZ20033454A3/cs unknown
- 2002-06-10 KR KR1020037017054A patent/KR100926410B1/ko active IP Right Grant
- 2002-06-10 SI SI200230844T patent/SI1404304T1/sl unknown
- 2002-06-10 ES ES02743173T patent/ES2324769T3/es not_active Expired - Lifetime
- 2002-06-10 AU AU2002345024A patent/AU2002345024B2/en not_active Ceased
- 2002-06-10 PT PT02743173T patent/PT1404304E/pt unknown
- 2002-06-10 WO PCT/EP2002/006342 patent/WO2003002098A1/en active Application Filing
- 2002-06-10 AT AT02743173T patent/ATE432068T1/de active
- 2002-06-10 SK SK1550-2003A patent/SK287645B6/sk not_active IP Right Cessation
- 2002-06-10 EP EP02743173A patent/EP1404304B1/en not_active Expired - Lifetime
- 2002-06-10 RO ROA200301062A patent/RO122476B1/ro unknown
- 2002-06-10 CA CA002451519A patent/CA2451519C/en not_active Expired - Lifetime
- 2002-06-10 RU RU2004101231/15A patent/RU2286784C2/ru active
- 2002-06-10 MX MXPA03010430A patent/MXPA03010430A/es active IP Right Grant
- 2002-06-10 BR BR0210650-7A patent/BR0210650A/pt not_active Application Discontinuation
- 2002-06-10 PL PL366800A patent/PL206069B1/pl unknown
- 2002-06-10 CN CNB02812975XA patent/CN100490809C/zh not_active Expired - Lifetime
- 2002-06-10 NZ NZ530289A patent/NZ530289A/en unknown

Also Published As

Publication number	Publication date
JP2004536829A (ja)	2004-12-09
HUP0400386A3 (en)	2006-02-28
NZ530289A (en)	2004-11-26
EE200400005A (et)	2004-02-16
CA2451519A1 (en)	2003-01-09
HUP0400386A2 (hu)	2004-08-30
PL206069B1 (pl)	2010-06-30
RO122476B1 (ro)	2009-07-30
EP1404304B1 (en)	2009-05-27
RU2286784C2 (ru)	2006-11-10
BR0210650A (pt)	2004-10-05
WO2003002098A1 (en)	2003-01-09
MXPA03010430A (es)	2004-12-06
KR20040007756A (ko)	2004-01-24
JP4041460B2 (ja)	2008-01-30
DK1404304T3 (da)	2009-07-13
PL366800A1 (en)	2005-02-07
CN1520285A (zh)	2004-08-11
KR100926410B1 (ko)	2009-11-12
EE05357B1 (et)	2010-12-15
CA2451519C (en)	2007-11-06
SK15502003A3 (sk)	2004-05-04
ATE432068T1 (de)	2009-06-15
HU229803B1 (en)	2014-07-28
PT1404304E (pt)	2009-06-26
CZ20033454A3 (cs)	2004-08-18
ES2324769T3 (es)	2009-08-14
SI1404304T1 (sl)	2009-10-31
CN100490809C (zh)	2009-05-27
AU2002345024B2 (en)	2006-09-07
EP1404304A1 (en)	2004-04-07
RU2004101231A (ru)	2005-04-20

Publication	Publication Date	Title
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