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SK281229B6 - 2,6-diaminopurínové deriváty, spôsob ich výroby, ich použitie a farmaceutické prostriedky s ich obsahom - Google Patents

2,6-diaminopurínové deriváty, spôsob ich výroby, ich použitie a farmaceutické prostriedky s ich obsahom Download PDF

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Publication number
SK281229B6
SK281229B6 SK918-95A SK91895A SK281229B6 SK 281229 B6 SK281229 B6 SK 281229B6 SK 91895 A SK91895 A SK 91895A SK 281229 B6 SK281229 B6 SK 281229B6
Authority
SK
Slovakia
Prior art keywords
amino
ethyl
diphenylethyl
deoxy
purin
Prior art date
Application number
SK918-95A
Other languages
English (en)
Slovak (sk)
Other versions
SK91895A3 (en
Inventor
Michael Gregson
Barry Edward Ayres
George Blanch Ewan
Frank Ellis
John Knight
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of SK91895A3 publication Critical patent/SK91895A3/sk
Publication of SK281229B6 publication Critical patent/SK281229B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • C07H19/167—Purine radicals with ribosyl as the saccharide radical

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Pulmonology (AREA)
  • Transplantation (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
SK918-95A 1993-01-20 1994-01-18 2,6-diaminopurínové deriváty, spôsob ich výroby, ich použitie a farmaceutické prostriedky s ich obsahom SK281229B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939301000A GB9301000D0 (en) 1993-01-20 1993-01-20 Chemical compounds
PCT/EP1994/000145 WO1994017090A1 (en) 1993-01-20 1994-01-18 2,6-diaminopurine derivatives

Publications (2)

Publication Number Publication Date
SK91895A3 SK91895A3 (en) 1996-04-03
SK281229B6 true SK281229B6 (sk) 2001-01-18

Family

ID=10728948

Family Applications (1)

Application Number Title Priority Date Filing Date
SK918-95A SK281229B6 (sk) 1993-01-20 1994-01-18 2,6-diaminopurínové deriváty, spôsob ich výroby, ich použitie a farmaceutické prostriedky s ich obsahom

Country Status (29)

Country Link
US (2) US5925624A (es)
EP (1) EP0680488B1 (es)
JP (1) JP3768232B2 (es)
KR (1) KR960700261A (es)
CN (1) CN1043997C (es)
AP (1) AP457A (es)
AT (1) ATE164849T1 (es)
AU (1) AU679714B2 (es)
CA (1) CA2153688A1 (es)
CZ (1) CZ187995A3 (es)
DE (1) DE69409503T2 (es)
DK (1) DK0680488T3 (es)
EC (1) ECSP941104A (es)
ES (1) ES2117249T3 (es)
FI (1) FI953489L (es)
GB (1) GB9301000D0 (es)
HU (1) HU211914A9 (es)
IL (1) IL108372A (es)
IS (1) IS4121A (es)
NO (1) NO305603B1 (es)
NZ (1) NZ259880A (es)
PE (1) PE54194A1 (es)
PL (1) PL309975A1 (es)
RU (1) RU2129561C1 (es)
SI (1) SI9400021A (es)
SK (1) SK281229B6 (es)
TW (1) TW267168B (es)
WO (1) WO1994017090A1 (es)
ZA (1) ZA94335B (es)

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CN1119440A (zh) 1996-03-27
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AP9400613A0 (en) 1994-01-31
DE69409503T2 (de) 1998-08-06
PL309975A1 (en) 1995-11-13
SK91895A3 (en) 1996-04-03
JPH08505864A (ja) 1996-06-25
TW267168B (es) 1996-01-01
AU679714B2 (en) 1997-07-10
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NZ259880A (en) 1996-11-26
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RU2129561C1 (ru) 1999-04-27
IS4121A (is) 1994-07-21
EP0680488A1 (en) 1995-11-08
CA2153688A1 (en) 1994-08-04
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ZA94335B (en) 1994-10-24
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HU211914A9 (en) 1996-01-29
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US5925624A (en) 1999-07-20
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US5889178A (en) 1999-03-30
IL108372A0 (en) 1994-04-12
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CN1043997C (zh) 1999-07-07
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FI953489A7 (fi) 1995-09-13
FI953489L (fi) 1995-09-13

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