SI2144506T1 - 3-substituirana-(1,2,3)-benzotriazinon spojine za povečanje glutamatnih sinaptičnih odgovorov - Google Patents

3-substituirana-(1,2,3)-benzotriazinon spojine za povečanje glutamatnih sinaptičnih odgovorov

Info

Publication number: SI2144506T1
Authority: SI; Slovenia
Prior art keywords: substituted; synaptic responses; glutamatergic synaptic; benzotriazinone; compound
Prior art date: 2007-01-03

Application number

SI200730806T

Other languages

English (en)

Inventor

Alexis Cordi

Gary Rogers

Rudolf Mueller

Original Assignee

Servier Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-01-03

Filing date

2007-12-28

Publication date

2012-01-31

2007-12-28 Application filed by Servier Lab filed Critical Servier Lab

2012-01-31 Publication of SI2144506T1 publication Critical patent/SI2144506T1/sl

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Psychiatry (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

SI200730806T 2007-01-03 2007-12-28 3-substituirana-(1,2,3)-benzotriazinon spojine za povečanje glutamatnih sinaptičnih odgovorov SI2144506T1 (sl)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US87850307P	2007-01-03	2007-01-03
US92143307P	2007-04-02	2007-04-02
EP07868093A EP2144506B1 (en)	2007-01-03	2007-12-28	3-substituted-[1,2,3]-benzotriazinone compound for enhancing glutamatergic synaptic responses
PCT/US2007/026416 WO2008085506A1 (en)	2007-01-03	2007-12-28	3-substituted-[1,2,3]-benzotriazinone compound for enhancing glutamatergic synaptic responses

Publications (1)

Publication Number	Publication Date
SI2144506T1 true SI2144506T1 (sl)	2012-01-31

Family

ID=39608956

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SI200730806T SI2144506T1 (sl)	2007-01-03	2007-12-28	3-substituirana-(1,2,3)-benzotriazinon spojine za povečanje glutamatnih sinaptičnih odgovorov

Country Status (38)

Country	Link
US (1)	US8173644B2 (sl)
EP (1)	EP2144506B1 (sl)
JP (1)	JP5139446B2 (sl)
CN (1)	CN101616592B (sl)
AP (1)	AP2502A (sl)
AR (1)	AR064740A1 (sl)
AT (1)	ATE527269T1 (sl)
AU (1)	AU2007342365B2 (sl)
BR (1)	BRPI0720749A2 (sl)
CA (1)	CA2674460C (sl)
CR (1)	CR10906A (sl)
CU (1)	CU23804B7 (sl)
CY (1)	CY1112493T1 (sl)
DK (1)	DK2144506T3 (sl)
EA (1)	EA017437B1 (sl)
EC (1)	ECSP099499A (sl)
ES (1)	ES2374995T3 (sl)
GE (1)	GEP20125438B (sl)
GT (1)	GT200900189A (sl)
HK (1)	HK1140105A1 (sl)
HN (1)	HN2009001268A (sl)
HR (1)	HRP20110970T1 (sl)
IL (1)	IL199651A (sl)
MA (1)	MA31160B1 (sl)
ME (1)	ME00819B (sl)
MX (1)	MX2009007242A (sl)
MY (1)	MY154877A (sl)
NI (1)	NI200900131A (sl)
NZ (1)	NZ578293A (sl)
PL (1)	PL2144506T3 (sl)
PT (1)	PT2144506E (sl)
RS (1)	RS52108B (sl)
SG (1)	SG163545A1 (sl)
SI (1)	SI2144506T1 (sl)
SV (1)	SV2009003322A (sl)
TN (1)	TN2009000277A1 (sl)
WO (1)	WO2008085506A1 (sl)
ZA (1)	ZA200904826B (sl)

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KR20090098999A (ko) *	2007-01-03	2009-09-18	코텍스 파마슈티칼스, 인크.	글루타메이트에 의한 시냅스 반응을 향상시키기 위한 3-치환된-[1,2,3]벤조트리아지논 화합물
TW200911768A (en)	2007-05-17	2009-03-16	Cortex Pharma Inc	Di-substituted amides for enhancing glutamatergic synaptic responses
US8168632B2 (en)	2007-08-10	2012-05-01	Cortex Pharmaceuticals, Inc.	Bicyclic amide derivatives for the treatment of respiratory disorders
BRPI0823262A2 (pt)	2007-08-10	2013-09-24	Cortex Pharma Inc	mÉtodo de tratamento de depressço respiratària e uso de um composto na fabricaÇço de um medicamento para o tratamento de depressço respiratària
US20110257186A1 (en) *	2010-04-15	2011-10-20	Staubli Ursula V	Compositions and methods for treating visual disorders
US9242938B2 (en)	2011-11-22	2016-01-26	Beijing Medisan Technology Co., Ltd	Glycine reuptake inhibitor and use thereof
FR3019464B1 (fr)	2014-04-07	2016-05-06	Servier Lab	Nouvelle association entre le 8-cyclopropyl-3-[2-(3-fluorophenyl)ethyl]-7,8-dihydro-3h-[1,3]oxazino[6,5-g] [1,2,3]benzotriazine-4,9-dione et un inhibiteur de l'acetylcholinesterase et les compositions pharmaceutiques qui la contiennent
FR3034019B1 (fr)	2015-03-26	2017-03-17	Servier Lab	Nouvelle association entre le 8-cyclopropyl-3-[2-(3-fluorophenyl)ethyl]-7,8-dihydro-3h-[1,3]oxazino[6,5-g] [1,2,3]benzotriazine-4,9-dione et un antidepresseur et les compositions pharmaceutiques qui la contiennent
US9878989B2 (en)	2015-06-26	2018-01-30	Takeda Pharmaceutical Company Limited	Heterocyclic compound
CN106226509B (zh) *	2016-08-12	2019-09-06	中国人民解放军第四军医大学	一种在小鼠前扣带回皮层诱发dse现象的方法

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WO1998011892A1 (en)	1996-09-17	1998-03-26	The Regents Of The University Of California	Positive ampa receptor modulation to enhance brain neurotrophic factor expression
US6110935A (en) *	1997-02-13	2000-08-29	The Regents Of The University Of California	Benzofurazan compounds for enhancing glutamatergic synaptic responses
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PL342843A1 (en)	1998-02-18	2001-07-16	Neurosearch As	Novel compounds and their use as positive ampa receptor modulators
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TW200911768A (en) *	2007-05-17	2009-03-16	Cortex Pharma Inc	Di-substituted amides for enhancing glutamatergic synaptic responses
BRPI0823262A2 (pt)	2007-08-10	2013-09-24	Cortex Pharma Inc	mÉtodo de tratamento de depressço respiratària e uso de um composto na fabricaÇço de um medicamento para o tratamento de depressço respiratària
US20100267728A1 (en)	2007-09-20	2010-10-21	Cortex Pharmaceuticals, Inc.	3-substituted-1,2,3-triazin-4-one's and 3 substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses

2007
- 2007-12-28 WO PCT/US2007/026416 patent/WO2008085506A1/en active Application Filing
- 2007-12-28 US US12/448,784 patent/US8173644B2/en not_active Expired - Fee Related
- 2007-12-28 DK DK07868093.1T patent/DK2144506T3/da active
- 2007-12-28 AU AU2007342365A patent/AU2007342365B2/en not_active Ceased
- 2007-12-28 ZA ZA200904826A patent/ZA200904826B/xx unknown
- 2007-12-28 AT AT07868093T patent/ATE527269T1/de active
- 2007-12-28 CN CN2007800508375A patent/CN101616592B/zh not_active Expired - Fee Related
- 2007-12-28 SI SI200730806T patent/SI2144506T1/sl unknown
- 2007-12-28 JP JP2009544857A patent/JP5139446B2/ja not_active Expired - Fee Related
- 2007-12-28 PL PL07868093T patent/PL2144506T3/pl unknown
- 2007-12-28 EP EP07868093A patent/EP2144506B1/en active Active
- 2007-12-28 MX MX2009007242A patent/MX2009007242A/es active IP Right Grant
- 2007-12-28 AP AP2009004931A patent/AP2502A/xx active
- 2007-12-28 PT PT07868093T patent/PT2144506E/pt unknown
- 2007-12-28 EA EA200900925A patent/EA017437B1/ru not_active IP Right Cessation
- 2007-12-28 GE GEAP200711384A patent/GEP20125438B/en unknown
- 2007-12-28 ES ES07868093T patent/ES2374995T3/es active Active
- 2007-12-28 RS RS20110587A patent/RS52108B/en unknown
- 2007-12-28 MY MYPI20092796A patent/MY154877A/en unknown
- 2007-12-28 BR BRPI0720749-2A patent/BRPI0720749A2/pt not_active Application Discontinuation
- 2007-12-28 ME MEP-2009-238A patent/ME00819B/me unknown
- 2007-12-28 NZ NZ578293A patent/NZ578293A/en not_active IP Right Cessation
- 2007-12-28 SG SG201004695-1A patent/SG163545A1/en unknown
- 2007-12-28 CA CA2674460A patent/CA2674460C/en not_active Expired - Fee Related
2008
- 2008-01-03 AR ARP080100022A patent/AR064740A1/es not_active Application Discontinuation
2009
- 2009-06-30 TN TNP2009000277A patent/TN2009000277A1/fr unknown
- 2009-07-01 NI NI200900131A patent/NI200900131A/es unknown
- 2009-07-02 GT GT200900189A patent/GT200900189A/es unknown
- 2009-07-02 CR CR10906A patent/CR10906A/es not_active Application Discontinuation
- 2009-07-02 SV SV2009003322A patent/SV2009003322A/es unknown
- 2009-07-02 IL IL199651A patent/IL199651A/en active IP Right Grant
- 2009-07-03 HN HN2009001268A patent/HN2009001268A/es unknown
- 2009-07-03 CU CU20090117A patent/CU23804B7/es active IP Right Grant
- 2009-07-07 EC EC2009009499A patent/ECSP099499A/es unknown
- 2009-07-31 MA MA32135A patent/MA31160B1/fr unknown
2010
- 2010-06-29 HK HK10106349.3A patent/HK1140105A1/xx not_active IP Right Cessation
2011
- 2011-12-23 HR HR20110970T patent/HRP20110970T1/hr unknown
- 2011-12-28 CY CY20111101287T patent/CY1112493T1/el unknown

Also Published As

Publication number	Publication date
CR10906A (es)	2009-10-23
CU20090117A7 (es)	2011-10-05
CA2674460A1 (en)	2008-07-17
US8173644B2 (en)	2012-05-08
EP2144506A1 (en)	2010-01-20
BRPI0720749A2 (pt)	2014-01-14
HN2009001268A (es)	2011-12-27
HK1140105A1 (en)	2010-10-08
US20100137295A1 (en)	2010-06-03
GT200900189A (es)	2011-08-02
JP2010514838A (ja)	2010-05-06
AP2502A (en)	2012-10-23
PL2144506T3 (pl)	2012-04-30
GEP20125438B (en)	2012-03-26
SG163545A1 (en)	2010-08-30
CN101616592B (zh)	2013-06-05
EA200900925A1 (ru)	2009-12-30
NI200900131A (es)	2010-03-11
CA2674460C (en)	2014-07-15
MA31160B1 (fr)	2010-02-01
CN101616592A (zh)	2009-12-30
EA017437B1 (ru)	2012-12-28
NZ578293A (en)	2012-01-12
EP2144506A4 (en)	2010-05-05
AP2009004931A0 (en)	2009-08-31
HRP20110970T1 (hr)	2012-01-31
RS52108B (en)	2012-08-31
MX2009007242A (es)	2009-09-02
AU2007342365B2 (en)	2012-11-15
SV2009003322A (es)	2010-02-05
ES2374995T3 (es)	2012-02-23
DK2144506T3 (da)	2012-03-05
WO2008085506A1 (en)	2008-07-17
ME00819B (me)	2012-03-20
AR064740A1 (es)	2009-04-22
IL199651A (en)	2015-08-31
JP5139446B2 (ja)	2013-02-06
ECSP099499A (es)	2009-10-30
TN2009000277A1 (en)	2010-10-18
IL199651A0 (en)	2010-04-15
AU2007342365A1 (en)	2008-07-17
ATE527269T1 (de)	2011-10-15
EP2144506B1 (en)	2011-10-05
ZA200904826B (en)	2010-09-29
CY1112493T1 (el)	2015-12-09
CU23804B7 (es)	2012-03-15
MY154877A (en)	2015-08-14
PT2144506E (pt)	2011-12-21

Publication	Publication Date	Title
HK1140105A1 (en)	2010-10-08	3-substituted-[1,2,3]-benzotriazinone compound for enhancing glutamatergic synaptic responses
ZA200905065B (en)	2010-04-28	3-substituted-[1,2,3]benzotriazinone compounds for enhancing glutamatergic synaptic responses
BRPI0815717A2 (pt)	2015-02-10	Compostos de imidazopirazina.
IL201973A0 (en)	2010-06-16	3,3-spiroindolinone derivatives
BRPI0816970A2 (pt)	2015-03-24	1,3-dissubstituídas-4-fenil-1h-piridin-2-onas
IL225694A0 (en)	2013-06-27	Compounds 6,5- dihydro-h1-pyridine-2-one
EP2361902A4 (en)	2012-04-25	4,6-DIAMINONICOTINSÄUREAMIDVERBINDUNG
ZA201001797B (en)	2010-11-24	1,1,1-trifluoro-2-hydroxy-3-phenylpropane derivatives
HK1147677A1 (en)	2011-08-19	Bicyclic amides for enhancing glutamatergic synaptic responses
BRPI0815059A2 (pt)	2015-02-10	Derivado de 1,3-di-hidroisoindol
PL378889A1 (pl)	2007-08-06	Raportowanie wyników wyszukiwania
BRPI0916395A2 (pt)	2016-02-16	compostos de 1,6-di-hidro-2h-3-oxa-6-aza-as-indaceno
EP2202231A4 (en)	2011-09-28	2,3-DIHYDROIMINOISOINDOLE DERIVATIVE
BRPI0816542A2 (pt)	2015-10-13	receptáculo para, particulamente, produtos agrícolas.
HK1161684A1 (en)	2012-08-03	5,6-dihydro-1h-pyridin-2-one compounds 56- -1h--2-
BRPI0818848A2 (pt)	2015-04-14	Compostos de 2,3-di-idro-benzofurano
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AU2007901207A0 (en)	2007-03-22	Animal contianment arrangement
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AU2007903661A0 (en)	2007-07-19	Chain
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ITBO20050004U1 (it)	2006-07-15	Raccordo per tettarella
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