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SG11202106166TA - Peptide binder - Google Patents

Peptide binder

Info

Publication number
SG11202106166TA
SG11202106166TA SG11202106166TA SG11202106166TA SG11202106166TA SG 11202106166T A SG11202106166T A SG 11202106166TA SG 11202106166T A SG11202106166T A SG 11202106166TA SG 11202106166T A SG11202106166T A SG 11202106166TA SG 11202106166T A SG11202106166T A SG 11202106166TA
Authority
SG
Singapore
Prior art keywords
peptide binder
peptide
binder
Prior art date
Application number
SG11202106166TA
Inventor
Perez Maria Mendez
Nils Rackelmann
Stefan Guessregen
Martin Will
Thomas Boehme
Garea Ana Villar
Michael Podeschwa
Laurent Bialy
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=68806785&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11202106166T(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of SG11202106166TA publication Critical patent/SG11202106166TA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/62—Insulins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/28—Insulins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • A61K47/64—Drug-peptide, drug-protein or drug-polyamino acid conjugates, i.e. the modifying agent being a peptide, protein or polyamino acid which is covalently bonded or complexed to a therapeutically active agent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Molecular Biology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SG11202106166TA 2018-12-11 2019-12-10 Peptide binder SG11202106166TA (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP18306658 2018-12-11
EP18306657 2018-12-11
EP18306659 2018-12-11
PCT/EP2019/084433 WO2020120479A1 (en) 2018-12-11 2019-12-10 Peptide binder

Publications (1)

Publication Number Publication Date
SG11202106166TA true SG11202106166TA (en) 2021-07-29

Family

ID=68806785

Family Applications (3)

Application Number Title Priority Date Filing Date
SG11202106167XA SG11202106167XA (en) 2018-12-11 2019-12-10 Insulin conjugates
SG11202106166TA SG11202106166TA (en) 2018-12-11 2019-12-10 Peptide binder
SG11202106168VA SG11202106168VA (en) 2018-12-11 2019-12-10 Insulin analogs having reduced insulin receptor binding affinity

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG11202106167XA SG11202106167XA (en) 2018-12-11 2019-12-10 Insulin conjugates

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG11202106168VA SG11202106168VA (en) 2018-12-11 2019-12-10 Insulin analogs having reduced insulin receptor binding affinity

Country Status (15)

Country Link
US (3) US11098102B2 (en)
EP (3) EP3894391A1 (en)
JP (3) JP2022513775A (en)
KR (3) KR20210102347A (en)
CN (3) CN113423691A (en)
AU (3) AU2019398579A1 (en)
BR (3) BR112021011156A2 (en)
CA (3) CA3122637A1 (en)
CO (1) CO2021007453A2 (en)
IL (3) IL283800A (en)
MX (3) MX2021006972A (en)
PH (1) PH12021551339A1 (en)
SG (3) SG11202106167XA (en)
TW (3) TW202039437A (en)
WO (3) WO2020120479A1 (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
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KR20210102347A (en) 2018-12-11 2021-08-19 사노피 Insulin analogues with reduced insulin receptor binding affinity
CN112876388B (en) * 2021-01-14 2023-03-31 山东大学 GPR120 agonist and preparation method and application thereof
CN116162147B (en) * 2021-11-24 2023-10-03 成都奥达生物科技有限公司 Long-acting insulin analogue
CN114230451A (en) * 2021-12-29 2022-03-25 上海药坦药物研究开发有限公司 Preparation method of halogenated acid compounds
JP2025508329A (en) * 2022-01-26 2025-03-26 サノフイ Insulin conjugates
CN119403824A (en) 2022-06-23 2025-02-07 赛诺菲 Single-chain insulin and its Fc conjugate
CN115947822B (en) * 2022-07-04 2023-08-18 北京惠之衡生物科技有限公司 Long-acting acylated insulin derivative, and pharmaceutical composition and application thereof
WO2024051787A1 (en) * 2022-09-09 2024-03-14 北京惠之衡生物科技有限公司 Long-acting acylated insulin derivative and use thereof

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Also Published As

Publication number Publication date
KR20210102346A (en) 2021-08-19
US12195510B2 (en) 2025-01-14
WO2020120479A1 (en) 2020-06-18
CA3122637A1 (en) 2020-06-18
CN113395982A (en) 2021-09-14
AU2019398579A1 (en) 2021-07-29
US20250206798A1 (en) 2025-06-26
US11098102B2 (en) 2021-08-24
MX2021006972A (en) 2021-08-16
CN113423691A (en) 2021-09-21
JP2022513775A (en) 2022-02-09
CO2021007453A2 (en) 2021-06-21
IL283800A (en) 2021-07-29
WO2020120463A1 (en) 2020-06-18
CA3122632A1 (en) 2020-06-18
WO2020120477A1 (en) 2020-06-18
IL283801A (en) 2021-07-29
KR20210102345A (en) 2021-08-19
SG11202106168VA (en) 2021-07-29
AU2019398658A1 (en) 2021-07-29
EP3893934A1 (en) 2021-10-20
KR20210102347A (en) 2021-08-19
JP2022513776A (en) 2022-02-09
US20220048968A1 (en) 2022-02-17
BR112021011099A2 (en) 2021-10-26
PH12021551339A1 (en) 2021-11-29
EP3894435A1 (en) 2021-10-20
BR112021011156A2 (en) 2021-10-26
BR112021011050A2 (en) 2021-08-31
TW202039539A (en) 2020-11-01
IL283803A (en) 2021-07-29
TW202039438A (en) 2020-11-01
JP2022511567A (en) 2022-01-31
MX2021006970A (en) 2021-07-15
CA3122636A1 (en) 2020-06-18
CN113396157A (en) 2021-09-14
US20200181223A1 (en) 2020-06-11
EP3894391A1 (en) 2021-10-20
SG11202106167XA (en) 2021-07-29
TW202039437A (en) 2020-11-01
AU2019398402A1 (en) 2021-07-29
MX2021006969A (en) 2021-07-15

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