SE376420B - - Google Patents

Info

Publication number: SE376420B
Authority: SE; Sweden

Application number

SE7102758A

Inventor

T J Schwan

S E Burrous

J L Butterfield

Original Assignee

Norwich Pharma Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1970-03-05

Filing date

1971-03-04

Publication date

1975-05-26

1971-03-04 Application filed by Norwich Pharma Co filed Critical Norwich Pharma Co

1975-05-26 Publication of SE376420B publication Critical patent/SE376420B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/10—Oxygen or sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/34—One oxygen atom
- C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Joining Of Building Structures In Genera (AREA)
Indole Compounds (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)

SE7102758A 1970-03-05 1971-03-04 SE376420B (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US1698270A	1970-03-05	1970-03-05

Publications (1)

Publication Number	Publication Date
SE376420B true SE376420B (de)	1975-05-26

Family

ID=21780073

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7102758A SE376420B (de)	1970-03-05	1971-03-04

Country Status (14)

Country	Link
US (1)	US3681349A (de)
AT (1)	AT305288B (de)
BE (1)	BE763745A (de)
CH (1)	CH555343A (de)
DE (1)	DE2110445C3 (de)
DK (1)	DK127427B (de)
ES (1)	ES388780A1 (de)
FR (1)	FR2085673B1 (de)
GB (1)	GB1294626A (de)
IL (1)	IL36189A0 (de)
NL (1)	NL7102519A (de)
NO (1)	NO130728C (de)
SE (1)	SE376420B (de)
ZA (1)	ZA71928B (de)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL39003A (en) *	1971-03-25	1975-02-10	Morton Norwich Products Inc	1-(substituted benzyl)tetrahydro-2-(1h)-pyrimidones and their preparation
US3957785A (en) *	1971-12-02	1976-05-18	Societa' Farmaceutici Italia S.P.A.	Bβ-Pyrimidino-aminomethyl-10α-ergoline and 10α-methoxyergoline derivatives
US3956325A (en) *	1974-01-21	1976-05-11	Smithkline Corporation	5-Heterocyclic-1,2,3,6-tetrahydro-4(5H) pyrimidinone
US4003900A (en) *	1976-03-11	1977-01-18	Morton-Norwich Products, Inc.	1-Benzyl-5-chloro-2-(1H)-pyrimidone
US4002627A (en) *	1976-03-26	1977-01-11	Morton-Norwich Products, Inc.	1-Benzyl-3-methyl-3,4,5,6-tetrahydro-2(1H) pyrimidone
US4052399A (en) *	1976-09-13	1977-10-04	Morton-Norwich Products, Inc.	1-[2-(Hexahydro-1H-azepino)ethyl]-2(1H)pyrimidone dihydrochloride
US4052400A (en) *	1976-10-29	1977-10-04	Morton-Norwich Products, Inc.	Hypertensive 1-substituted 2(1h)-pyrimidones
US8835426B2 (en) *	2007-02-26	2014-09-16	Vitae Pharmaceuticals, Inc.	Cyclic urea and carbamate inhibitors of 11β-hydroxysteroid dehydrogenase 1
EP2183228B1 (de) *	2007-07-26	2014-08-20	Vitae Pharmaceuticals, Inc.	ZYKLISCHE 11ß-HYDROXYSTEROID-DEHYDROGENASE-1-HEMMER
AR069207A1 (es) *	2007-11-07	2010-01-06	Vitae Pharmaceuticals Inc	Ureas ciclicas como inhibidores de la 11 beta - hidroxi-esteroide deshidrogenasa 1
CA2708303A1 (en)	2007-12-11	2009-06-18	Vitae Pharmaceuticals, Inc.	Cyclic urea inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1
TW200934490A (en) *	2008-01-07	2009-08-16	Vitae Pharmaceuticals Inc	Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
WO2009094169A1 (en)	2008-01-24	2009-07-30	Vitae Pharmaceuticals, Inc.	Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1
CA2714532A1 (en) *	2008-02-11	2009-08-20	Vitae Pharmaceuticals, Inc.	1,3-oxazepan-2-one and 1,3-diazepan-2-one inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1
CA2715290A1 (en) *	2008-02-15	2009-08-20	Vitae Pharmaceuticals, Inc.	Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
JP5538356B2 (ja) *	2008-03-18	2014-07-02	ヴァイティーファーマシューティカルズ，インコーポレイテッド	１１β−ヒドロキシステロイドデヒドロゲナーゼ１型の阻害剤
TW200946520A (en) *	2008-05-01	2009-11-16	Vitae Pharmaceuticals Inc	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
CA2723039A1 (en) *	2008-05-01	2009-11-05	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2291370B1 (de) *	2008-05-01	2013-11-27	Vitae Pharmaceuticals, Inc.	Cyclische inhibitoren von 11beta-hydroxysteroiddehydrogenase 1
WO2009134384A1 (en) *	2008-05-01	2009-11-05	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
KR20110050459A (ko) *	2008-07-25	2011-05-13	비타이 파마슈티컬즈, 인코포레이티드	11베타-하이드록시스테로이드 탈수소효소 1의 고리형 억제제
WO2010127237A2 (en) *	2009-04-30	2010-11-04	Boehringer Ingelheim International Gmbh	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
CN102105454A (zh)	2008-07-25	2011-06-22	贝林格尔.英格海姆国际有限公司	合成1型11β-羟基类固醇脱氢酶的抑制剂
WO2010010157A2 (en)	2008-07-25	2010-01-28	Boehringer Ingelheim International Gmbh	INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1
EP2393807B1 (de)	2009-02-04	2013-08-14	Boehringer Ingelheim International GmbH	Zyklische 11beta-hydroxysteroid-dehydrogenase-1-hemmer
TW201039034A (en) *	2009-04-27	2010-11-01	Chunghwa Picture Tubes Ltd	Pixel structure and the method of forming the same
MA33216B1 (fr)	2009-04-30	2012-04-02	Boehringer Ingelheim Int	Inhibiteurs cycliques de la 11béta-hydroxysteroïde déshydrogénase 1
JP5656986B2 (ja)	2009-06-11	2015-01-21	ヴァイティーファーマシューティカルズ，インコーポレイテッド	１，３−オキサジナン−２−オン構造に基づく１１β−ヒドロキシステロイドデヒドロゲナーゼ１の環状阻害剤
WO2011002910A1 (en)	2009-07-01	2011-01-06	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8552212B2 (en)	2009-11-05	2013-10-08	Boehringer Ingelheim International Gmbh	Chiral phosphorus ligands
AR078887A1 (es) *	2009-11-06	2011-12-07	Boehringer Ingelheim Int	Derivados arilo y heteroarilcarbonilo de hexahidroindenopiridina y octahidrobenzoquinolina y composiciones farmaceuticas que los contienen.
US8648192B2 (en)	2010-05-26	2014-02-11	Boehringer Ingelheim International Gmbh	2-oxo-1,2-dihydropyridin-4-ylboronic acid derivatives
US8933072B2 (en)	2010-06-16	2015-01-13	Vitae Pharmaceuticals, Inc.	Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
JP5813106B2 (ja)	2010-06-25	2015-11-17	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	代謝障害の処置のための１１−β−ＨＳＤ１のインヒビターとしてのアザスピロヘキサノン
KR20130137628A (ko)	2010-11-02	2013-12-17	베링거 인겔하임 인터내셔날 게엠베하	대사 장애를 치료하기 위한 약제학적 병용물
TWI537258B (zh)	2010-11-05	2016-06-11	百靈佳殷格翰國際股份有限公司	六氫茚并吡啶及八氫苯并喹啉之芳基－及雜環芳基羰基衍生物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE562987A (de) *	1956-12-05
DE1121617B (de) *	1959-05-26	1962-01-11	Huels Chemische Werke Ag	Verfahren zur Herstellung von Tetrahydropyrimidin-2-onderivaten
DE1545601A1 (de) *	1965-07-22	1969-08-07	Basf Ag	Verfahren zur Herstellung von Hexahydro-pyrimidinderivaten
DE1670368A1 (de) *	1966-07-16	1970-11-05	Cassella Farbwerke Mainkur Ag	Verfahren zur Herstellung aralkylsubstituierter Lactame und Cyclischer Harnstoffe
DE1670241A1 (de) *	1967-07-01	1971-01-28	Basf Ag	Verfahren zur Herstellung von 2-Oxohexahydropyrimidinen

1970
- 1970-03-05 US US16982A patent/US3681349A/en not_active Expired - Lifetime
1971
- 1971-02-15 ZA ZA710928A patent/ZA71928B/xx unknown
- 1971-02-15 IL IL36189A patent/IL36189A0/xx unknown
- 1971-02-25 NL NL7102519A patent/NL7102519A/xx unknown
- 1971-03-02 ES ES388780A patent/ES388780A1/es not_active Expired
- 1971-03-03 BE BE763745A patent/BE763745A/xx unknown
- 1971-03-03 NO NO802/71A patent/NO130728C/no unknown
- 1971-03-04 SE SE7102758A patent/SE376420B/xx unknown
- 1971-03-04 DK DK100371AA patent/DK127427B/da unknown
- 1971-03-04 FR FR7107502A patent/FR2085673B1/fr not_active Expired
- 1971-03-04 DE DE2110445A patent/DE2110445C3/de not_active Expired
- 1971-03-05 CH CH325271A patent/CH555343A/de not_active IP Right Cessation
- 1971-03-05 AT AT194271A patent/AT305288B/de active
- 1971-04-19 GB GB22882/71A patent/GB1294626A/en not_active Expired

Also Published As

Publication number	Publication date
DK127427B (da)	1973-11-05
BE763745A (fr)	1971-09-03
ES388780A1 (es)	1975-03-01
NL7102519A (de)	1971-09-07
FR2085673B1 (de)	1974-09-06
CH555343A (de)	1974-10-31
DE2110445C3 (de)	1975-05-28
IL36189A0 (en)	1971-04-28
FR2085673A1 (de)	1971-12-31
ZA71928B (en)	1972-09-27
US3681349A (en)	1972-08-01
DE2110445B2 (de)	1974-10-10
GB1294626A (en)	1972-11-01
DE2110445A1 (de)	1971-11-04
AT305288B (de)	1973-02-26
NO130728C (de)	1975-01-29
NO130728B (de)	1974-10-21

Publication	Publication Date	Title
FR2085673B1 (de)	1974-09-06
AU1473870A (de)	1971-11-11
AU2044470A (de)	1972-03-30
AU1336970A (de)	1971-10-07
AU2130570A (de)	1972-04-27
AU1716970A (de)	1972-01-06
AU1833270A (de)	1972-02-10
AU1326870A (de)	1971-10-28
AU1517670A (de)	1971-11-18
AU2085370A (de)	1972-04-13
AU2017870A (de)	1972-03-23
AU2130770A (de)	1972-04-27
AU1328670A (de)	1971-10-07
AU1974970A (de)	1972-03-16
AU1689770A (de)	1972-01-06
AU1789870A (de)	1972-01-27
AU1603270A (de)	1971-12-09
AU1591370A (de)	1971-12-09
AU1581370A (de)	1971-12-09
AU1247570A (de)	1971-09-16
AU2115870A (de)	1972-04-20
AU1918570A (de)	1972-03-02
AU2061170A (de)	1972-04-13
AU1277070A (de)	1971-09-23
AU1881070A (de)	1972-02-17